AU2003264910A1 - Process for selective alkylation of macrolide and azalide derivatives - Google Patents
Process for selective alkylation of macrolide and azalide derivativesInfo
- Publication number
- AU2003264910A1 AU2003264910A1 AU2003264910A AU2003264910A AU2003264910A1 AU 2003264910 A1 AU2003264910 A1 AU 2003264910A1 AU 2003264910 A AU2003264910 A AU 2003264910A AU 2003264910 A AU2003264910 A AU 2003264910A AU 2003264910 A1 AU2003264910 A1 AU 2003264910A1
- Authority
- AU
- Australia
- Prior art keywords
- macrolide
- selective alkylation
- azalide derivatives
- azalide
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 230000029936 alkylation Effects 0.000 title 1
- 238000005804 alkylation reaction Methods 0.000 title 1
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US47434803P | 2003-05-30 | 2003-05-30 | |
US60/474,348 | 2003-05-30 | ||
PCT/HR2003/000048 WO2004106353A1 (en) | 2003-05-30 | 2003-09-04 | Process for selective alkylation of macrolide and azalide derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2003264910A1 true AU2003264910A1 (en) | 2005-01-21 |
Family
ID=33490713
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2003264910A Abandoned AU2003264910A1 (en) | 2003-05-30 | 2003-09-04 | Process for selective alkylation of macrolide and azalide derivatives |
Country Status (3)
Country | Link |
---|---|
CN (1) | CN100381453C (zh) |
AU (1) | AU2003264910A1 (zh) |
WO (1) | WO2004106353A1 (zh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103923142B (zh) * | 2014-04-30 | 2017-01-11 | 浙江震元制药有限公司 | 一种罗红霉素中间体的制备方法 |
CN105801642B (zh) * | 2016-03-11 | 2019-03-26 | 北京理工大学 | 一种制备6,11-双-o-甲基红霉素a的方法 |
CN110494428A (zh) * | 2017-02-14 | 2019-11-22 | 耶路撒冷希伯来大学伊森姆研究发展公司 | 羟基链烯酸的环化方法及其产物 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SI9011409A (en) * | 1990-07-18 | 1995-10-31 | Pliva Pharm & Chem Works | O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them |
WO1999020639A2 (en) * | 1997-10-16 | 1999-04-29 | Pliva, Farmaceutska Industrija ,Dionicko, Drustvo | NOVEL 3,6-HEMIKETALS FROM THE CLASS OF 9a-AZALIDES |
-
2003
- 2003-09-04 AU AU2003264910A patent/AU2003264910A1/en not_active Abandoned
- 2003-09-04 WO PCT/HR2003/000048 patent/WO2004106353A1/en unknown
-
2004
- 2004-05-27 CN CNB2004800148681A patent/CN100381453C/zh not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
WO2004106353A1 (en) | 2004-12-09 |
CN1798755A (zh) | 2006-07-05 |
CN100381453C (zh) | 2008-04-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |