AU2003269850A8 - Hemisuccinate salts of heterocyclic dpp-iv inhibitors - Google Patents

Hemisuccinate salts of heterocyclic dpp-iv inhibitors

Info

Publication number
AU2003269850A8
AU2003269850A8 AU2003269850A AU2003269850A AU2003269850A8 AU 2003269850 A8 AU2003269850 A8 AU 2003269850A8 AU 2003269850 A AU2003269850 A AU 2003269850A AU 2003269850 A AU2003269850 A AU 2003269850A AU 2003269850 A8 AU2003269850 A8 AU 2003269850A8
Authority
AU
Australia
Prior art keywords
dpp
heterocyclic
inhibitors
hemisuccinate
salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003269850A
Other versions
AU2003269850A1 (en
Inventor
Anette Frost Jensen
Lars Nygaard
Kaare Gyberg Rasmussen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novo Nordisk AS
Original Assignee
Novo Nordisk AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk AS filed Critical Novo Nordisk AS
Publication of AU2003269850A1 publication Critical patent/AU2003269850A1/en
Publication of AU2003269850A8 publication Critical patent/AU2003269850A8/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2003269850A 2002-10-08 2003-10-08 Hemisuccinate salts of heterocyclic dpp-iv inhibitors Abandoned AU2003269850A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DKPA200201507 2002-10-08
DKPA200201507 2002-10-08
US41867702P 2002-10-15 2002-10-15
US60/418,677 2002-10-15
PCT/DK2003/000668 WO2004033455A2 (en) 2002-10-08 2003-10-08 Hemisuccinate salts of heterocyclic dpp-iv inhibitors

Publications (2)

Publication Number Publication Date
AU2003269850A1 AU2003269850A1 (en) 2004-05-04
AU2003269850A8 true AU2003269850A8 (en) 2004-05-04

Family

ID=32094934

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003269850A Abandoned AU2003269850A1 (en) 2002-10-08 2003-10-08 Hemisuccinate salts of heterocyclic dpp-iv inhibitors

Country Status (2)

Country Link
AU (1) AU2003269850A1 (en)
WO (1) WO2004033455A2 (en)

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US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
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Also Published As

Publication number Publication date
AU2003269850A1 (en) 2004-05-04
WO2004033455A2 (en) 2004-04-22
WO2004033455A3 (en) 2004-05-27

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase