ATE429T1 - 11-METHYLENE STEROIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM. - Google Patents

11-METHYLENE STEROIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM.

Info

Publication number
ATE429T1
ATE429T1 AT80101470T AT80101470T ATE429T1 AT E429 T1 ATE429 T1 AT E429T1 AT 80101470 T AT80101470 T AT 80101470T AT 80101470 T AT80101470 T AT 80101470T AT E429 T1 ATE429 T1 AT E429T1
Authority
AT
Austria
Prior art keywords
preparation
pharmaceutical preparations
preparations containing
methylene steroids
steroids
Prior art date
Application number
AT80101470T
Other languages
German (de)
Inventor
Helmut Dr. Hofmeister
Rudolf Prof. Dr. Wiechert
Klaus Dr. Annen
Henry Dr. Laurent
Hermann Dr. Steinbeck
Original Assignee
Schering Aktiengesellschaft Berlin Und Bergkamen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Aktiengesellschaft Berlin Und Bergkamen filed Critical Schering Aktiengesellschaft Berlin Und Bergkamen
Application granted granted Critical
Publication of ATE429T1 publication Critical patent/ATE429T1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/006—Ketals at position 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

11-Methylene steroids of Formula I <IMAGE> wherein R is hydrogen or acyl, and X is oxygen or two hydrogen atoms have valuable pharmacological properties.
AT80101470T 1979-03-30 1980-03-20 11-METHYLENE STEROIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM. ATE429T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19792913381 DE2913381A1 (en) 1979-03-30 1979-03-30 11-METHYLENESTEROIDS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM
EP80101470A EP0017094B1 (en) 1979-03-30 1980-03-20 11-methylene steroids, process for their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
ATE429T1 true ATE429T1 (en) 1981-12-15

Family

ID=6067313

Family Applications (1)

Application Number Title Priority Date Filing Date
AT80101470T ATE429T1 (en) 1979-03-30 1980-03-20 11-METHYLENE STEROIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM.

Country Status (10)

Country Link
US (1) US4277468A (en)
EP (1) EP0017094B1 (en)
JP (1) JPS55130999A (en)
AT (1) ATE429T1 (en)
AU (1) AU529541B2 (en)
CA (1) CA1146533A (en)
DE (2) DE2913381A1 (en)
DK (1) DK115780A (en)
ES (1) ES489682A1 (en)
IE (1) IE49572B1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3042529A1 (en) * 1980-11-07 1982-06-24 Schering Ag, 1000 Berlin Und 4619 Bergkamen 11-METHYLENE (DELTA) (UP ARROW) 1 (UP ARROW) (UP ARROW) 5 (UP ARROW) STEROIDS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM
US4557867A (en) * 1984-01-25 1985-12-10 The Upjohn Company 11β-Difluoromethyl and (E)- and (Z)-11-fluoromethylene steriods
US4567000A (en) * 1984-08-31 1986-01-28 The Upjohn Company 11-Difluoromethylene steroids

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE651797A (en) * 1962-10-17
DE1934272A1 (en) * 1969-07-02 1971-01-14 Schering Ag d-18-methyl-17 alpha-alkynyl-4-estren-17 beta-ols
FI54128C (en) * 1972-12-09 1978-10-10 Akzo Nv FREQUENCY REFRIGERATION FOR NY 11,11-ALKYLIDENSTEROIDER UR OESTRAN- OCH 19-NORPREGNANSERIEN MED FOERBAETTRAD HORMONELL VERKAN

Also Published As

Publication number Publication date
DE3060093D1 (en) 1982-01-28
DK115780A (en) 1980-10-01
CA1146533A (en) 1983-05-17
EP0017094B1 (en) 1981-11-25
DE2913381A1 (en) 1980-10-16
AU5698580A (en) 1980-10-02
US4277468A (en) 1981-07-07
JPS55130999A (en) 1980-10-11
JPS629600B2 (en) 1987-02-28
IE49572B1 (en) 1985-10-30
ES489682A1 (en) 1980-09-16
IE800640L (en) 1980-09-30
AU529541B2 (en) 1983-06-09
EP0017094A1 (en) 1980-10-15

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Legal Events

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