AU2616199A - Novel bicyclene-substituted oxazolidinones - Google Patents

Novel bicyclene-substituted oxazolidinones

Info

Publication number
AU2616199A
AU2616199A AU26161/99A AU2616199A AU2616199A AU 2616199 A AU2616199 A AU 2616199A AU 26161/99 A AU26161/99 A AU 26161/99A AU 2616199 A AU2616199 A AU 2616199A AU 2616199 A AU2616199 A AU 2616199A
Authority
AU
Australia
Prior art keywords
bicyclene
novel
substituted oxazolidinones
oxazolidinones
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU26161/99A
Inventor
Stephan Bartel
Rainer Endermann
Walter Guarnieri
Dieter Habich
Hein-Peter Kroll
Siegfried Raddatz
Bernd dr. Riedl
Ulrich Rosentreter
Martin Dr. Ruppelt
Andreas Stolle
Hanno dr. Wild
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of AU2616199A publication Critical patent/AU2616199A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
AU26161/99A 1998-01-22 1999-01-09 Novel bicyclene-substituted oxazolidinones Abandoned AU2616199A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19802239 1998-01-22
DE19802239A DE19802239A1 (en) 1998-01-22 1998-01-22 New oxazolidinone derivatives useful as antimicrobial agents against Gram-positive and some Gram-negative bacteria, mycobacteria, etc.
PCT/EP1999/000096 WO1999037641A1 (en) 1998-01-22 1999-01-09 Novel bicyclene-substituted oxazolidinones

Publications (1)

Publication Number Publication Date
AU2616199A true AU2616199A (en) 1999-08-09

Family

ID=7855292

Family Applications (1)

Application Number Title Priority Date Filing Date
AU26161/99A Abandoned AU2616199A (en) 1998-01-22 1999-01-09 Novel bicyclene-substituted oxazolidinones

Country Status (5)

Country Link
EP (1) EP1049692A1 (en)
JP (1) JP2002501065A (en)
AU (1) AU2616199A (en)
DE (1) DE19802239A1 (en)
WO (1) WO1999037641A1 (en)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1142162C (en) 1999-05-27 2004-03-17 法玛西雅厄普约翰美国公司 Bicyclic oxazolidinones as antibacterial agents
MXPA02000985A (en) * 1999-07-28 2002-07-30 Upjohn Co Oxazolidinones and their use as antiinfectives.
DE19962924A1 (en) 1999-12-24 2001-07-05 Bayer Ag Substituted oxazolidinones and their use
PE20011124A1 (en) * 2000-03-31 2001-10-28 Upjohn Co NEW BENZOSULTAM OXAZOLIDINONE ANTIBACTERIAL AGENTS
CA2423599A1 (en) 2000-10-17 2002-04-25 Pharmacia & Upjohn Company Methods of producing oxazolidinone compounds
PE20020689A1 (en) 2000-11-17 2002-08-03 Upjohn Co OXAZOLIDINONES WITH A HETEROCYCLE OF 6 OR 7 MEMBERS UNITED WITH ANNULAR LINK TO BENZENE
DE10129725A1 (en) 2001-06-20 2003-01-02 Bayer Ag Combination therapy of substituted oxazolidinones
AR038536A1 (en) 2002-02-25 2005-01-19 Upjohn Co N-ARIL-2-OXAZOLIDINONA-5- CARBOXAMIDS AND ITS DERIVATIVES
US7141588B2 (en) 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
DE60304360T2 (en) 2002-08-12 2006-11-16 Pharmacia & Upjohn Co. Llc, Kalamazoo N-ARYL-2-OXAZOLIDINONE AND DERIVATIVES
WO2004026848A1 (en) 2002-09-20 2004-04-01 Lupin Limited Oxazolidinone derivatives, process for their preperation and their use as antimycobacterial agents
ES2271660T3 (en) 2002-11-21 2007-04-16 PHARMACIA & UPJOHN COMPANY LLC DERIVATIVES OF N- (4-PIPERAZIN-1-IL) -FENIL-2-OXAZOLIDINONA-5-CARBOXAMIDE AND RELATED COMPOUNDS AS ANTIBACTERIAL AGENTS.
DE10300111A1 (en) 2003-01-07 2004-07-15 Bayer Healthcare Ag Process for the preparation of 5-chloro-N - ({(5S) -2-oxo-3- [4- (3-oxo-4-morpholinyl) phenyl] -1,3-oxazolidin-5-yl} methyl ) -2-thiophenecarboxamide
US7304050B2 (en) 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
DE10355461A1 (en) 2003-11-27 2005-06-23 Bayer Healthcare Ag Solid, high bioavailabilty oral formulations of N-substituted 5-chloro-2-thiophene-carboxamide derivative in hydrophilized form, useful for combating thrombo-embolic diseases
DE102005045518A1 (en) 2005-09-23 2007-03-29 Bayer Healthcare Ag New 5-thienylaminocarbonylmethyl-oxazolidin-2-one derivatives, useful for treating and preventing thromboembolic disease, are selective inhibitors of coagulation factor Xa
US7790745B2 (en) 2005-10-21 2010-09-07 Bristol-Myers Squibb Company Tetrahydroisoquinoline LXR Modulators
CA2642406A1 (en) * 2006-02-14 2007-08-23 Pfizer Products Inc. Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents
JP2014522396A (en) * 2011-05-27 2014-09-04 テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション Substituted 2-benzylidene-2H-benzo [b] [1,4] thiazin-3 (4H) -one, derivatives thereof and therapeutic use thereof
MX362338B (en) 2013-04-16 2019-01-11 Idorsia Pharmaceuticals Ltd Antibacterial biaromatic derivatives.
AR102256A1 (en) 2014-10-15 2017-02-15 Actelion Pharmaceuticals Ltd ANTIBACTERIAL BASIC BIAROMATIC DERIVATIVES WITH REPLACEMENT OF AMINOALCOXI

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE68929303T2 (en) * 1988-09-15 2002-05-02 Upjohn Co 3- (nitrogen substituted) phenyl-5-beta-amidomethyloxazoliden-2-one
DE4425612A1 (en) * 1994-07-20 1996-04-04 Bayer Ag 6-membered nitrogen-containing heteroaryl oxazolidinones
ZA968661B (en) * 1995-11-17 1998-04-14 Upjohn Co Oxazolidinone antibacterial agent with tricyclic substituents.
DE19601265A1 (en) * 1996-01-16 1997-07-17 Bayer Ag 2-oxo and 2-thio-1,2-dihydroquinolinyl oxazolidinones
DE19649095A1 (en) * 1996-02-06 1997-08-07 Bayer Ag New 5-(acyl-aminomethyl)-3-hetero-aryl-oxazolidinone compounds
DE19604223A1 (en) * 1996-02-06 1997-08-07 Bayer Ag New substituted oxazolidinones

Also Published As

Publication number Publication date
WO1999037641A1 (en) 1999-07-29
EP1049692A1 (en) 2000-11-08
DE19802239A1 (en) 1999-07-29
JP2002501065A (en) 2002-01-15

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase