ATE546138T1 - Verwendung von steroid-sulfatase-inhibitoren zur behandlung von vorzeitigen wehen - Google Patents

Verwendung von steroid-sulfatase-inhibitoren zur behandlung von vorzeitigen wehen

Info

Publication number
ATE546138T1
ATE546138T1 AT09786717T AT09786717T ATE546138T1 AT E546138 T1 ATE546138 T1 AT E546138T1 AT 09786717 T AT09786717 T AT 09786717T AT 09786717 T AT09786717 T AT 09786717T AT E546138 T1 ATE546138 T1 AT E546138T1
Authority
AT
Austria
Prior art keywords
steroid sulfatase
premature labor
sulfatase inhibitors
treat premature
present
Prior art date
Application number
AT09786717T
Other languages
English (en)
Inventor
Ernest Loumaye
Valerie Cayron-Elizondo
Jean-Pierre Gotteland
Original Assignee
Preglem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Preglem Sa filed Critical Preglem Sa
Application granted granted Critical
Publication of ATE546138T1 publication Critical patent/ATE546138T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06Antiabortive agents; Labour repressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pyrane Compounds (AREA)
AT09786717T 2008-07-28 2009-07-27 Verwendung von steroid-sulfatase-inhibitoren zur behandlung von vorzeitigen wehen ATE546138T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8408208P 2008-07-28 2008-07-28
EP08161229A EP2149371A1 (de) 2008-07-28 2008-07-28 Verwendung von Steroid-Sulfatase-Hemmern zur Behandlung von Frühgeburtsleiden
PCT/IB2009/053256 WO2010013187A1 (en) 2008-07-28 2009-07-27 Use of steroid sulfatase inhibitors for the treatment of preterm labor

Publications (1)

Publication Number Publication Date
ATE546138T1 true ATE546138T1 (de) 2012-03-15

Family

ID=39791507

Family Applications (1)

Application Number Title Priority Date Filing Date
AT09786717T ATE546138T1 (de) 2008-07-28 2009-07-27 Verwendung von steroid-sulfatase-inhibitoren zur behandlung von vorzeitigen wehen

Country Status (14)

Country Link
US (1) US20110118224A1 (de)
EP (3) EP2149371A1 (de)
JP (1) JP2011529485A (de)
KR (2) KR20160060791A (de)
AT (1) ATE546138T1 (de)
AU (1) AU2009277972B2 (de)
BR (1) BRPI0916404A2 (de)
CA (1) CA2728795C (de)
DK (2) DK2484351T3 (de)
ES (2) ES2570879T3 (de)
HU (1) HUE027778T2 (de)
PL (2) PL2323646T3 (de)
PT (1) PT2323646E (de)
WO (1) WO2010013187A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114728013A (zh) * 2019-09-23 2022-07-08 斯坦福大学托管董事会 延长妊娠以及月经或妊娠的并发症的治疗方法
US12426782B2 (en) 2020-11-06 2025-09-30 The Board Of Trustees Of The Leland Stanford Junior University Systems and temporal alignment methods for evaluation of gestational age and time to delivery
US20240082208A1 (en) * 2021-01-08 2024-03-14 Industry-Academic Cooperation Foundation, Yonsei University Antiviral pharmaceutical composition comprising steroid sulfatase inhibitor
EP4313061A4 (de) * 2021-03-31 2025-03-05 The Board of Trustees of the Leland Stanford Junior University Formulierungen zur verlängerung der gestation und für komplikationen der menstruation oder gestation
WO2024259428A2 (en) * 2023-06-16 2024-12-19 The Board Of Trustees Of The Leland Stanford Junior University Estrogenic compounds and formulations for gestation-related complications

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6476011B1 (en) * 1991-08-28 2002-11-05 Sterix Limited Methods for introducing an estrogenic compound
US6011024A (en) * 1991-08-28 2000-01-04 Imperial College Of Science Technology & Medicine Steroid sulphatase inhibitors
GB9118478D0 (en) * 1991-08-29 1991-10-16 Imperial College Steroid sulphatase inhibitors
DE4429397C2 (de) * 1994-08-09 2003-11-20 Jenapharm Gmbh Estra-1,3,5(10)-trien-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
GB9422777D0 (en) 1994-11-11 1995-01-04 Imperial College Assay
US5705495A (en) * 1995-10-19 1998-01-06 Jenapharm Gmbh & Co. Kg. Sulfamate derivatives of 1,3,5(10)-estratriene derivatives, methods for their production and pharmaceuticals containing these compounds
US6642220B1 (en) * 1996-12-05 2003-11-04 Sterix Limited Compounds that inhibit oestrone sulphatase; compositions thereof; and methods employing the same
GB2331987B (en) * 1997-12-04 2002-11-27 Imperial College Polycyclic sulphamate inhibitors of oestrone sulphatase
US6585954B1 (en) * 1998-03-26 2003-07-01 Kyowa Hakko Kogyo Co., Ltd. Method for searching steroid sulfatase inhibitors
DE60209811T2 (de) 2001-10-18 2006-10-12 Sterix Ltd., Slough Steroidale verbindungen zur inhibierung von steroidsulfatasen
AU2003272964A1 (en) * 2002-10-09 2004-05-04 Kyowa Hakko Kogyo Co., Ltd. Remedy for hormone-dependent cancer
JP4719144B2 (ja) 2003-03-24 2011-07-06 ステリックス リミテッド ステロイドスルファターゼのインヒビターとしてのエストロゲン誘導体
GB0511190D0 (en) * 2005-06-01 2005-07-06 Sterix Ltd Use
GB0604142D0 (en) 2006-03-01 2006-04-12 Sterix Ltd Compound

Also Published As

Publication number Publication date
DK2484351T3 (en) 2016-05-17
CA2728795A1 (en) 2010-02-04
PL2323646T3 (pl) 2012-07-31
AU2009277972B2 (en) 2014-06-12
HK1170952A1 (en) 2013-03-15
AU2009277972A1 (en) 2010-02-04
PT2323646E (pt) 2012-04-27
ES2382768T3 (es) 2012-06-13
JP2011529485A (ja) 2011-12-08
US20110118224A1 (en) 2011-05-19
CA2728795C (en) 2018-03-27
WO2010013187A1 (en) 2010-02-04
EP2323646B1 (de) 2012-02-22
KR20160060791A (ko) 2016-05-30
EP2323646A1 (de) 2011-05-25
DK2323646T3 (da) 2012-05-07
BRPI0916404A2 (pt) 2016-02-16
PL2484351T3 (pl) 2016-08-31
EP2484351A1 (de) 2012-08-08
KR20110038070A (ko) 2011-04-13
EP2149371A1 (de) 2010-02-03
HUE027778T2 (en) 2016-11-28
EP2484351B1 (de) 2016-02-24
ES2570879T3 (es) 2016-05-20

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