AU2871195A - Methods for the synthesis of diketopiperazines - Google Patents

Methods for the synthesis of diketopiperazines

Info

Publication number
AU2871195A
AU2871195A AU28711/95A AU2871195A AU2871195A AU 2871195 A AU2871195 A AU 2871195A AU 28711/95 A AU28711/95 A AU 28711/95A AU 2871195 A AU2871195 A AU 2871195A AU 2871195 A AU2871195 A AU 2871195A
Authority
AU
Australia
Prior art keywords
diketopiperazines
synthesis
methods
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU28711/95A
Inventor
David Campbell
Mark A. Gallop
Eric M. Gordon
Gary C Look
Dinesh Patel
Anna Katrin Szardenings
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Affymax Technologies NV
Original Assignee
Affymax Technologies NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1995/007878 external-priority patent/WO1995035278A1/en
Application filed by Affymax Technologies NV filed Critical Affymax Technologies NV
Publication of AU2871195A publication Critical patent/AU2871195A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/53—Immunoassay; Biospecific binding assay; Materials therefor
    • G01N33/543—Immunoassay; Biospecific binding assay; Materials therefor with an insoluble carrier for immobilising immunochemicals
    • G01N33/54353—Immunoassay; Biospecific binding assay; Materials therefor with an insoluble carrier for immobilising immunochemicals with ligand attached to the carrier via a chemical coupling agent
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/68—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids
AU28711/95A 1994-06-23 1995-06-23 Methods for the synthesis of diketopiperazines Abandoned AU2871195A (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US393318 1982-06-29
US26557894A 1994-06-23 1994-06-23
US265578 1994-06-23
US39331895A 1995-02-22 1995-02-22
WOUS9507878 1995-06-22
PCT/US1995/007878 WO1995035278A1 (en) 1994-06-22 1995-06-22 Methods for synthesizing diverse collections of pyrrolidine compounds
PCT/US1995/007964 WO1996000391A1 (en) 1994-06-23 1995-06-23 Methods for the synthesis of diketopiperazines

Publications (1)

Publication Number Publication Date
AU2871195A true AU2871195A (en) 1996-01-19

Family

ID=27377866

Family Applications (1)

Application Number Title Priority Date Filing Date
AU28711/95A Abandoned AU2871195A (en) 1994-06-23 1995-06-23 Methods for the synthesis of diketopiperazines

Country Status (2)

Country Link
AU (1) AU2871195A (en)
WO (1) WO1996000391A1 (en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5990112A (en) * 1996-06-18 1999-11-23 Affymax Technologies N.V. Inhibitors of metalloproteases pharmaceutical compositions comprising same and methods of their use
US5811241A (en) * 1995-09-13 1998-09-22 Cortech, Inc. Method for preparing and identifying N-substitued 1,4-piperazines and N-substituted 1,4-piperazinediones
US5846839A (en) * 1995-12-22 1998-12-08 Glaxo Group Limited Methods for hard-tagging an encoded synthetic library
DE19610103A1 (en) 1996-03-15 1997-09-18 Basf Ag Cycloalkyl derivatives and their synthesis on solid phase
DE19621177A1 (en) 1996-05-24 1997-11-27 Basf Ag Carbohydrate derivatives and their synthesis on solid phase
US5932579A (en) 1996-06-18 1999-08-03 Affymax Technologies N.V. Collagenase-1 and stromelysin-1 inhibitors, pharmaceutical compositions comprising same and methods of their use
DE19626762A1 (en) 1996-07-03 1998-01-08 Basf Ag Enzymatically cleavable linker for solid phase synthesis
KR19990071182A (en) * 1998-02-27 1999-09-15 성재갑 Method for preparing diketopiperazine derivatives using solid phase reaction
CN101632669B (en) 2000-08-04 2011-05-18 Dmi生物科学公司 Method of using diketopiperazines and composition containing them
AU2001284697A1 (en) 2000-08-04 2002-02-18 Dmi Biosciences, Inc. Method of synthesizing diketopiperazines
US6815214B2 (en) 2000-12-29 2004-11-09 Celltech R & D, Inc. Pharmaceutical uses and synthesis of diketopiperazines
KR20120091266A (en) 2003-05-15 2012-08-17 디엠아이 바이오사이언시스, 인크 Treatment of t-cell mediated diseases
JP5856843B2 (en) 2008-05-27 2016-02-10 アンピオ ファーマシューティカルズ，インコーポレイテッド Pharmaceutical composition using diketopiperazine
TR201907804T4 (en) * 2009-07-30 2019-06-21 Spiral Therapeutics Inc Apaf-1 inhibitor compounds.
CA2810844C (en) 2010-09-07 2017-03-21 Dmi Acquisition Corp. Diketopiperazine compositions for the treatment of metabolic syndrome and related conditions
SG10201608087WA (en) 2011-10-10 2016-11-29 Ampio Pharmaceuticals Inc Implantable medical devices with increased immune tolerance, and methods for making and implanting
ES2795803T3 (en) 2011-10-10 2020-11-24 Ampio Pharmaceuticals Inc Degenerative arthropathy treatment
AU2012328605B9 (en) 2011-10-28 2017-08-03 Ampio Pharmaceuticals, Inc. Treatment of rhinitis
EA201500943A1 (en) 2013-03-15 2016-08-31 Ампио Фармасьютикалс, Инк. COMPOSITIONS FOR MOBILIZATION, HOUMING, REPRODUCTION AND DIFFERENTION OF STEM CELLS AND METHODS OF APPLICATION OF COMPOSITIONS
WO2015194035A1 (en) * 2014-06-20 2015-12-23 サントリーホールディングス株式会社 Cyclic dipeptide-containing composition
US9956217B2 (en) 2014-08-18 2018-05-01 Ampio Pharmaceuticals, Inc. Treatment of joint conditions
EP3310375A4 (en) 2015-06-22 2019-02-20 Ampio Pharmaceuticals, Inc. Use of low molecular weight fractions of human serum albumin in treating diseases
US10561736B1 (en) 2019-01-09 2020-02-18 Spiral Therapeutics, Inc. Apoptosis inhibitor formulations for prevention of hearing loss
WO2021195265A1 (en) 2020-03-24 2021-09-30 Ampio Pharmaceuticals, Inc. Methods for treating diseases associated with respiratory viruses

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5650489A (en) * 1990-07-02 1997-07-22 The Arizona Board Of Regents Random bio-oligomer library, a method of synthesis thereof, and a method of use thereof
US5324483B1 (en) * 1992-10-08 1996-09-24 Warner Lambert Co Apparatus for multiple simultaneous synthesis

Also Published As

Publication number Publication date
WO1996000391A1 (en) 1996-01-04

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