AU2003252990B2 - Bicyclic heteroaromatic compounds as kinase inhibitors - Google Patents

Bicyclic heteroaromatic compounds as kinase inhibitors Download PDF

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Publication number
AU2003252990B2
AU2003252990B2 AU2003252990A AU2003252990A AU2003252990B2 AU 2003252990 B2 AU2003252990 B2 AU 2003252990B2 AU 2003252990 A AU2003252990 A AU 2003252990A AU 2003252990 A AU2003252990 A AU 2003252990A AU 2003252990 B2 AU2003252990 B2 AU 2003252990B2
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AU2003252990A1 (en
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Daniel Christopher Brookings
Jeremy Martin Davis
Barry John Langham
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UCB SA
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UCB SA
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
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  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Communicable Diseases (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
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  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Urology & Nephrology (AREA)
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  • Cardiology (AREA)
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  • Ophthalmology & Optometry (AREA)
AU2003252990A 2002-08-13 2003-08-11 Bicyclic heteroaromatic compounds as kinase inhibitors Ceased AU2003252990B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0218800.1 2002-08-13
GBGB0218800.1A GB0218800D0 (en) 2002-08-13 2002-08-13 Chemical compounds
PCT/GB2003/003501 WO2004014920A1 (en) 2002-08-13 2003-08-11 Bicyclic heteroaromatic compounds as kinase inhibitors

Publications (2)

Publication Number Publication Date
AU2003252990A1 AU2003252990A1 (en) 2004-02-25
AU2003252990B2 true AU2003252990B2 (en) 2009-07-09

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ID=9942221

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003252990A Ceased AU2003252990B2 (en) 2002-08-13 2003-08-11 Bicyclic heteroaromatic compounds as kinase inhibitors

Country Status (7)

Country Link
US (1) US7592455B2 (https=)
EP (1) EP1539769A1 (https=)
JP (1) JP2005537300A (https=)
AU (1) AU2003252990B2 (https=)
CA (1) CA2495518A1 (https=)
GB (1) GB0218800D0 (https=)
WO (1) WO2004014920A1 (https=)

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CA2528603A1 (en) * 2003-06-20 2004-12-29 Celltech R & D Limited Thienopyridone derivatives as kinase inhibitors
US7482452B2 (en) 2003-06-20 2009-01-27 Celltech R&D Limited Process for preparing 3-aminothienopyridone derivatives
CA2528602A1 (en) * 2003-06-20 2004-12-29 Celltech R & D Limited Thienopyridone derivatives as kinase inhibitors
JP2007509123A (ja) * 2003-10-24 2007-04-12 セルテック アール アンド ディ リミテッド キナーゼ阻害剤としてのチエノ−ピリジノン誘導体
WO2007059219A1 (en) 2005-11-15 2007-05-24 Vertex Pharmaceuticals Incorporated Azaindazoles useful as inhibitors of kinases
AR059898A1 (es) 2006-03-15 2008-05-07 Janssen Pharmaceutica Nv Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2
EP2091952A1 (en) * 2006-12-19 2009-08-26 F. Hoffmann-Roche AG Pyrazolo ý3, 4 -d¨pyrimidine p38 map kinase inhibitors
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
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EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
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