ATE458482T1 - Verwendung von amino substituierten benzimidazolen - Google Patents

Verwendung von amino substituierten benzimidazolen

Info

Publication number
ATE458482T1
ATE458482T1 AT06723256T AT06723256T ATE458482T1 AT E458482 T1 ATE458482 T1 AT E458482T1 AT 06723256 T AT06723256 T AT 06723256T AT 06723256 T AT06723256 T AT 06723256T AT E458482 T1 ATE458482 T1 AT E458482T1
Authority
AT
Austria
Prior art keywords
amino substituted
substituted benzimidazoles
compounds
benzimidazoles
amino
Prior art date
Application number
AT06723256T
Other languages
German (de)
English (en)
Inventor
Elisabeth Defossa
Karl Schoenafinger
Gerhard Jaehne
Christian Buning
Georg Tschank
Ulrich Werner
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Application granted granted Critical
Publication of ATE458482T1 publication Critical patent/ATE458482T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT06723256T 2005-03-19 2006-03-07 Verwendung von amino substituierten benzimidazolen ATE458482T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005012875A DE102005012875B4 (de) 2005-03-19 2005-03-19 Verwendung von Amino substituierten 8-N-Benzimidazolen
PCT/EP2006/002057 WO2006099942A2 (de) 2005-03-19 2006-03-07 Verwendung von amino substituierten benzimidazolen

Publications (1)

Publication Number Publication Date
ATE458482T1 true ATE458482T1 (de) 2010-03-15

Family

ID=36933932

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06723256T ATE458482T1 (de) 2005-03-19 2006-03-07 Verwendung von amino substituierten benzimidazolen

Country Status (11)

Country Link
US (1) US8003668B2 (OSRAM)
EP (1) EP1863488B1 (OSRAM)
JP (1) JP2008533066A (OSRAM)
AT (1) ATE458482T1 (OSRAM)
AU (1) AU2006226639A1 (OSRAM)
BR (1) BRPI0608451A2 (OSRAM)
CA (1) CA2602236A1 (OSRAM)
DE (2) DE102005012875B4 (OSRAM)
IL (1) IL185807A0 (OSRAM)
MX (1) MX2007010836A (OSRAM)
WO (1) WO2006099942A2 (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2121626A1 (en) * 2006-12-15 2009-11-25 Pfizer Products Inc. Benzimidazole derivatives
NZ581889A (en) 2007-06-29 2011-05-27 Pfizer Benzimidazole derivatives
MX359989B (es) 2012-02-17 2018-10-18 Siga Tech Inc Fármacos antivirales para el tratamiento de la infección por arenavirus.
AU2018351059B2 (en) 2017-10-19 2022-05-12 Teijin Pharma Limited Benzimidazole derivatives and their uses
KR20210125471A (ko) 2018-10-05 2021-10-18 안나푸르나 바이오, 인코포레이티드 Apj 수용체 활성과 관련된 병태를 치료하기 위한 화합물 및 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997012613A1 (en) * 1995-10-05 1997-04-10 Warner-Lambert Company Method for treating and preventing inflammation and atherosclerosis
US6340681B1 (en) * 1999-07-16 2002-01-22 Pfizer Inc 2-benzimidazolylamine compounds as ORL-1-receptor agonists
WO2003104233A1 (en) * 2002-06-07 2003-12-18 Altana Pharma Ag 4,5-dihydro-imidazo (4,5,1-ij) quinolin-6-ones derivatives and their use as poly (adp-ribosyl) transferase (parp) inhibitors

Also Published As

Publication number Publication date
US20080090870A1 (en) 2008-04-17
WO2006099942A3 (de) 2007-06-21
JP2008533066A (ja) 2008-08-21
EP1863488A2 (de) 2007-12-12
DE102005012875B4 (de) 2006-11-16
BRPI0608451A2 (pt) 2009-12-29
IL185807A0 (en) 2008-01-06
DE102005012875A1 (de) 2006-09-21
US8003668B2 (en) 2011-08-23
EP1863488B1 (de) 2010-02-24
DE502006006241D1 (de) 2010-04-08
AU2006226639A1 (en) 2006-09-28
MX2007010836A (es) 2007-11-09
CA2602236A1 (en) 2006-09-28
WO2006099942A2 (de) 2006-09-28
WO2006099942A8 (de) 2006-11-09

Similar Documents

Publication Publication Date Title
IL185808A0 (en) Amide-substituted 8-n-benzimidazoles, metohd for the production thereof, and use of the same as medicaments
EA201170521A1 (ru) Новые соединения
EA200870019A1 (ru) Лактамовые соединения и способы их применения
EA201001358A1 (ru) Активаторы глюкокиназы
GT200600046A (es) Terapia de combinacion
NO20074943L (no) Roflumilast for behandlingen av diabetes mellitus
EA201100302A1 (ru) Лечение диабета у пациентов, для которых лечение метформином является неприемлемым
NO20082594L (no) Pyrimidinylbenzotiofenforbindelser
EA201200631A1 (ru) Ингибиторы репликации вируса иммунодефицита человека
EA200800201A1 (ru) Кристаллические формы 4-метил-n-[3-(4-метилимидазол-1-ил)-5-трифторметилфенил]-3-(4-пиридин-3-илпиримидин-2-иламино)бензамида
DK2026803T3 (da) Sammensætninger af R(+) og S(-) pramipexol og fremgangsmåder til anvendelse heraf
EA200870446A1 (ru) Пиридон сульфонамиды и пиридон сульфамиды в качестве ингибиторов мек
ATE476418T1 (de) Benzamidderivate und assoziierte verwendungen
NO20080626L (no) Inhibitorer av fibroblastaktiverende protein alfa
EA200700096A1 (ru) Производные 2-карбамид-4-фенилтиазола, способ их получения и их применение в терапии
EA200870515A1 (ru) Моноциклические гетероарильные соединения
CL2007000595A1 (es) Compuestos derivados de piperidina; composicion farmaceutica y uso para el tratamiento y/o profilaxis de enfermedades seleccionadas entre hipertension, insuficiencia cardiaca congestiva e insuficiencia renal entre otras.
EA200601777A1 (ru) Новое применение пептидных соединений для лечения боли при болезненной диабетической нейропатии
EA201000391A1 (ru) Соединение, представляющее собой ингибитор гликогенфосфорилазы, и его фармацевтическая композиция
NO20081292L (no) Pentasykliske kinaseinhibitorer
EA200702567A1 (ru) Ингибиторы дипептидил пептидазы iv, основанные на пирролопиридине
EA201001408A1 (ru) Производные пиразинона как стимуляторы секреции инсулина, способы их получения и их применение для лечения диабетов
EA200701995A1 (ru) Способы уменьшения кальцификации
IL185807A0 (en) Use of amino-substituted benzimidazoles
EA201000392A1 (ru) Соединение, представляющее собой ингибитор гликогенфосфорилазы, и его фармацевтическая композиция