ATE499358T1 - Synthese von piperazinen, piperidinen und verwandten verbindungen - Google Patents

Synthese von piperazinen, piperidinen und verwandten verbindungen

Info

Publication number
ATE499358T1
ATE499358T1 AT07813680T AT07813680T ATE499358T1 AT E499358 T1 ATE499358 T1 AT E499358T1 AT 07813680 T AT07813680 T AT 07813680T AT 07813680 T AT07813680 T AT 07813680T AT E499358 T1 ATE499358 T1 AT E499358T1
Authority
AT
Austria
Prior art keywords
piperazines
piperidines
synthesis
related compounds
compounds
Prior art date
Application number
AT07813680T
Other languages
English (en)
Inventor
Hugh Alfred Burgoon
Ramanaiah C Kanamarlapudi
Wenxue Wu
Original Assignee
Lexicon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lexicon Pharmaceuticals Inc filed Critical Lexicon Pharmaceuticals Inc
Application granted granted Critical
Publication of ATE499358T1 publication Critical patent/ATE499358T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
AT07813680T 2006-08-04 2007-08-02 Synthese von piperazinen, piperidinen und verwandten verbindungen ATE499358T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83567906P 2006-08-04 2006-08-04
PCT/US2007/075026 WO2008019279A2 (en) 2006-08-04 2007-08-02 Synthesis of piperazines, piperidines and related compounds

Publications (1)

Publication Number Publication Date
ATE499358T1 true ATE499358T1 (de) 2011-03-15

Family

ID=38828564

Family Applications (1)

Application Number Title Priority Date Filing Date
AT07813680T ATE499358T1 (de) 2006-08-04 2007-08-02 Synthese von piperazinen, piperidinen und verwandten verbindungen

Country Status (7)

Country Link
US (1) US7919618B2 (de)
EP (1) EP2084144B1 (de)
AR (1) AR062203A1 (de)
AT (1) ATE499358T1 (de)
DE (1) DE602007012748D1 (de)
TW (1) TW200815401A (de)
WO (1) WO2008019279A2 (de)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0611439A2 (pt) 2005-05-13 2010-09-08 Lexicon Pharmaceuticals Inc compostos multicìclicos e métodos para uso dos mesmos
US20060258691A1 (en) 2005-05-13 2006-11-16 Joseph Barbosa Methods and compositions for improving cognition
WO2008019276A2 (en) 2006-08-04 2008-02-14 Lexicon Pharmaceuticals, Inc. Solid forms of (3'-chlorobiphenyl-4-yl)(1-(pyrimidin-2-yl)piperidin-4-yl)methanone and methods of their use

Also Published As

Publication number Publication date
AR062203A1 (es) 2008-10-22
US7919618B2 (en) 2011-04-05
EP2084144B1 (de) 2011-02-23
TW200815401A (en) 2008-04-01
US20080177070A1 (en) 2008-07-24
DE602007012748D1 (de) 2011-04-07
WO2008019279A3 (en) 2008-04-03
EP2084144A2 (de) 2009-08-05
WO2008019279A2 (en) 2008-02-14

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties