AU2003251431A1 - Synthesis of discodermolide - Google Patents

Synthesis of discodermolide

Info

Publication number
AU2003251431A1
AU2003251431A1 AU2003251431A AU2003251431A AU2003251431A1 AU 2003251431 A1 AU2003251431 A1 AU 2003251431A1 AU 2003251431 A AU2003251431 A AU 2003251431A AU 2003251431 A AU2003251431 A AU 2003251431A AU 2003251431 A1 AU2003251431 A1 AU 2003251431A1
Authority
AU
Australia
Prior art keywords
discodermolide
synthesis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003251431A
Inventor
Gordon Florence
Guido Koch
Olivier Loiseleur
Stuart John Mickel
Ian Paterson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Cambridge University Technical Services Ltd CUTS
Original Assignee
Novartis AG
Cambridge University Technical Services Ltd CUTS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0223731A external-priority patent/GB0223731D0/en
Application filed by Novartis AG, Cambridge University Technical Services Ltd CUTS filed Critical Novartis AG
Publication of AU2003251431A1 publication Critical patent/AU2003251431A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AU2003251431A 2002-07-22 2003-07-21 Synthesis of discodermolide Abandoned AU2003251431A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US39797302P 2002-07-22 2002-07-22
US60/397,973 2002-07-22
GB0223731A GB0223731D0 (en) 2002-10-11 2002-10-11 Organic compounds
GB0223731.1 2002-10-11
PCT/EP2003/007940 WO2004009574A1 (en) 2002-07-22 2003-07-21 Synthesis of discodermolide

Publications (1)

Publication Number Publication Date
AU2003251431A1 true AU2003251431A1 (en) 2004-02-09

Family

ID=30772052

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003251431A Abandoned AU2003251431A1 (en) 2002-07-22 2003-07-21 Synthesis of discodermolide

Country Status (2)

Country Link
AU (1) AU2003251431A1 (en)
WO (1) WO2004009574A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20227359B (en) 2017-12-13 2022-03-10 Lupin Ltd Substituted bicyclic heterocyclic compounds as prmt5 inhibitors
CN110041160A (en) * 2018-01-16 2019-07-23 南通诺泰生物医药技术有限公司 Iodo- 4- benzyloxy-3- methyl-1-ene compound of (3R)-2- and its preparation method and application

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9315802D0 (en) * 1993-07-30 1993-09-15 Roussel Lab Ltd Chemical compounds
US5789605A (en) * 1996-12-03 1998-08-04 Trustees Of The University Of Pennsylvania Synthetic techniques and intermediates for polyhydroxy, dienyl lactones and mimics thereof
TWI251591B (en) * 2000-08-07 2006-03-21 Novartis Ag Process for preparing discodermolide and analogues thereof
GB0101599D0 (en) * 2001-01-22 2001-03-07 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
WO2004009574A1 (en) 2004-01-29

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