AU2016349833A1 - Use of proteasome inhibitors to treat ocular disorders - Google Patents
Use of proteasome inhibitors to treat ocular disorders Download PDFInfo
- Publication number
- AU2016349833A1 AU2016349833A1 AU2016349833A AU2016349833A AU2016349833A1 AU 2016349833 A1 AU2016349833 A1 AU 2016349833A1 AU 2016349833 A AU2016349833 A AU 2016349833A AU 2016349833 A AU2016349833 A AU 2016349833A AU 2016349833 A1 AU2016349833 A1 AU 2016349833A1
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- Australia
- Prior art keywords
- group
- eye
- composition
- ocular
- proteasome inhibitor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
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- A61K9/0012—Galenical forms characterised by the site of application
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US62/251,937 | 2015-11-06 | ||
| PCT/US2016/058402 WO2017078953A1 (en) | 2015-11-06 | 2016-10-24 | Use of proteasome inhibitors to treat ocular disorders |
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| JP7213891B2 (ja) * | 2018-01-30 | 2023-01-27 | ユニベルシテイト ゲント | 白内障を処置するのに使用するための組成物 |
| BR112021011210A2 (pt) * | 2018-12-10 | 2021-08-24 | EternaTear, Inc. | Formulações oftálmicas que proporcionam lubrificação ocular durável |
| CN110840860B (zh) * | 2019-11-22 | 2021-12-31 | 国家纳米科学中心 | 一种纳米药物及其制备方法和应用 |
| US20230050398A1 (en) * | 2021-08-04 | 2023-02-16 | Harrow Ip, Llc | Methods for increasing shelf-life of ophthalmic pharmaceutical compositions |
| US11471475B1 (en) | 2022-03-08 | 2022-10-18 | Ralph P. Stone | Ophthalmic suspension vehicles and related methods for pharmaceutical ingredient delivery |
| US11679078B1 (en) | 2022-03-08 | 2023-06-20 | EternaTear, Inc. | Ophthalmic formulations and related methods |
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| CN1138542C (zh) * | 1998-04-02 | 2004-02-18 | 诺瓦提斯公司 | 通过特定应用的抗氧化剂稳定药物组合物的方法 |
| EP1830838B1 (en) * | 2004-12-03 | 2012-10-03 | Dana-Farber Cancer Institute, Inc. | Compositions and methods for treating neoplastic diseases |
| WO2006127525A2 (en) * | 2005-05-20 | 2006-11-30 | Jack Arbiser | Proteasome inhibitors and uses thereof |
| JP2009512723A (ja) * | 2005-10-24 | 2009-03-26 | チバ ホールディング インコーポレーテッド | 易酸化性薬剤の保護 |
| RU2456990C2 (ru) * | 2006-09-15 | 2012-07-27 | Янссен Фармацевтика Нв | Комбинации специфичных ингибиторов гистоновых деацетилаз класса i с ингибиторами протеасом |
| CN101541303A (zh) * | 2006-09-29 | 2009-09-23 | 庄臣及庄臣视力保护公司 | 用于治疗眼变态反应性的方法和眼科装置 |
| EP2127638A1 (en) * | 2008-05-30 | 2009-12-02 | Santen Pharmaceutical Co., Ltd | Method and composition for treating ocular hypertension and glaucoma |
| CN103566049B (zh) * | 2012-08-08 | 2017-08-04 | 浙江医药股份有限公司新昌制药厂 | 用于提高眼睛中视黄斑色素密度并预防或治疗年龄相关性视黄斑衰退症的组合物 |
-
2016
- 2016-10-24 CA CA3004587A patent/CA3004587A1/en not_active Abandoned
- 2016-10-24 US US15/773,920 patent/US20180325854A1/en not_active Abandoned
- 2016-10-24 JP JP2018544025A patent/JP2018533629A/ja active Pending
- 2016-10-24 CN CN201680077578.4A patent/CN108883081A/zh active Pending
- 2016-10-24 EP EP16862704.0A patent/EP3370709A4/en not_active Withdrawn
- 2016-10-24 WO PCT/US2016/058402 patent/WO2017078953A1/en not_active Ceased
- 2016-10-24 AU AU2016349833A patent/AU2016349833A1/en not_active Abandoned
-
2018
- 2018-05-06 IL IL259153A patent/IL259153A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL259153A (en) | 2018-06-28 |
| WO2017078953A1 (en) | 2017-05-11 |
| EP3370709A1 (en) | 2018-09-12 |
| CN108883081A (zh) | 2018-11-23 |
| EP3370709A4 (en) | 2019-12-18 |
| JP2018533629A (ja) | 2018-11-15 |
| CA3004587A1 (en) | 2017-05-11 |
| US20180325854A1 (en) | 2018-11-15 |
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