AU2002247726A1 - 2-Thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industry - Google Patents
2-Thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industryInfo
- Publication number
- AU2002247726A1 AU2002247726A1 AU2002247726A AU2002247726A AU2002247726A1 AU 2002247726 A1 AU2002247726 A1 AU 2002247726A1 AU 2002247726 A AU2002247726 A AU 2002247726A AU 2002247726 A AU2002247726 A AU 2002247726A AU 2002247726 A1 AU2002247726 A1 AU 2002247726A1
- Authority
- AU
- Australia
- Prior art keywords
- thio
- pharmaceutical industry
- imidazole derivatives
- substituted imidazole
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229940041158 antibacterial for systemic use Imidazole derivatives Drugs 0.000 title 1
- 229940042051 antimycotic for systemic use Imidazole derivatives Drugs 0.000 title 1
- 229940093910 gyncological antiinfectives Imidazole derivatives Drugs 0.000 title 1
- 150000002460 imidazoles Chemical class 0.000 title 1
- 229940079865 intestinal antiinfectives Imidazole derivatives Drugs 0.000 title 1
- 238000005020 pharmaceutical industry Methods 0.000 title 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10107683A DE10107683A1 (en) | 2001-02-19 | 2001-02-19 | 2-Thio-substituted imidazole derivatives and their use in pharmacy |
| DE10107683.5 | 2001-02-19 | ||
| PCT/EP2002/001746 WO2002066458A2 (en) | 2001-02-19 | 2002-02-19 | 2-thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industry |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| AU2002247726A1 true AU2002247726A1 (en) | 2003-02-27 |
| AU2002247726B2 AU2002247726B2 (en) | 2006-01-19 |
| AU2002247726C1 AU2002247726C1 (en) | 2006-08-17 |
Family
ID=7674545
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002247726A Ceased AU2002247726C1 (en) | 2001-02-19 | 2002-02-19 | 2-Thio-substituted imidazole derivatives and the use thereof in the pharmaceutical industry |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7253191B2 (en) |
| EP (1) | EP1362045B1 (en) |
| JP (1) | JP2004521913A (en) |
| KR (1) | KR100642231B1 (en) |
| CN (1) | CN1291984C (en) |
| AT (1) | ATE282605T1 (en) |
| AU (1) | AU2002247726C1 (en) |
| BR (1) | BR0207254A (en) |
| CA (1) | CA2453078A1 (en) |
| CZ (1) | CZ20032224A3 (en) |
| DE (2) | DE10107683A1 (en) |
| DK (1) | DK1362045T3 (en) |
| ES (1) | ES2233808T3 (en) |
| HK (1) | HK1056725A1 (en) |
| HU (1) | HUP0303155A3 (en) |
| IL (1) | IL157050A0 (en) |
| IS (1) | IS6914A (en) |
| MX (1) | MXPA03007380A (en) |
| PL (1) | PL367397A1 (en) |
| PT (1) | PT1362045E (en) |
| RU (1) | RU2284326C2 (en) |
| SK (1) | SK10242003A3 (en) |
| WO (1) | WO2002066458A2 (en) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10107683A1 (en) | 2001-02-19 | 2002-08-29 | Merckle Gmbh Chem Pharm Fabrik | 2-Thio-substituted imidazole derivatives and their use in pharmacy |
| DE10222103A1 (en) | 2002-05-17 | 2003-11-27 | Merckle Gmbh Chem Pharm Fabrik | New 2-(substituted thio)-imidazole derivatives are immunomodulators and cytokine release inhibitors, useful for treating diseases associated with immune system disorders, e.g. cancer or rheumatoid arthritis |
| DE10238045A1 (en) * | 2002-08-20 | 2004-03-04 | Merckle Gmbh Chem.-Pharm. Fabrik | 2-Thio-substituted imidazole derivatives and their use in pharmacy |
| DE10256881A1 (en) * | 2002-12-05 | 2004-06-24 | Beiersdorf Ag | New topical use of bis-arylimidazo [1,2-a] thiolane derivatives |
| JP2008500311A (en) * | 2004-05-26 | 2008-01-10 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Mercaptoimidazoles as CCR2 receptor antagonists |
| WO2005118578A1 (en) | 2004-05-26 | 2005-12-15 | Janssen Pharmaceutica N.V. | Mercaptoimidazoles as ccr2 receptor antagonists |
| CA2573066A1 (en) * | 2004-08-11 | 2006-02-16 | Janssen Pharmaceutica N.V. | Mercaptoimidazoles as ccr2 receptor antagonists |
| US20100273833A1 (en) * | 2005-02-28 | 2010-10-28 | Wolfgang Albrecht | 2-sulfinyl- and 2-sulfonyl-substituted imidazole derivatives and their use as cytokine inhibitors |
| EP1894925A1 (en) * | 2006-08-24 | 2008-03-05 | Merckle Gmbh | Imidazole compounds having an antiinflammatory effect |
| WO2008085008A1 (en) * | 2007-01-11 | 2008-07-17 | Mogam Biotechnology Research Institute | T-cell inhibiting compounds and their use for the treatment of t-cell-mediated diseases |
| US8143294B2 (en) | 2007-12-31 | 2012-03-27 | Michael Burnet | 2-sulfanyl-substituted imidazole derivatives and their use as cytokine inhibitors |
| CN102249992A (en) * | 2011-07-05 | 2011-11-23 | 广东工业大学 | Method for preparing 2-aminoisonicotinic acid |
| DE102013102069A1 (en) | 2013-03-01 | 2014-09-04 | Fsp Fluid Systems Partners Holding Ag | Proportional directional valve and hydraulic circuit and hydropneumatic suspension system with such a valve |
| WO2017151409A1 (en) | 2016-02-29 | 2017-09-08 | University Of Florida Research Foundation, Incorporated | Chemotherapeutic methods |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO120426B (en) * | 1965-10-21 | 1970-10-19 | Geigy Ag J R | |
| US4190666A (en) * | 1975-08-11 | 1980-02-26 | E. I. Du Pont De Nemours And Company | Anti-inflammatory 4,5-diarly-2-(substituted-thio)imidazoles and their corresponding sulfoxides and sulfones |
| DK16778A (en) | 1977-02-09 | 1978-08-10 | Du Pont | IMIDAZOLE DERIVATIVES THEIR USES AND MANUFACTURE |
| CY1302A (en) * | 1978-04-11 | 1985-12-06 | Ciba Geigy Ag | Mercapto-imidazole derivatives,their preparation,their pharmaceutical compositions and applications |
| DE2823197A1 (en) | 1978-05-24 | 1979-11-29 | Schering Ag | NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| DE3025484A1 (en) * | 1980-07-03 | 1982-02-04 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| DE3141063A1 (en) * | 1981-10-13 | 1983-04-28 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| DE3504678A1 (en) * | 1985-02-12 | 1986-08-14 | A. Nattermann & Cie GmbH, 5000 Köln | Novel imidazolyl-oxyalkanoic acids and -thioalkanoic acids, derivatives thereof, and processes for their preparation |
| US4686231A (en) | 1985-12-12 | 1987-08-11 | Smithkline Beckman Corporation | Inhibition of 5-lipoxygenase products |
| JPS6440467A (en) | 1987-08-04 | 1989-02-10 | Hisamitsu Pharmaceutical Co | Novel substituted diphenylimidazole derivative |
| FR2626691B1 (en) | 1988-02-02 | 1990-05-25 | France Etat | GENERALIZED DIGITAL MULTIPLIER AND DIGITAL FILTER IMPLEMENTING THIS MULTIPLIER |
| CA2073443A1 (en) | 1990-01-12 | 1991-07-13 | Andrew William Bridge | 2-substituted 4,5-diphenyl-imidazoles |
| IL104369A0 (en) | 1992-01-13 | 1993-05-13 | Smithkline Beecham Corp | Novel compounds and compositions |
| US5364875A (en) * | 1992-05-11 | 1994-11-15 | The Du Pont Merck Pharmaceutical Company | Imidazoles linked to bicyclic heterocyclic groups for the treatment of atherosclerosis |
| US5474995A (en) | 1993-06-24 | 1995-12-12 | Merck Frosst Canada, Inc. | Phenyl heterocycles as cox-2 inhibitors |
| AU7629594A (en) | 1993-07-21 | 1995-02-20 | Smithkline Beecham Corporation | Imidazoles for treating cytokine mediated disease |
| US5620999A (en) | 1994-07-28 | 1997-04-15 | Weier; Richard M. | Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation |
| US6040320A (en) * | 1997-06-30 | 2000-03-21 | Ortho-Mcneil Pharmaceutical, Inc. | 2-substituted imidazoles useful in the treatment of inflammatory diseases |
| DE19842833B4 (en) | 1998-09-18 | 2005-04-14 | Merckle Gmbh | 2-Arylalkylthio-imidazoles, 2-Arylalkenylthio-imidazoles and 2-Arylalkinylthio-imidazole as anti-inflammatory and inhibitors of cytokine release |
| DE10107683A1 (en) | 2001-02-19 | 2002-08-29 | Merckle Gmbh Chem Pharm Fabrik | 2-Thio-substituted imidazole derivatives and their use in pharmacy |
-
2001
- 2001-02-19 DE DE10107683A patent/DE10107683A1/en not_active Withdrawn
-
2002
- 2002-02-19 IL IL15705002A patent/IL157050A0/en unknown
- 2002-02-19 CZ CZ20032224A patent/CZ20032224A3/en unknown
- 2002-02-19 US US10/467,064 patent/US7253191B2/en not_active Expired - Fee Related
- 2002-02-19 EP EP02716791A patent/EP1362045B1/en not_active Expired - Lifetime
- 2002-02-19 CN CNB028051548A patent/CN1291984C/en not_active Expired - Fee Related
- 2002-02-19 KR KR1020037010839A patent/KR100642231B1/en not_active IP Right Cessation
- 2002-02-19 AU AU2002247726A patent/AU2002247726C1/en not_active Ceased
- 2002-02-19 DK DK02716791T patent/DK1362045T3/en active
- 2002-02-19 DE DE50201565T patent/DE50201565D1/en not_active Expired - Lifetime
- 2002-02-19 ES ES02716791T patent/ES2233808T3/en not_active Expired - Lifetime
- 2002-02-19 WO PCT/EP2002/001746 patent/WO2002066458A2/en active IP Right Grant
- 2002-02-19 SK SK1024-2003A patent/SK10242003A3/en not_active Application Discontinuation
- 2002-02-19 AT AT02716791T patent/ATE282605T1/en not_active IP Right Cessation
- 2002-02-19 RU RU2003128068/04A patent/RU2284326C2/en not_active IP Right Cessation
- 2002-02-19 PT PT02716791T patent/PT1362045E/en unknown
- 2002-02-19 HU HU0303155A patent/HUP0303155A3/en unknown
- 2002-02-19 CA CA002453078A patent/CA2453078A1/en not_active Abandoned
- 2002-02-19 MX MXPA03007380A patent/MXPA03007380A/en active IP Right Grant
- 2002-02-19 PL PL02367397A patent/PL367397A1/en not_active Application Discontinuation
- 2002-02-19 BR BR0207254-8A patent/BR0207254A/en not_active IP Right Cessation
- 2002-02-19 JP JP2002565973A patent/JP2004521913A/en active Pending
-
2003
- 2003-08-15 IS IS6914A patent/IS6914A/en unknown
- 2003-12-11 HK HK03109068A patent/HK1056725A1/en not_active IP Right Cessation
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