AU2002227931A1 - Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as medicament, and pharmaceutical preparations containing these compounds - Google Patents
Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as medicament, and pharmaceutical preparations containing these compoundsInfo
- Publication number
- AU2002227931A1 AU2002227931A1 AU2002227931A AU2002227931A AU2002227931A1 AU 2002227931 A1 AU2002227931 A1 AU 2002227931A1 AU 2002227931 A AU2002227931 A AU 2002227931A AU 2002227931 A AU2002227931 A AU 2002227931A AU 2002227931 A1 AU2002227931 A1 AU 2002227931A1
- Authority
- AU
- Australia
- Prior art keywords
- substituted
- compounds
- ortho
- meta
- medicament
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10059418.2 | 2000-11-30 | ||
DE10059418A DE10059418A1 (en) | 2000-11-30 | 2000-11-30 | Ortho, meta-substituted bisaryl compounds, processes for their preparation, their use as medicaments and pharmaceutical preparations containing them |
PCT/EP2001/013294 WO2002044137A1 (en) | 2000-11-30 | 2001-11-17 | Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as a medicament, and pharmaceutical preparations containing these compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002227931A1 true AU2002227931A1 (en) | 2002-08-15 |
AU2002227931B2 AU2002227931B2 (en) | 2006-07-13 |
Family
ID=7665215
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002227931A Ceased AU2002227931B2 (en) | 2000-11-30 | 2001-11-17 | Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as medicament, and pharmaceutical preparations containing these compounds |
AU2793102A Pending AU2793102A (en) | 2000-11-30 | 2001-11-17 | Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as a medicament, and pharmaceutical preparations containing these compounds |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2793102A Pending AU2793102A (en) | 2000-11-30 | 2001-11-17 | Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as a medicament, and pharmaceutical preparations containing these compounds |
Country Status (29)
Country | Link |
---|---|
US (2) | US6605625B2 (en) |
EP (1) | EP1339675B1 (en) |
JP (1) | JP4051283B2 (en) |
KR (1) | KR100968056B1 (en) |
CN (1) | CN1290825C (en) |
AR (1) | AR031430A1 (en) |
AT (1) | ATE289292T1 (en) |
AU (2) | AU2002227931B2 (en) |
BR (1) | BR0115769A (en) |
CA (1) | CA2430273C (en) |
CZ (1) | CZ301631B6 (en) |
DE (2) | DE10059418A1 (en) |
EE (1) | EE05240B1 (en) |
ES (1) | ES2236341T3 (en) |
HK (1) | HK1061231A1 (en) |
HR (1) | HRP20030436B1 (en) |
HU (1) | HUP0303317A3 (en) |
IL (2) | IL156097A0 (en) |
MX (1) | MXPA03004386A (en) |
NO (1) | NO328599B1 (en) |
NZ (1) | NZ526177A (en) |
PL (1) | PL206245B1 (en) |
PT (1) | PT1339675E (en) |
RS (1) | RS50403B (en) |
RU (1) | RU2278858C2 (en) |
SK (1) | SK286708B6 (en) |
TW (1) | TWI254039B (en) |
WO (1) | WO2002044137A1 (en) |
ZA (1) | ZA200303893B (en) |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10060807A1 (en) * | 2000-12-07 | 2002-06-20 | Aventis Pharma Gmbh | Ortho, ortho-substituted nitrogen-containing bisaryl compounds, processes for their preparation, their use as medicaments and pharmaceutical preparations containing them |
GB0124936D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124934D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124938D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124941D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124931D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124933D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124939D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
PL212910B1 (en) * | 2002-02-12 | 2012-12-31 | Smithkline Beecham Corp | Nicotinamide derivates useful as p38 inhibitors |
GB0217757D0 (en) | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | Novel compounds |
AU2003258630A1 (en) | 2002-08-19 | 2004-03-11 | Glaxo Group Limited | Pyrimidine derivatives as selective cox-2 inhibitors |
GB0221443D0 (en) | 2002-09-16 | 2002-10-23 | Glaxo Group Ltd | Pyridine derivates |
ES2571779T3 (en) * | 2002-12-13 | 2016-05-26 | Ym Biosciences Australia Pty | Nicotinamide-based kinase inhibitors |
CA2508171C (en) * | 2002-12-13 | 2012-08-28 | Cytopia Pty Ltd | Nicotinamide-based kinase inhibitors |
AU2003291839B2 (en) * | 2002-12-13 | 2009-01-22 | Ym Biosciences Australia Pty Ltd | Nicotinamide-based kinase inhibitors |
GB0308185D0 (en) * | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
GB0315950D0 (en) | 2003-06-11 | 2003-08-13 | Xention Discovery Ltd | Compounds |
DE10341233A1 (en) * | 2003-09-08 | 2005-03-24 | Aventis Pharma Deutschland Gmbh | Composition, useful to treat e.g. atrial fibrillation, atrial flutter and atrial arrhythmia, comprises at least one beta-blocker and at least one compound of a phenylcarboxylic acid amide derivative |
US20050054673A1 (en) * | 2003-09-08 | 2005-03-10 | Aventis Pharma Deutschland Gmbh | Combination of phenylcarboxylic acid amides with beta-adrenoreceptor blockers and their use for the treatment of atrial arrhythmias |
US7691879B2 (en) * | 2003-09-23 | 2010-04-06 | Merck Sharp & Dohme Corp. | Isoquinoline potassium channel inhibitors |
US7647300B2 (en) * | 2004-01-26 | 2010-01-12 | Google Inc. | Methods and systems for output of search results |
GB0402143D0 (en) * | 2004-01-30 | 2004-03-03 | Smithkline Beecham Corp | Novel compounds |
GB0403744D0 (en) * | 2004-02-20 | 2004-03-24 | Astrazeneca Ab | Chemical process |
JP2007528420A (en) * | 2004-03-11 | 2007-10-11 | グラクソ グループ リミテッド | Novel M3 muscarinic acetylcholine receptor antagonist |
GB0412986D0 (en) | 2004-06-10 | 2004-07-14 | Xention Discovery Ltd | Compounds |
CN1993348A (en) * | 2004-07-29 | 2007-07-04 | 默克公司 | Potassium channel inhibitors |
US7569589B2 (en) | 2004-07-29 | 2009-08-04 | Merck & Co., Inc. | Potassium channel inhibitors |
US20080051416A1 (en) * | 2004-10-05 | 2008-02-28 | Smithkline Beecham Corporation | Novel Compounds |
US7932247B2 (en) | 2004-11-15 | 2011-04-26 | Glaxo Group Limited | M3 muscarinic acetylcholine receptor antagonists |
US7576212B2 (en) | 2004-12-09 | 2009-08-18 | Xention Limited | Thieno[2,3-B] pyridines as potassium channel inhibitors |
GB0512429D0 (en) * | 2005-06-17 | 2005-07-27 | Smithkline Beecham Corp | Novel compound |
AU2006276292B2 (en) * | 2005-07-22 | 2010-09-16 | Merck Sharp & Dohme Corp. | Potassium channel inhibitors |
GB0525164D0 (en) | 2005-12-09 | 2006-01-18 | Xention Discovery Ltd | Compounds |
NZ572231A (en) * | 2006-04-27 | 2010-12-24 | Sanofi Aventis Deutschland | Inhibitors of the task-1 and task-3 ion channel |
TW200845991A (en) | 2007-01-12 | 2008-12-01 | Smithkline Beecham Corp | N-substituted glycine derivatives: hydroxylase inhibitors |
CL2008000986A1 (en) * | 2007-04-06 | 2008-10-17 | Neurocrine Biosciences Inc | COMPOUND DERIVED FROM NITROGEN HETEROCICLES, GnRH RECEPTOR AGONISTS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUND; AND USE TO TREAT AN AFFECTION RELATED TO SEX HORMONES, ENDOMETRIOSIS, DISMENORREA, OV DISEASE |
PA8775801A1 (en) | 2007-04-06 | 2009-05-15 | Neurocrine Biosciences Inc | ANTIGONIST OF THE RECEIVER OF GONADOTROPINE LIBERATING HORMONE AND PROCEDURES RELATED TO THEMSELVES |
GB0815782D0 (en) | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
GB0815784D0 (en) | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
GB0815781D0 (en) | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
GB201105659D0 (en) | 2011-04-01 | 2011-05-18 | Xention Ltd | Compounds |
NO3175985T3 (en) | 2011-07-01 | 2018-04-28 | ||
CA2862670A1 (en) | 2012-01-27 | 2013-08-01 | Gilead Sciences, Inc. | Combination therapies using late sodium ion channel blockers and potassium ion channel blockers |
TWI773657B (en) | 2015-12-18 | 2022-08-11 | 美商亞德利克斯公司 | Substituted 4-phenyl pyridine compounds as non-systemic tgr5 agonists |
CN107573292B (en) * | 2017-09-04 | 2022-06-24 | 江苏艾立康医药科技有限公司 | Pyrazine derivatives acting on prolyl hydroxylase |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19675036I2 (en) * | 1990-02-19 | 2004-10-21 | Novartis Ag | Acyl compounds. |
GB9220137D0 (en) * | 1992-09-23 | 1992-11-04 | Pfizer Ltd | Therapeutic agents |
WO1995001326A1 (en) * | 1993-06-30 | 1995-01-12 | The Wellcome Foundation Limited | Anti-atherosclerotic diaryl compounds |
GB9416972D0 (en) * | 1994-08-23 | 1994-10-12 | Smithkline Beecham Plc | Carbon side chain/indole/indolene |
DE4430638A1 (en) * | 1994-08-29 | 1996-03-07 | Bayer Ag | Use of substituted 4-phenyl-6-amino-nicotinic acid derivatives as a medicament |
DE4432101A1 (en) * | 1994-09-09 | 1996-03-14 | Hoechst Ag | Amino acid-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic agent, and medicament containing them |
US5670504A (en) | 1995-02-23 | 1997-09-23 | Merck & Co. Inc. | 2,6-diaryl pyridazinones with immunosuppressant activity |
US6083986A (en) * | 1996-07-26 | 2000-07-04 | Icagen, Inc. | Potassium channel inhibitors |
US5935945A (en) | 1996-10-31 | 1999-08-10 | Merck & Co., Inc. | Methods of treating or preventing cardiac arrhythmia |
US5969017A (en) | 1996-10-31 | 1999-10-19 | Merck & Co., Inc. | Methods of treating or preventing cardiac arrhythmia |
KR100241350B1 (en) * | 1997-10-27 | 2000-02-01 | 정선종 | Electronic certificate paper generation method |
US6333337B1 (en) * | 1998-01-27 | 2001-12-25 | Icagen, Inc. | Potassium channel inhibitors |
JP2002523451A (en) * | 1998-09-01 | 2002-07-30 | ブリストル−マイヤーズ スクイブ カンパニー | Potassium channel inhibitors and methods |
WO2000015603A1 (en) * | 1998-09-11 | 2000-03-23 | Ajinomoto Co., Inc. | Benzene derivatives and medicinal use thereof |
DE19947457A1 (en) * | 1999-10-02 | 2001-04-05 | Aventis Pharma Gmbh | New 2'-aminomethyl-biphenyl-2-carboxamide derivatives, are potassium channel blockers especially useful for treating re-entry or supraventricular arrhythmia or atrial fibrillation or flutter |
-
2000
- 2000-11-30 DE DE10059418A patent/DE10059418A1/en not_active Withdrawn
-
2001
- 2001-11-17 EE EEP200300183A patent/EE05240B1/en not_active IP Right Cessation
- 2001-11-17 BR BR0115769-8A patent/BR0115769A/en not_active Application Discontinuation
- 2001-11-17 PT PT01989479T patent/PT1339675E/en unknown
- 2001-11-17 AU AU2002227931A patent/AU2002227931B2/en not_active Ceased
- 2001-11-17 RU RU2003119153/04A patent/RU2278858C2/en not_active IP Right Cessation
- 2001-11-17 JP JP2002546507A patent/JP4051283B2/en not_active Expired - Fee Related
- 2001-11-17 NZ NZ526177A patent/NZ526177A/en unknown
- 2001-11-17 KR KR1020037007255A patent/KR100968056B1/en not_active IP Right Cessation
- 2001-11-17 CZ CZ20031502A patent/CZ301631B6/en not_active IP Right Cessation
- 2001-11-17 IL IL15609701A patent/IL156097A0/en unknown
- 2001-11-17 AU AU2793102A patent/AU2793102A/en active Pending
- 2001-11-17 DE DE50105386T patent/DE50105386D1/en not_active Expired - Lifetime
- 2001-11-17 ES ES01989479T patent/ES2236341T3/en not_active Expired - Lifetime
- 2001-11-17 SK SK653-2003A patent/SK286708B6/en not_active IP Right Cessation
- 2001-11-17 CA CA2430273A patent/CA2430273C/en not_active Expired - Fee Related
- 2001-11-17 CN CNB01819740XA patent/CN1290825C/en not_active Expired - Fee Related
- 2001-11-17 MX MXPA03004386A patent/MXPA03004386A/en active IP Right Grant
- 2001-11-17 RS YUP-376/03A patent/RS50403B/en unknown
- 2001-11-17 AT AT01989479T patent/ATE289292T1/en active
- 2001-11-17 HU HU0303317A patent/HUP0303317A3/en unknown
- 2001-11-17 WO PCT/EP2001/013294 patent/WO2002044137A1/en active IP Right Grant
- 2001-11-17 EP EP01989479A patent/EP1339675B1/en not_active Expired - Lifetime
- 2001-11-17 PL PL362700A patent/PL206245B1/en not_active IP Right Cessation
- 2001-11-28 TW TW090129358A patent/TWI254039B/en not_active IP Right Cessation
- 2001-11-28 AR ARP010105540A patent/AR031430A1/en unknown
- 2001-11-29 US US09/995,771 patent/US6605625B2/en not_active Expired - Fee Related
-
2003
- 2003-05-20 ZA ZA200303893A patent/ZA200303893B/en unknown
- 2003-05-25 IL IL156097A patent/IL156097A/en not_active IP Right Cessation
- 2003-05-28 NO NO20032438A patent/NO328599B1/en not_active IP Right Cessation
- 2003-05-29 HR HR20030436A patent/HRP20030436B1/en not_active IP Right Cessation
- 2003-06-04 US US10/453,646 patent/US6924392B2/en not_active Expired - Fee Related
-
2004
- 2004-06-16 HK HK04104352A patent/HK1061231A1/en not_active IP Right Cessation
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