AU3119989A - Amino acid derivatives - Google Patents

Amino acid derivatives

Info

Publication number
AU3119989A
AU3119989A AU31199/89A AU3119989A AU3119989A AU 3119989 A AU3119989 A AU 3119989A AU 31199/89 A AU31199/89 A AU 31199/89A AU 3119989 A AU3119989 A AU 3119989A AU 3119989 A AU3119989 A AU 3119989A
Authority
AU
Australia
Prior art keywords
amino acid
acid derivatives
derivatives
amino
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU31199/89A
Other versions
AU626835B2 (en
Inventor
Joachim Dr. Gante
Klaus-Otto Dr Minck
Peter Dr. Raddatz
Claus J. Dr. Schmitges
Johannes Dr. Sombroek
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH
Publication of AU3119989A publication Critical patent/AU3119989A/en
Application granted granted Critical
Publication of AU626835B2 publication Critical patent/AU626835B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0207—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0227—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU31199/89A 1988-03-18 1989-03-10 Amino acid derivatives Ceased AU626835B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3809145 1988-03-18
DE3809145A DE3809145A1 (en) 1988-03-18 1988-03-18 AMINOSAEUREDERIVATE

Publications (2)

Publication Number Publication Date
AU3119989A true AU3119989A (en) 1989-09-21
AU626835B2 AU626835B2 (en) 1992-08-13

Family

ID=6350109

Family Applications (1)

Application Number Title Priority Date Filing Date
AU31199/89A Ceased AU626835B2 (en) 1988-03-18 1989-03-10 Amino acid derivatives

Country Status (7)

Country Link
EP (1) EP0342325A3 (en)
JP (1) JPH024749A (en)
KR (1) KR890014580A (en)
AU (1) AU626835B2 (en)
DE (1) DE3809145A1 (en)
HU (1) HU203116B (en)
ZA (1) ZA892059B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU610588B2 (en) * 1987-05-26 1991-05-23 Merck Patent Gesellschaft Mit Beschrankter Haftung Amino acid derivatives
US6797820B2 (en) 1999-12-17 2004-09-28 Vicuron Pharmaceuticals Inc. Succinate compounds, compositions and methods of use and preparation

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07501056A (en) * 1991-11-01 1995-02-02 スミスクライン・ビーチャム・コーポレイション Guanidine-containing HIV protease inhibitor
JP4679981B2 (en) * 2005-07-01 2011-05-11 エヌ・イーケムキャット株式会社 Method for deprotecting 9-fluorenylmethoxycarbonyl group

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4727060A (en) * 1984-11-13 1988-02-23 Ciba-Geigy Corporation Novel 5-amino-4-hydroxyvaleryl derivatives
ES2066755T3 (en) * 1986-06-10 1995-03-16 Merck Patent Gmbh DERIVATIVES OF RENINE INHIBITING AMINO ACIDS.
DE3789101T2 (en) * 1986-12-19 1994-07-21 Sankyo Co Renin inhibiting oligopeptides, their preparation and their application.

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU610588B2 (en) * 1987-05-26 1991-05-23 Merck Patent Gesellschaft Mit Beschrankter Haftung Amino acid derivatives
US6797820B2 (en) 1999-12-17 2004-09-28 Vicuron Pharmaceuticals Inc. Succinate compounds, compositions and methods of use and preparation

Also Published As

Publication number Publication date
JPH024749A (en) 1990-01-09
KR890014580A (en) 1989-10-24
EP0342325A2 (en) 1989-11-23
AU626835B2 (en) 1992-08-13
HU203116B (en) 1991-05-28
EP0342325A3 (en) 1991-01-16
ZA892059B (en) 1989-11-29
HUT53121A (en) 1990-09-28
DE3809145A1 (en) 1989-09-28

Similar Documents

Publication Publication Date Title
AU3613089A (en) Amino acid derivatives
AU3079789A (en) Amino acid derivatives
AU634526B2 (en) Amino acid derivatives
AU646640B2 (en) Amino acid derivatives
AU5058290A (en) Amino acid derivatives
AU616819B2 (en) Beta-amino-boronic acid derivatives
AU1261788A (en) Amino acid derivatives
AU2330788A (en) Amino acid derivatives
AU8587791A (en) Amino acid derivatives
AU5252290A (en) Amino acid derivatives
AU7276091A (en) Amino acid derivatives
AU599401B2 (en) Amino acid derivatives
AU2997789A (en) Renin-inhibiting amino acid derivatives
AU3329289A (en) Amino acid derivatives
AU7927891A (en) Amino acid derivatives
AU3255589A (en) Amino acid derivatives
AU2298288A (en) Amino acid derivatives
AU1630088A (en) Amino acid derivatives
AU622734B2 (en) Amino acid derivatives
AU632928B2 (en) Amino acid derivatives
AU6733190A (en) Amino acid derivative
AU3119989A (en) Amino acid derivatives
AU634219B2 (en) Amino acid derivatives
AU623631B2 (en) Amino acid derivatives
AU6311890A (en) Amino acid derivatives