ATE542812T1 - SUBSTITUTED INDOLYLALKYLAMINO DERIVATIVES AS NEW INHIBITORS OF HISTONE DEACETYLASE - Google Patents
SUBSTITUTED INDOLYLALKYLAMINO DERIVATIVES AS NEW INHIBITORS OF HISTONE DEACETYLASEInfo
- Publication number
- ATE542812T1 ATE542812T1 AT05767934T AT05767934T ATE542812T1 AT E542812 T1 ATE542812 T1 AT E542812T1 AT 05767934 T AT05767934 T AT 05767934T AT 05767934 T AT05767934 T AT 05767934T AT E542812 T1 ATE542812 T1 AT E542812T1
- Authority
- AT
- Austria
- Prior art keywords
- indolylalkylamino
- derivatives
- substituted
- histone deacetylase
- new inhibitors
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
This invention comprises the novel compounds of formula (I) wherein R, R, R, X and Y have defined meanings, having histone deacelylase inhibiting enzymatic activity; their preparation, compositions containing them and their, use as drugs.(I)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04077172 | 2004-07-28 | ||
| US59218204P | 2004-07-29 | 2004-07-29 | |
| PCT/EP2005/053612 WO2006010750A1 (en) | 2004-07-28 | 2005-07-25 | Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE542812T1 true ATE542812T1 (en) | 2012-02-15 |
Family
ID=34928411
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05767934T ATE542812T1 (en) | 2004-07-28 | 2005-07-25 | SUBSTITUTED INDOLYLALKYLAMINO DERIVATIVES AS NEW INHIBITORS OF HISTONE DEACETYLASE |
Country Status (10)
| Country | Link |
|---|---|
| CN (1) | CN1993353B (en) |
| AT (1) | ATE542812T1 (en) |
| DK (1) | DK1781639T3 (en) |
| ES (1) | ES2381117T3 (en) |
| ME (1) | ME01444B (en) |
| PT (1) | PT1781639E (en) |
| RS (1) | RS52304B (en) |
| SI (1) | SI1781639T1 (en) |
| UA (1) | UA93352C2 (en) |
| ZA (1) | ZA200700764B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115487191B (en) * | 2016-02-22 | 2024-05-14 | 中国科学院上海巴斯德研究所 | Quisinostat, a novel high-efficiency antimalarial drug |
| CN107721980B (en) * | 2017-08-25 | 2019-07-12 | 南京医科大学 | The weary oxygen targeted prodrug and its application of a kind of fluorouracil and Quisinosta |
| CN112485233B (en) * | 2020-11-03 | 2022-08-26 | 山东师范大学 | Nano sensor for detecting deacetylase and detection method and application thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE398105T1 (en) * | 2002-03-13 | 2008-07-15 | Janssen Pharmaceutica Nv | CARBONYLAMINO DERIVATIVES AS NEW INHIBITORS OF HISTONE DEACETYLASE |
-
2005
- 2005-07-25 SI SI200531516T patent/SI1781639T1/en unknown
- 2005-07-25 RS RS20120165A patent/RS52304B/en unknown
- 2005-07-25 ME MEP-2012-53A patent/ME01444B/en unknown
- 2005-07-25 DK DK05767934.2T patent/DK1781639T3/en active
- 2005-07-25 ES ES05767934T patent/ES2381117T3/en active Active
- 2005-07-25 CN CN2005800256290A patent/CN1993353B/en active Active
- 2005-07-25 PT PT05767934T patent/PT1781639E/en unknown
- 2005-07-25 AT AT05767934T patent/ATE542812T1/en active
- 2005-07-25 UA UAA200614022A patent/UA93352C2/en unknown
-
2007
- 2007-01-26 ZA ZA200700764A patent/ZA200700764B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2381117T3 (en) | 2012-05-23 |
| DK1781639T3 (en) | 2012-05-14 |
| RS52304B (en) | 2012-12-31 |
| CN1993353B (en) | 2010-12-01 |
| CN1993353A (en) | 2007-07-04 |
| UA93352C2 (en) | 2011-02-10 |
| ZA200700764B (en) | 2008-09-25 |
| PT1781639E (en) | 2012-05-02 |
| SI1781639T1 (en) | 2012-06-29 |
| ME01444B (en) | 2013-12-20 |
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