ATE523495T1 - Substituierte pyrazolinverbindungen, deren herstellung und verwendung als medikamente - Google Patents
Substituierte pyrazolinverbindungen, deren herstellung und verwendung als medikamenteInfo
- Publication number
- ATE523495T1 ATE523495T1 AT06762612T AT06762612T ATE523495T1 AT E523495 T1 ATE523495 T1 AT E523495T1 AT 06762612 T AT06762612 T AT 06762612T AT 06762612 T AT06762612 T AT 06762612T AT E523495 T1 ATE523495 T1 AT E523495T1
- Authority
- AT
- Austria
- Prior art keywords
- preparation
- medications
- substituted pyrazoline
- pyrazoline compounds
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05384005A EP1757587A1 (de) | 2005-07-15 | 2005-07-15 | Substituierte Pyrazolinderivate, ihre Herstellung und Verwendung als Arzneimittel |
US70548105P | 2005-08-05 | 2005-08-05 | |
PCT/EP2006/006969 WO2007009695A1 (en) | 2005-07-15 | 2006-07-15 | Substituted pyrazoline compounds, their preparation and use as medicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE523495T1 true ATE523495T1 (de) | 2011-09-15 |
Family
ID=35311564
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT06762612T ATE523495T1 (de) | 2005-07-15 | 2006-07-15 | Substituierte pyrazolinverbindungen, deren herstellung und verwendung als medikamente |
Country Status (7)
Country | Link |
---|---|
US (1) | US20070015810A1 (de) |
EP (2) | EP1757587A1 (de) |
AT (1) | ATE523495T1 (de) |
ES (1) | ES2372307T3 (de) |
PE (1) | PE20070246A1 (de) |
TW (1) | TW200745043A (de) |
WO (1) | WO2007009695A1 (de) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200533657A (en) * | 2004-02-17 | 2005-10-16 | Esteve Labor Dr | Substituted pyrazoline compounds, their preparation and use as medicaments |
EP1743892A1 (de) * | 2005-07-15 | 2007-01-17 | Laboratorios del Dr. Esteve S.A. | Substituierte Pyrazolin Verbindungen, deren Herstellung und Verwendung als Medikament |
CA2666193A1 (en) | 2006-08-08 | 2008-02-14 | Sanofi-Aventis | Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
EP2042175A1 (de) * | 2007-09-21 | 2009-04-01 | Laboratorios del Dr. Esteve S.A. | Dosierungsschemata von CB1-Rezeptor-Liganden für die Behandlung von Fettleibigkeit |
WO2009097995A1 (de) * | 2008-02-07 | 2009-08-13 | Sanofi-Aventis | Neue phenyl-substituierte imidazolidine, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
EP2310372B1 (de) | 2008-07-09 | 2012-05-23 | Sanofi | Heterocyclische Verbindungen, Verfahren zu ihrer Herstellung, Arzneimitteln mit diesen Verbindungen und ihre Verwendung |
EP2151234A1 (de) * | 2008-07-28 | 2010-02-10 | Laboratorios Del. Dr. Esteve, S.A. | Pharmazeutische Formulierung mit einer CB1-Rezeptorverbindung in einer festen Lösung und/oder festen Dispersion |
WO2010068601A1 (en) | 2008-12-08 | 2010-06-17 | Sanofi-Aventis | A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof |
EP2470552B1 (de) | 2009-08-26 | 2013-11-13 | Sanofi | Neuartige kristalline heteroaromatische Fluorglycosidhydrate, Pharmazeutika, die diese Verbindungen umfassen, und deren Verwendung |
EP2582709B1 (de) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
EP2683704B1 (de) | 2011-03-08 | 2014-12-17 | Sanofi | Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
WO2012120052A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
US8710050B2 (en) | 2011-03-08 | 2014-04-29 | Sanofi | Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
US8871758B2 (en) | 2011-03-08 | 2014-10-28 | Sanofi | Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof |
EP2683705B1 (de) | 2011-03-08 | 2015-04-22 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
JP2017028024A (ja) * | 2015-07-17 | 2017-02-02 | 富士通株式会社 | 部品搭載基板、部品内蔵基板、部品搭載基板の製造方法および部品内蔵基板の製造方法 |
WO2020237043A1 (en) * | 2019-05-22 | 2020-11-26 | President And Fellows Of Harvard College | Human tactile prepulse inhibition assay |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2613720B1 (fr) * | 1987-04-10 | 1990-01-19 | Esteve Labor Dr | Derives d'aryl-heteroaryl carbinols avec activite analgesique |
FR2742147B1 (fr) * | 1995-12-06 | 1998-02-27 | Esteve Labor Dr | Procede de separation de carbinols |
US20020156104A1 (en) * | 1997-06-13 | 2002-10-24 | Jerry L. Adams | Novel pyrazole and pyrazoline substituted compounds |
ES2130079B1 (es) * | 1997-07-10 | 2000-01-16 | Esteve Labor Dr | Resolucion de aminas |
ES2130083B1 (es) * | 1997-08-04 | 2000-01-16 | Esteve Labor Dr | Procedimiento para la obtencion de los enantiomeros de cizolirtina. |
ES2150353B1 (es) * | 1998-04-15 | 2001-07-01 | Esteve Labor Dr | Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos. |
ES2137138B1 (es) * | 1998-05-29 | 2000-09-16 | Esteve Labor Dr | Derivados de pirazolinas, su preparacion y su aplicacion como medicamentos. |
EP1177188B1 (de) * | 1999-05-12 | 2005-10-12 | Ortho-McNeil Pharmaceutical, Inc. | Pyrazolecarboxamide zur behandlung von fettleibigkeit und anderen erkrankungen |
ATE349439T1 (de) * | 2000-06-22 | 2007-01-15 | Pharmos Corp | Neue nicht psychotropische cannabinoide |
HUP0303070A2 (hu) * | 2000-08-01 | 2003-12-29 | Ono Pharmaceutical Co., Ltd. | 3,4-Dihidro-izokinolin-származékok és ezeket hatóanyagként tartalmazó gyógyszerkészítmények |
CN100366614C (zh) * | 2001-03-22 | 2008-02-06 | 索尔瓦药物有限公司 | 具有cb1-拮抗活性的4,5-二氢-1h-吡唑衍生物 |
ES2183720B1 (es) * | 2001-06-18 | 2004-01-16 | Esteve Labor Dr | Procedimiento para la preparacion de derivados de 1,5-diaril-3-trifluorometil-delta2-pirazolinas racemicas y enantiomericamente puras. |
ES2180449B1 (es) * | 2001-07-06 | 2004-01-16 | Esteve Labor Dr | Derivados de aril (o heteroaril) azolilcarbinoles para el tratamiento de la incontinencia urinaria. |
US6509367B1 (en) * | 2001-09-22 | 2003-01-21 | Virginia Commonwealth University | Pyrazole cannabinoid agonist and antagonists |
US7378428B2 (en) * | 2002-01-31 | 2008-05-27 | Ono Pharmaceutical Co., Ltd. | Nitrogen-containing bicyclic compounds and drugs containing the same as the active ingredient |
US20050137251A1 (en) * | 2002-03-18 | 2005-06-23 | Aaron Garzon | Dexanabinol and dexanabinol analogs regulate inflammation related genes |
CA2496164C (en) * | 2002-08-23 | 2010-11-09 | Chiron Corporation | Benzimidazole quinolinones and uses thereof |
SE0300010D0 (sv) * | 2003-01-07 | 2003-01-07 | Astrazeneca Ab | Novel Compounds |
US20060172019A1 (en) * | 2003-03-07 | 2006-08-03 | Ralston Stuart H | Cannabinoid receptor inverse agonists and neutral antagonists as therapeutic agents for the treatment of bone disorders |
WO2005012256A1 (en) * | 2003-07-22 | 2005-02-10 | Astex Therapeutics Limited | 3, 4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators |
US7745476B2 (en) * | 2004-01-30 | 2010-06-29 | Solvay Pharmaceuticals B.V. | 1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity |
TW200533657A (en) * | 2004-02-17 | 2005-10-16 | Esteve Labor Dr | Substituted pyrazoline compounds, their preparation and use as medicaments |
ITMI20041033A1 (it) * | 2004-05-24 | 2004-08-24 | Neuroscienze S C A R L | Composti farmaceutici |
WO2006044556A2 (en) * | 2004-10-14 | 2006-04-27 | Galileo Pharmaceuticals, Inc. | Dual inhibitors of lipoxygenase for treating diabetes |
WO2006045799A2 (en) * | 2004-10-25 | 2006-05-04 | Solvay Pharmaceuticals Gmbh | Pharmaceutical compositions comprising cb1 cannabinoid receptor antagonists and potassium channel openers for the treatment of diabetes mellitus type i, obesity and related conditions |
-
2005
- 2005-07-15 EP EP05384005A patent/EP1757587A1/de not_active Withdrawn
-
2006
- 2006-07-14 US US11/457,691 patent/US20070015810A1/en not_active Abandoned
- 2006-07-14 PE PE2006000848A patent/PE20070246A1/es not_active Application Discontinuation
- 2006-07-14 TW TW095125886A patent/TW200745043A/zh unknown
- 2006-07-15 AT AT06762612T patent/ATE523495T1/de not_active IP Right Cessation
- 2006-07-15 EP EP06762612A patent/EP1910299B1/de not_active Not-in-force
- 2006-07-15 ES ES06762612T patent/ES2372307T3/es active Active
- 2006-07-15 WO PCT/EP2006/006969 patent/WO2007009695A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
EP1757587A1 (de) | 2007-02-28 |
ES2372307T3 (es) | 2012-01-18 |
PE20070246A1 (es) | 2007-05-30 |
TW200745043A (en) | 2007-12-16 |
US20070015810A1 (en) | 2007-01-18 |
EP1910299A1 (de) | 2008-04-16 |
WO2007009695A1 (en) | 2007-01-25 |
EP1910299B1 (de) | 2011-09-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |