ATE541573T1 - Pharmazeutische zusammensetzung enthaltend lapatinib - Google Patents

Pharmazeutische zusammensetzung enthaltend lapatinib

Info

Publication number
ATE541573T1
ATE541573T1 AT09782127T AT09782127T ATE541573T1 AT E541573 T1 ATE541573 T1 AT E541573T1 AT 09782127 T AT09782127 T AT 09782127T AT 09782127 T AT09782127 T AT 09782127T AT E541573 T1 ATE541573 T1 AT E541573T1
Authority
AT
Austria
Prior art keywords
pharmaceutical composition
composition containing
lapatinib
containing lapatinib
composition
Prior art date
Application number
AT09782127T
Other languages
English (en)
Inventor
Katrin Rimkus
Frank Muskulus
Sandra Brueck
Jana Paetz
Original Assignee
Ratiopharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39884161&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE541573(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ratiopharm Gmbh filed Critical Ratiopharm Gmbh
Application granted granted Critical
Publication of ATE541573T1 publication Critical patent/ATE541573T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
AT09782127T 2008-08-25 2009-08-24 Pharmazeutische zusammensetzung enthaltend lapatinib ATE541573T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08014984A EP2158913A1 (de) 2008-08-25 2008-08-25 Pharmazeutische Zusammensetzung mit N-[3-chlor-4-(3-fluorophenyl)methoxy)phenyl)6-(5(((2-(methylsulfonyl)ethyl)amino)methyl)-2-furyl)-4-chinazolinamin
PCT/EP2009/060890 WO2010023188A1 (en) 2008-08-25 2009-08-24 Pharmaceutical composition comprising n-[3-chloro-4-[(3- fluorophenyl)methoxy]phenyl]-6-[5[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furyl]-4- quinazolinamine

Publications (1)

Publication Number Publication Date
ATE541573T1 true ATE541573T1 (de) 2012-02-15

Family

ID=39884161

Family Applications (1)

Application Number Title Priority Date Filing Date
AT09782127T ATE541573T1 (de) 2008-08-25 2009-08-24 Pharmazeutische zusammensetzung enthaltend lapatinib

Country Status (7)

Country Link
US (1) US8586091B2 (de)
EP (2) EP2158913A1 (de)
AT (1) ATE541573T1 (de)
CA (1) CA2735206C (de)
ES (1) ES2378134T3 (de)
RU (1) RU2011107140A (de)
WO (1) WO2010023188A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2958552B1 (de) 2013-02-19 2017-06-21 Hexal AG Pharmazeutische zusammensetzung mit n-[3-chlor-4-(3-fluorbenzyloxy)phenyl]-6-[5({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]chinazolin-4-amin oder ein pharmazeutisch akzeptables salz, solvat oder solvatisiertes salz daraus
WO2018137020A1 (en) 2017-01-25 2018-08-02 Pacey Medtech Ltd. Distributed pressure fenestrated urethral compression apparatus for treatment of male urinary sphincter deficiency with preservation of blood flow
EP3687500A1 (de) * 2017-09-29 2020-08-05 Crititech, Inc. Glucocorticoidpartikel und deren verwendung
TWI832871B (zh) 2018-06-29 2024-02-21 美商英塞特公司 Axl/mer 抑制劑之調配物
EP3846787A4 (de) * 2018-09-03 2022-05-25 BDR Pharmaceuticals International Private Limited Neuartige zusammensetzung von lapatinib in oraler fester darreichungsform und verfahren zu ihrer herstellung

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8623557D0 (en) * 1986-10-01 1986-11-05 Boots Co Plc Therapeutic agents
RS49779B (sr) 1998-01-12 2008-06-05 Glaxo Group Limited, Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze
KR100815681B1 (ko) 2000-06-30 2008-03-20 글락소 그룹 리미티드 퀴나졸린 디토실레이트 염 화합물
ES2233227T1 (es) * 2003-03-26 2005-06-16 Teva Pharmaceutical Industries Ltd. Procedimiento para la preparacion de ingredientes farmaceuticos activos con un area superficial especifica.
US20080026067A1 (en) 2004-04-20 2008-01-31 Kuwabe Shin-Itsu Method for Increasing Specific Surface Area of Slightly Soluble Drug
WO2005120504A2 (en) 2004-06-03 2005-12-22 Smithkline Beecham (Cork) Limited Cancer treatment method
EP2277595A3 (de) 2004-06-24 2011-09-28 Novartis Vaccines and Diagnostics, Inc. Verbindungen zur Immunopotenzierung
ES2426007T3 (es) 2004-12-17 2013-10-18 Smithkline Beecham (Cork) Limited Método para el tratamiento del cáncer
KR20080002939A (ko) 2005-04-12 2008-01-04 엘란 파마 인터내셔널 리미티드 나노입자형 퀴나졸린 유도체 제제
KR101356748B1 (ko) 2005-04-19 2014-02-06 스미스클라인 비이참 (코르크) 리미티드 약제 조성물
WO2007143483A2 (en) * 2006-06-01 2007-12-13 Smithkline Beecham Corporation Combination of pazopanib and lapatinib for treating cancer
EP2088862A4 (de) * 2006-11-28 2009-12-02 Smithkline Beecham Cork Ltd Krebsbehandlungsverfahren
EP2158912A1 (de) * 2008-08-25 2010-03-03 Ratiopharm GmbH Pharmazeutische Zusammensetzung mit N-[3-chlor-4-(3-fluorophenyl)methoxy)phenyl)6-(5(((2-(methylsulfonyl)ethyl)amino)methyl)-2-furyl)-4-chinazolinamin
CA2740977A1 (en) * 2008-11-03 2010-06-03 Natco Pharma Limited A novel process for the preparation of lapatinib and its pharmaceutically acceptable salts

Also Published As

Publication number Publication date
US20110305762A1 (en) 2011-12-15
US8586091B2 (en) 2013-11-19
CA2735206A1 (en) 2010-03-04
RU2011107140A (ru) 2012-09-27
WO2010023188A1 (en) 2010-03-04
ES2378134T3 (es) 2012-04-09
EP2320902A1 (de) 2011-05-18
EP2158913A1 (de) 2010-03-03
EP2320902B1 (de) 2012-01-18
CA2735206C (en) 2016-11-01

Similar Documents

Publication Publication Date Title
CL2009000349A1 (es) Compuestos derivados de 4,5-dihidro-oxazol-2-ilamina; procedimiento de preparacion; composicion farmaceutica; y su uso para el tratamiento de la enfermedad de alzheimer.
JO2973B1 (en) Fumarate salt for (alpha-beta-R) -6-bromo-alpha-[2- (methylamino) ethyl-2-methoxy-alpha-1-naphthalenyl-beta-phenyl-3-quinoline ethanol
CY1119474T1 (el) Κρυσταλλικες μορφες 5-χλωρο-ν2-(2-ισοπροποξυ-5-μεθυλ-4-πιπεριδιν-4-υλ-φαινυλ)-ν4[2-(προπανο-2-σουλφονυλ)-φαινυλ]-πυριμιδιν-2,4-διαμινης
EA201500430A1 (ru) Соединения боронатного эфира и его фармацевтические составы
BRPI0923728A2 (pt) "método de preparação de compostos de di-hidroindeno amida, suas composições farmacêuticas contendo esses compostos e uso como inibidor de proteína quinase".
CY1109010T1 (el) γ-ΚΡΥΣΤΑΛΛΙΚΗ ΜΟΡΦΗ ΤΗΣ ΥΔΡΟΧΛΩΡΙΚΗΣ ΙΒΑΒΡΑΔΙΝΗΣ, ΜΕΘΟΔΟΣ ΠΑΡΑΣΚΕΥΗΣ ΤΗΣ ΚΑΙ ΦΑΡΜΑΚΕΥΤΙΚΕΣ ΣΥΝΘΕΣΕΙΣ ΠΟΥ ΤΗΝ ΠΕΡΙΕΧΟΥΝ
CY1109998T1 (el) Ενδυναμωτες υποδοχεων γλουταμινικου
BRPI0906064A2 (pt) "peptídeo, processo para obtenção de um peptídeo de fórmula geral (i), composição cosmética ou farmacêutica e uso de um peptídeo de fórmula geral (i)"
FR16C1025I1 (fr) Sel de 4-[[4-[[4-(2-Cyanoethenyl)-2,6-dimethylphenyl]amino]-2-Pyrimidinyl]amino]benzonitrile
EA200970500A1 (ru) СОЕДИНЕНИЯ ТЕТРАГИДРОЦИКЛОПЕНТА[b]ИНДОЛА В КАЧЕСТВЕ МОДУЛЯТОРОВ РЕЦЕПТОРА АНДРОГЕНОВ
HK1113790A1 (en) Selurampanel
NO20071299L (no) Vedvarende frigivelse farmasoytisk sammensetning av tolterodine
BR112014011981A2 (pt) formulações farmacêuticas
ATE541573T1 (de) Pharmazeutische zusammensetzung enthaltend lapatinib
EA201001747A1 (ru) Бензоксазиноновые производные, действующие в качестве агониста бета-2-адренорецептора, для лечения респираторных расстройств
EA200801614A1 (ru) Фармацевтическая композиция, содержащая монтелукаст
MY150988A (en) Novel derivatives of ( bridged piperazinyl)-1-alkanone and use thereof as p75 inhibitors
WO2007076091A3 (en) Treatment of viral infections using a tissue factor inhibitor
ATE460934T1 (de) Pharmazeutische zubereitungen von ciprofloxacin
ATE496899T1 (de) Tetrahydro- und dihydrochinazolinone
GB2418855B (en) Use of ethyl lactate as an excipient for pharmaceutical compositions
UA92469C2 (en) Fumarate of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl amino benzonitrile
CR9032A (es) Fumarato de 4-((4-((4-(2-cianoetenil)-2,6-dimetilfenil)amino-2- pirimidinil)amino)benzonitrilo
BRPI1006611A2 (pt) "n' -(metilsulfonil)-1 - [tiofen-2-il]-1, 4-dihidropiridina -3- carbohidrazida, composto de fórmula (i), composição farmacêutica, método de tratamento de uma neuropatia e uso de um composto"
EA200901205A1 (ru) Фармацевтическая композиция, содержащая соль розиглитазона