ATE424387T1 - Chinolinderivate als neurokininrezeptor- antagonisten - Google Patents
Chinolinderivate als neurokininrezeptor- antagonistenInfo
- Publication number
- ATE424387T1 ATE424387T1 AT05768021T AT05768021T ATE424387T1 AT E424387 T1 ATE424387 T1 AT E424387T1 AT 05768021 T AT05768021 T AT 05768021T AT 05768021 T AT05768021 T AT 05768021T AT E424387 T1 ATE424387 T1 AT E424387T1
- Authority
- AT
- Austria
- Prior art keywords
- neurokinine
- receptor antagonists
- quinoline derivatives
- neurokinin
- schizophrenia
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/50—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 4
- C07D215/52—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 4 with aryl radicals attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0417559.2A GB0417559D0 (en) | 2004-08-06 | 2004-08-06 | Therapeutic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE424387T1 true ATE424387T1 (de) | 2009-03-15 |
Family
ID=32982650
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT05768021T ATE424387T1 (de) | 2004-08-06 | 2005-07-28 | Chinolinderivate als neurokininrezeptor- antagonisten |
Country Status (10)
Country | Link |
---|---|
US (1) | US20080312274A1 (de) |
EP (1) | EP1776343B1 (de) |
JP (1) | JP2008509122A (de) |
CN (1) | CN1993330A (de) |
AT (1) | ATE424387T1 (de) |
AU (1) | AU2005268603A1 (de) |
CA (1) | CA2575697A1 (de) |
DE (1) | DE602005013094D1 (de) |
GB (1) | GB0417559D0 (de) |
WO (1) | WO2006013394A1 (de) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0509405D0 (en) * | 2005-05-10 | 2005-06-15 | Merck Sharp & Dohme | Therapeutic compounds |
JP6306708B2 (ja) * | 2014-07-22 | 2018-04-04 | 株式会社日立ハイテクノロジーズ | 細胞分散装置およびそれを用いた自動継代培養システム |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0940391B1 (de) * | 1994-05-27 | 2004-08-18 | GlaxoSmithKline S.p.A. | Chinolinderivate als Tachykinin NK3 Rezeptor Antagonisten |
GB0228288D0 (en) * | 2002-12-04 | 2003-01-08 | Smithkline Beecham Corp | Chemical compounds |
GB0303086D0 (en) * | 2003-02-11 | 2003-03-19 | Merck Sharp & Dohme | New compounds |
-
2004
- 2004-08-06 GB GBGB0417559.2A patent/GB0417559D0/en not_active Ceased
-
2005
- 2005-07-28 AU AU2005268603A patent/AU2005268603A1/en not_active Abandoned
- 2005-07-28 CN CNA2005800264225A patent/CN1993330A/zh active Pending
- 2005-07-28 AT AT05768021T patent/ATE424387T1/de not_active IP Right Cessation
- 2005-07-28 US US11/659,401 patent/US20080312274A1/en not_active Abandoned
- 2005-07-28 DE DE602005013094T patent/DE602005013094D1/de not_active Expired - Fee Related
- 2005-07-28 WO PCT/GB2005/050121 patent/WO2006013394A1/en active Application Filing
- 2005-07-28 EP EP05768021A patent/EP1776343B1/de not_active Not-in-force
- 2005-07-28 CA CA002575697A patent/CA2575697A1/en not_active Abandoned
- 2005-07-28 JP JP2007524404A patent/JP2008509122A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP1776343B1 (de) | 2009-03-04 |
EP1776343A1 (de) | 2007-04-25 |
US20080312274A1 (en) | 2008-12-18 |
GB0417559D0 (en) | 2004-09-08 |
DE602005013094D1 (de) | 2009-04-16 |
CA2575697A1 (en) | 2006-02-09 |
WO2006013394A1 (en) | 2006-02-09 |
JP2008509122A (ja) | 2008-03-27 |
CN1993330A (zh) | 2007-07-04 |
AU2005268603A1 (en) | 2006-02-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |