AU2001263139A1 - Novel synthesis of heteroarylamine intermediate compounds - Google Patents

Novel synthesis of heteroarylamine intermediate compounds

Info

Publication number
AU2001263139A1
AU2001263139A1 AU2001263139A AU6313901A AU2001263139A1 AU 2001263139 A1 AU2001263139 A1 AU 2001263139A1 AU 2001263139 A AU2001263139 A AU 2001263139A AU 6313901 A AU6313901 A AU 6313901A AU 2001263139 A1 AU2001263139 A1 AU 2001263139A1
Authority
AU
Australia
Prior art keywords
heteroarylamine
intermediate compounds
novel synthesis
novel
synthesis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001263139A
Inventor
Suresh R Kapadia
Jinhua J. Song
Nathan K. Yee
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharmaceuticals Inc
Original Assignee
BOEHRINGER INGELHEIM PHARMA
Boehringer Ingelheim Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BOEHRINGER INGELHEIM PHARMA, Boehringer Ingelheim Pharmaceuticals Inc filed Critical BOEHRINGER INGELHEIM PHARMA
Publication of AU2001263139A1 publication Critical patent/AU2001263139A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Disclosed are novel 2-(5-halopyridyl) and 2-(5-halopyrimidinyl) magnesium halides, processes of making and their use in the efficient synthesis in their respective 5-halo-2-substituted pyridines and pyrimidines.
AU2001263139A 2000-05-23 2001-05-23 Novel synthesis of heteroarylamine intermediate compounds Abandoned AU2001263139A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20632700P 2000-05-23 2000-05-23
US60206327 2000-05-23
PCT/US2001/015665 WO2001090072A1 (en) 2000-05-23 2001-05-15 Novel synthesis of heteroarylamine intermediate compounds

Publications (1)

Publication Number Publication Date
AU2001263139A1 true AU2001263139A1 (en) 2001-12-03

Family

ID=22765881

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001263139A Abandoned AU2001263139A1 (en) 2000-05-23 2001-05-23 Novel synthesis of heteroarylamine intermediate compounds

Country Status (8)

Country Link
US (5) US6635767B2 (en)
EP (1) EP1409460B1 (en)
AT (1) ATE461917T1 (en)
AU (1) AU2001263139A1 (en)
CA (1) CA2424916C (en)
DE (1) DE60141654D1 (en)
ES (1) ES2340361T3 (en)
WO (1) WO2001090072A1 (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2435446A1 (en) 2001-02-15 2002-08-29 Boehringer Ingelheim Pharmaceuticals, Inc. Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
GB2375969A (en) 2001-05-31 2002-12-04 Nokia Corp Electronic gaming
JP2006507346A (en) * 2002-11-22 2006-03-02 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド Preparation of aryl intermediate compounds using trialkylmagnesate reagents
US7034157B2 (en) * 2003-10-23 2006-04-25 Fina Technology, Inc. Catalyst components, process for their preparation and their use as catalyst components in polymerization of olefins
US7081506B2 (en) * 2003-10-23 2006-07-25 Fina Technology, Inc. Ethylene polymerization employing bis-imino pyridinyl transition metal catalyst components
GB0411951D0 (en) * 2004-05-28 2004-06-30 Lucite Int Uk Ltd Carbonylation of ester
RU2006147280A (en) 2004-07-19 2008-08-27 Пфайзер Продактс Инк. (Us) OBTAINING NEW SUBSTITUTED HALOGENOARENE COMPOUNDS
US7714127B2 (en) * 2005-10-06 2010-05-11 Boehringer Ingelheim Pharmaceuticals, Inc. Process for making heteroaryl amine intermediate compounds
US8420577B2 (en) * 2008-10-21 2013-04-16 Baker Hughes Incorporated Methods of making polyboronic compounds and compositions related thereto
US9534167B2 (en) 2008-10-21 2017-01-03 Baker Hughes Incorporated Fracturing method using polyboronic compound
US8389763B2 (en) * 2008-10-21 2013-03-05 Bj Services Company Methods of making polyboronic compounds and compositions related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2151467T3 (en) 1997-05-23 2005-03-01 Bayer Corporation ARILURES FOR THE TREATMENT OF INFLAMMATORY OR IMMUNOMODULATING DISEASES.
DE60014603T2 (en) * 1999-03-12 2006-02-16 Boehringer Ingelheim Pharmaceuticals, Inc., Ridgefield Heterocyclic urea and related compounds as anti-inflammatory agents

Also Published As

Publication number Publication date
DE60141654D1 (en) 2010-05-06
ATE461917T1 (en) 2010-04-15
US6590099B2 (en) 2003-07-08
US20010053850A1 (en) 2001-12-20
CA2424916C (en) 2009-04-28
US20020049333A1 (en) 2002-04-25
US6635767B2 (en) 2003-10-21
EP1409460B1 (en) 2010-03-24
EP1409460A1 (en) 2004-04-21
US20020068826A1 (en) 2002-06-06
WO2001090072A1 (en) 2001-11-29
US6593471B2 (en) 2003-07-15
ES2340361T3 (en) 2010-06-02
US6613909B2 (en) 2003-09-02
CA2424916A1 (en) 2001-11-29
US20020077475A1 (en) 2002-06-20
US20020045754A1 (en) 2002-04-18

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