AU2007245496A1 - Amino-ethyl-amino-aryl (AEAA) compounds and their use - Google Patents

Amino-ethyl-amino-aryl (AEAA) compounds and their use Download PDF

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Publication number
AU2007245496A1
AU2007245496A1 AU2007245496A AU2007245496A AU2007245496A1 AU 2007245496 A1 AU2007245496 A1 AU 2007245496A1 AU 2007245496 A AU2007245496 A AU 2007245496A AU 2007245496 A AU2007245496 A AU 2007245496A AU 2007245496 A1 AU2007245496 A1 AU 2007245496A1
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independently
ring
substituent
alkyl
compound according
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AU2007245496A
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Inventor
James Lindsay Carr
Mark David Charles
Caroline Heather Foxton
Julia Helen Gilliatt
Timothy Robin Hammonds
Neela Sumit Mistry
Gregoire Alexandre Pave
Tony Michael Raynham
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Cancer Research Technology Ltd
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Cancer Research Technology Ltd
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Priority claimed from GB0608269A external-priority patent/GB0608269D0/en
Application filed by Cancer Research Technology Ltd filed Critical Cancer Research Technology Ltd
Publication of AU2007245496A1 publication Critical patent/AU2007245496A1/en
Abandoned legal-status Critical Current

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    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
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    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine

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AU2007245496A 2006-04-26 2007-04-26 Amino-ethyl-amino-aryl (AEAA) compounds and their use Abandoned AU2007245496A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US74563006P 2006-04-26 2006-04-26
GB0608269A GB0608269D0 (en) 2006-04-26 2006-04-26 Therapeutic compounds
GB0608269.7 2006-04-26
US60/745,630 2006-04-26
PCT/GB2007/001537 WO2007125331A2 (en) 2006-04-26 2007-04-26 Amino-ethyl-amino-aryl (aeaa) compounds and their use

Publications (1)

Publication Number Publication Date
AU2007245496A1 true AU2007245496A1 (en) 2007-11-08

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AU2007245496A Abandoned AU2007245496A1 (en) 2006-04-26 2007-04-26 Amino-ethyl-amino-aryl (AEAA) compounds and their use

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US (1) US20090247519A1 (enExample)
EP (1) EP2024333A2 (enExample)
JP (1) JP2009534458A (enExample)
AU (1) AU2007245496A1 (enExample)
CA (1) CA2649995A1 (enExample)
IL (1) IL194899A0 (enExample)
MX (1) MX2008013718A (enExample)
WO (1) WO2007125331A2 (enExample)

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EP2099458A4 (en) * 2006-12-01 2011-05-11 Harvard College COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR PRESENTATION AND THERAPY
CN101778825A (zh) * 2007-03-22 2010-07-14 沃泰克斯药物股份有限公司 适用作詹纳斯激酶抑制剂的n-杂环类化合物
ES2535736T3 (es) 2008-06-10 2015-05-14 Novartis Ag Derivados de pirazina como bloqueadores de los canales de sodio epitelial
CN102137856A (zh) * 2008-06-13 2011-07-27 诺瓦提斯公司 作为蛋白激酶d抑制剂的可用于治疗ia心力衰竭和癌症的2,4’-联吡啶化合物
EP2440533B1 (en) 2009-06-12 2015-09-23 Socpra-Sciences Et Génie S.E.C. Guanine riboswitch binding compounds and their use as antibiotics
EP2480537A1 (en) * 2009-09-24 2012-08-01 Basf Se Aminoquinazoline compounds for combating invertebrate pests
US8759363B2 (en) * 2010-01-28 2014-06-24 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Quinazoline-based T cell proliferation inhibitors
JP2013529181A (ja) 2010-03-25 2013-07-18 ザ ジェイ. デヴィッド グラッドストーン インスティテューツ 神経障害を治療するための組成物および方法
US20220235013A1 (en) 2017-03-21 2022-07-28 Bayer Pharma Aktiengesellschaft 2-methyl-quinazolines
CA3097231A1 (en) 2018-04-18 2019-10-24 Bayer Pharma Aktiengesellschaft 2-methyl-aza-quinazolines
JP2022544700A (ja) * 2019-08-22 2022-10-20 バイオヘイブン・セラピューティクス・リミテッド 筋萎縮性側索硬化症および関連障害の治療のためにtdp-43に結合する分子
IL300351A (en) * 2020-08-07 2023-04-01 Athos Therapeutics Inc Small molecules for the treatment of autoimmune diseases and cancer
IL305584A (en) 2021-03-03 2023-10-01 Inst Biologii Doswiadczalnej Imienia Marcelego Nenckiego Polskiej Akademii Nauk Protein kinase D inhibitor for use in the prevention or treatment of hyperlipidemia
EP4052700A1 (en) * 2021-03-03 2022-09-07 Instytut Biologii doswiadczalnej imienia Marcelego Nenckiego Polskiej Akademii Nauk Inhibitor of protein kinase d (pkd) for use in prevention or treatment of obesity and a pharmaceutical composition for such use

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CA2649995A1 (en) 2007-11-08
JP2009534458A (ja) 2009-09-24
US20090247519A1 (en) 2009-10-01
EP2024333A2 (en) 2009-02-18
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