AU2002350869A1 - Polymorphous form of rimonabant, preperation method and pharmaceutical compositions containing same - Google Patents
Polymorphous form of rimonabant, preperation method and pharmaceutical compositions containing sameInfo
- Publication number
- AU2002350869A1 AU2002350869A1 AU2002350869A AU2002350869A AU2002350869A1 AU 2002350869 A1 AU2002350869 A1 AU 2002350869A1 AU 2002350869 A AU2002350869 A AU 2002350869A AU 2002350869 A AU2002350869 A AU 2002350869A AU 2002350869 A1 AU2002350869 A1 AU 2002350869A1
- Authority
- AU
- Australia
- Prior art keywords
- rimonabant
- pharmaceutical compositions
- compositions containing
- containing same
- polymorphous form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- JZCPYUJPEARBJL-UHFFFAOYSA-N Rimonabant Chemical compound CC=1C(C(=O)NN2CCCCC2)=NN(C=2C(=CC(Cl)=CC=2)Cl)C=1C1=CC=C(Cl)C=C1 JZCPYUJPEARBJL-UHFFFAOYSA-N 0.000 title 1
- 229960003015 Rimonabant Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR01/14579 | 2001-11-08 | ||
FR0114579A FR2831883B1 (en) | 2001-11-08 | 2001-11-08 | POLYMORPHIC FORM OF RIMONABANT, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
PCT/FR2002/003765 WO2003040105A1 (en) | 2001-11-08 | 2002-11-04 | Polymorphous form of rimonabant, preparation method and pharmaceutical compositions containing same |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002350869A1 true AU2002350869A1 (en) | 2003-07-24 |
AU2002350869B2 AU2002350869B2 (en) | 2007-07-26 |
Family
ID=8869285
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002350869A Ceased AU2002350869B2 (en) | 2001-11-08 | 2002-11-04 | Polymorphous form of rimonabant, preperation method and pharmaceutical compositions containing same |
Country Status (33)
Country | Link |
---|---|
US (2) | US20050043356A1 (en) |
EP (1) | EP1446384A1 (en) |
JP (2) | JP4181994B2 (en) |
KR (2) | KR20050043774A (en) |
CN (1) | CN100412063C (en) |
AP (1) | AP1830A (en) |
AR (1) | AR037253A1 (en) |
AU (1) | AU2002350869B2 (en) |
BR (1) | BR0213931A (en) |
CA (1) | CA2464145A1 (en) |
CO (1) | CO5580827A2 (en) |
CR (1) | CR7333A (en) |
EA (1) | EA006771B1 (en) |
EC (1) | ECSP045088A (en) |
FR (1) | FR2831883B1 (en) |
GE (1) | GEP20063894B (en) |
HR (1) | HRP20040403A2 (en) |
HU (1) | HUP0402043A3 (en) |
IL (2) | IL161533A0 (en) |
IS (1) | IS7226A (en) |
MA (1) | MA27080A1 (en) |
ME (1) | MEP21908A (en) |
MX (1) | MXPA04004394A (en) |
NO (1) | NO326648B1 (en) |
NZ (1) | NZ532369A (en) |
OA (1) | OA12721A (en) |
PL (1) | PL369372A1 (en) |
RS (1) | RS36904A (en) |
TN (1) | TNSN04079A1 (en) |
TW (1) | TW200302824A (en) |
UA (1) | UA76776C2 (en) |
WO (1) | WO2003040105A1 (en) |
ZA (1) | ZA200402999B (en) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2831883B1 (en) * | 2001-11-08 | 2004-07-23 | Sanofi Synthelabo | POLYMORPHIC FORM OF RIMONABANT, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
NZ537003A (en) | 2002-07-18 | 2008-03-28 | Cytos Biotechnology Ag | Hapten-carrier conjugates comprising virus like particles and uses thereof |
FR2861992B1 (en) * | 2003-11-10 | 2007-07-20 | Sanofi Synthelabo | PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION OF A PYRAZOLE-3-CARBOXAMIDE DERIVATIVE. |
WO2007003962A2 (en) | 2005-06-30 | 2007-01-11 | Prosidion Limited | Gpcr agonists |
EP1816125A1 (en) * | 2006-02-02 | 2007-08-08 | Ranbaxy Laboratories, Ltd. | Novel crystalline forms of an antagonist of CB1 cannabinoid receptor and preparation method thereof |
FR2897060B1 (en) * | 2006-02-08 | 2008-07-25 | Sanofi Aventis Sa | RIMONABANT MONOHYDRATE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
WO2008038143A2 (en) * | 2006-06-22 | 2008-04-03 | Medichem, S.A. | Novel solid forms of rimonabant and synthetic processes for their preparation |
WO2008044153A2 (en) * | 2006-08-29 | 2008-04-17 | Medichem, S.A. | Improved method for synthesizing rimonabant |
EP2057144A4 (en) * | 2006-09-01 | 2010-06-02 | Hetero Drugs Ltd | Novel polymorphs of rimonabant |
EP2061783A2 (en) * | 2006-09-11 | 2009-05-27 | Hetero Drugs Limited | Improved process for rimonabant |
WO2008035023A1 (en) * | 2006-09-19 | 2008-03-27 | Cipla Limited | Polymorphs of rimonabant |
WO2008056377A2 (en) * | 2006-11-06 | 2008-05-15 | Cadila Healthcare Limited | Polymorphic forms of rimonabant |
WO2008064615A2 (en) * | 2006-12-01 | 2008-06-05 | Zentiva, A.S. | Crystalline and amorphous forms of rimonabant and processes for obtaining them |
CN103145620A (en) * | 2006-12-18 | 2013-06-12 | 7Tm制药联合股份有限公司 | Cb1 receptor modulators |
AR064735A1 (en) | 2007-01-04 | 2009-04-22 | Prosidion Ltd | GPCR AGONISTS AND PHARMACEUTICAL COMPOSITION BASED ON THE COMPOUND |
PE20081849A1 (en) | 2007-01-04 | 2009-01-26 | Prosidion Ltd | PIPERIDIN-4-IL-PROPOXY-BENZAMIDE DERIVATIVES AS GPCR AGONISTS |
CA2674360A1 (en) | 2007-01-04 | 2008-07-10 | Prosidion Limited | Piperidine gpcr agonists |
RS52065B (en) | 2007-01-04 | 2012-06-30 | Prosidion Ltd | Piperidine gpcr agonists |
GB0700122D0 (en) | 2007-01-04 | 2007-02-14 | Prosidion Ltd | GPCR agonists |
EP1944297A1 (en) * | 2007-01-09 | 2008-07-16 | Miklós Vértessy | Solid and crystalline rimonabant and processes for preparation, and pharmaceutical composition thereof |
WO2008088900A2 (en) * | 2007-01-18 | 2008-07-24 | Teva Pharmaceutical Industries Ltd. | Polymorphic forms of rimonabant base and processes for preparation thereof |
EP1953144A1 (en) * | 2007-01-30 | 2008-08-06 | Sandoz AG | Novel polymorphic forms of N-piperidino-5-(4-chlorophenyl)-1-(2, 4-dichlorphenyl)-4-methyl-3-pyrazolecarboxamide |
FR2919862A1 (en) * | 2007-08-06 | 2009-02-13 | Sanofi Aventis Sa | RIMONABANT 3-METHYLBUTAN-1-OL SOLVATE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR2919863A1 (en) * | 2007-08-06 | 2009-02-13 | Sanofi Aventis Sa | RIMONABANT N-METHYLPYRROLIDONE SOLVATE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR2919864A1 (en) * | 2007-08-06 | 2009-02-13 | Sanofi Aventis Sa | RIMONABANT 1,4-DIOXANE SOLVATE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR2919865A1 (en) * | 2007-08-06 | 2009-02-13 | Sanofi Aventis Sa | RIMONABANT DMSO SOLVATE, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR2919867A1 (en) * | 2007-08-06 | 2009-02-13 | Sanofi Aventis Sa | RIMONABANT 2-METHOXYETHANOL SOLVATE AND PROCESS FOR PREPARING THE SAME |
GB0720389D0 (en) | 2007-10-18 | 2008-11-12 | Prosidion Ltd | G-Protein Coupled Receptor Agonists |
GB0720390D0 (en) | 2007-10-18 | 2007-11-28 | Prosidion Ltd | G-Protein coupled receptor agonists |
WO2009153804A1 (en) * | 2008-06-16 | 2009-12-23 | Cadila Healthcare Limited | Process for preparing form i of rimonabant |
WO2010079241A1 (en) | 2009-01-12 | 2010-07-15 | Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion | Use of antagonists and/or inverse agonists of cb1 receptors for the preparation of drugs that increase motor neuron excitability |
FR3008620A1 (en) * | 2013-07-22 | 2015-01-23 | Sanofi Sa | COMPRESSOR FORMULATION OF A PHOSPHATIDYLINOSITOL 3-KINASE INHIBITOR |
EP4046687A4 (en) * | 2019-10-16 | 2023-11-15 | Otsuka Pharmaceutical Co., Ltd. | Method for producing centanafadine |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2713225B1 (en) * | 1993-12-02 | 1996-03-01 | Sanofi Sa | Substituted N-piperidino-3-pyrazolecarboxamide. |
FR2692575B1 (en) * | 1992-06-23 | 1995-06-30 | Sanofi Elf | NOVEL PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
WO2003015700A2 (en) * | 2001-08-15 | 2003-02-27 | The Government Of The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services | Novel vasoconstrictor cannabinoid analogs |
FR2831883B1 (en) * | 2001-11-08 | 2004-07-23 | Sanofi Synthelabo | POLYMORPHIC FORM OF RIMONABANT, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
-
2001
- 2001-11-08 FR FR0114579A patent/FR2831883B1/en not_active Expired - Fee Related
-
2002
- 2002-04-11 UA UA20040402974A patent/UA76776C2/en unknown
- 2002-11-04 RS YU36904A patent/RS36904A/en unknown
- 2002-11-04 KR KR1020047006969A patent/KR20050043774A/en not_active Application Discontinuation
- 2002-11-04 WO PCT/FR2002/003765 patent/WO2003040105A1/en active Application Filing
- 2002-11-04 ME MEP-219/08A patent/MEP21908A/en unknown
- 2002-11-04 CN CNB028219686A patent/CN100412063C/en not_active Expired - Fee Related
- 2002-11-04 IL IL16153302A patent/IL161533A0/en unknown
- 2002-11-04 GE GE5606A patent/GEP20063894B/en unknown
- 2002-11-04 CA CA002464145A patent/CA2464145A1/en not_active Abandoned
- 2002-11-04 OA OA1200400131A patent/OA12721A/en unknown
- 2002-11-04 NZ NZ532369A patent/NZ532369A/en not_active IP Right Cessation
- 2002-11-04 AP APAP/P/2004/003024A patent/AP1830A/en active
- 2002-11-04 AU AU2002350869A patent/AU2002350869B2/en not_active Ceased
- 2002-11-04 HU HU0402043A patent/HUP0402043A3/en unknown
- 2002-11-04 EP EP02785580A patent/EP1446384A1/en not_active Withdrawn
- 2002-11-04 JP JP2003542151A patent/JP4181994B2/en not_active Expired - Fee Related
- 2002-11-04 MX MXPA04004394A patent/MXPA04004394A/en unknown
- 2002-11-04 US US10/494,211 patent/US20050043356A1/en not_active Abandoned
- 2002-11-04 PL PL02369372A patent/PL369372A1/en not_active Application Discontinuation
- 2002-11-04 KR KR1020097016373A patent/KR20090089485A/en not_active Application Discontinuation
- 2002-11-04 BR BR0213931-6A patent/BR0213931A/en not_active IP Right Cessation
- 2002-11-04 EA EA200400491A patent/EA006771B1/en not_active IP Right Cessation
- 2002-11-06 AR ARP020104228A patent/AR037253A1/en unknown
- 2002-11-07 TW TW091132763A patent/TW200302824A/en unknown
-
2004
- 2004-04-19 IS IS7226A patent/IS7226A/en unknown
- 2004-04-20 ZA ZA200402999A patent/ZA200402999B/en unknown
- 2004-04-20 IL IL161533A patent/IL161533A/en not_active IP Right Cessation
- 2004-04-27 EC EC2004005088A patent/ECSP045088A/en unknown
- 2004-04-28 MA MA27659A patent/MA27080A1/en unknown
- 2004-05-04 CR CR7333A patent/CR7333A/en unknown
- 2004-05-04 CO CO04040840A patent/CO5580827A2/en not_active Application Discontinuation
- 2004-05-06 HR HR20040403A patent/HRP20040403A2/en not_active Application Discontinuation
- 2004-05-07 TN TNP2004000079A patent/TNSN04079A1/en unknown
- 2004-05-07 NO NO20041879A patent/NO326648B1/en not_active IP Right Cessation
-
2008
- 2008-07-11 JP JP2008181474A patent/JP4931874B2/en not_active Expired - Fee Related
- 2008-10-28 US US12/259,701 patent/US20100190827A1/en not_active Abandoned
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU2002350869A1 (en) | Polymorphous form of rimonabant, preperation method and pharmaceutical compositions containing same | |
IL161533A0 (en) | Polymorphous form of rimonabant, preparation method and pharmaceutical compositions containing same | |
AU2002363236A1 (en) | Compounds, pharmaceutical compositions and methods of use therefor | |
HUP0500173A3 (en) | Alpha-sulphonamido-acetamide derivatives as beta-amyloid inhibitors and pharmaceutical compositions containing them | |
HUP0401898A3 (en) | 3-substituted-4-pyrimidone derivatives, pharmaceutical compositions containing them and their intermediates | |
HUP0401748A3 (en) | 2-amino-4,5-trisubstituted thiazolyl derivatives, process for their preparation and pharmaceutical compositions containing them | |
HUP0401900A3 (en) | 3-substituted-4-pyrimidone derivatives, pharmaceutical compositions containing them and their intermediates | |
HU0103063D0 (en) | New 2h-pyridazin-3-one derivatives, process for their preparation and pharmaceutical compositions containing them | |
IL158898A0 (en) | PHARMACEUTICAL COMPOSITIONS CONTAINING APOMORPHINE, 6aR-(-)-N-PROPYL-NORAPOMORPHINE AND DERIVATIVES THEREOF | |
AU2002364342A1 (en) | Heteroxylan film-forming composition for making capsules and resulting capsules | |
AU2002240359A1 (en) | Pharmaceutical composition for the treatment of alopecia | |
HUP0400549A3 (en) | Novel imidazole derivatives, production method thereof and pharmaceutical compositions containing them | |
PL356911A1 (en) | Novel heterocyclic derivatives, preparation method and pharmaceutical compositions containing same | |
AU2003251695A1 (en) | Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same | |
HUP0401018A3 (en) | 2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof | |
AU2002351388A1 (en) | Methods and compositions for controlled release of drugs | |
AU2002313065A1 (en) | Novel piperidinecarboxamide derivatives, method for preparing same and pharmaceutical compositions containing same | |
AU2001252711A1 (en) | Aqueous-prodrug compound comprising moiety of paclitxel or derivatives thereof, method of preparing same and pharmaceutical composition comprising same | |
IL158660A0 (en) | Novel piperidinecarboxamide derivatives, method for preparing same and pharmaceutical compositions containing same | |
AU2002306687A1 (en) | Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them | |
AU2002210632A1 (en) | Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same | |
HUP0402600A3 (en) | D-proline derivatives and pharmaceutical compositions containing them | |
SI1245565T1 (en) | Indenoindolone derivatives, process for their preparation and pharmaceutical compositions containing them | |
AU2002303552A1 (en) | Methods and compositions for prevention of angioproliferation | |
SI1241169T1 (en) | Isoindoloindolone derivatives, process for their preparation and pharmaceutical compositions containing them |