ATE421523T1 - Verfahren zur herstellung von 4-azasteroiden - Google Patents

Verfahren zur herstellung von 4-azasteroiden

Info

Publication number
ATE421523T1
ATE421523T1 AT05759142T AT05759142T ATE421523T1 AT E421523 T1 ATE421523 T1 AT E421523T1 AT 05759142 T AT05759142 T AT 05759142T AT 05759142 T AT05759142 T AT 05759142T AT E421523 T1 ATE421523 T1 AT E421523T1
Authority
AT
Austria
Prior art keywords
hydrogen
group
alkyl
cyano
coo
Prior art date
Application number
AT05759142T
Other languages
English (en)
Inventor
Yves Bessard
David Kuo
Original Assignee
Lonza Group Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Group Ag filed Critical Lonza Group Ag
Application granted granted Critical
Publication of ATE421523T1 publication Critical patent/ATE421523T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT05759142T 2004-07-05 2005-07-04 Verfahren zur herstellung von 4-azasteroiden ATE421523T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04015746A EP1619200A1 (de) 2004-07-05 2004-07-05 Verfahren zur Herstellung von 4-Azasteroiden

Publications (1)

Publication Number Publication Date
ATE421523T1 true ATE421523T1 (de) 2009-02-15

Family

ID=34925615

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05759142T ATE421523T1 (de) 2004-07-05 2005-07-04 Verfahren zur herstellung von 4-azasteroiden

Country Status (14)

Country Link
US (1) US20120226044A1 (de)
EP (2) EP1619200A1 (de)
JP (1) JP4981668B2 (de)
KR (1) KR20070028527A (de)
CN (1) CN1980950B (de)
AT (1) ATE421523T1 (de)
BR (1) BRPI0513039A (de)
CA (1) CA2570468C (de)
DE (1) DE602005012508D1 (de)
EA (1) EA014871B1 (de)
ES (1) ES2321423T3 (de)
HK (1) HK1106535A1 (de)
IL (1) IL180085A (de)
WO (1) WO2006002966A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20071905A1 (it) * 2007-10-04 2009-04-05 Tender Aps Derivati dell'idrocortisone e loro uso per indicazioni terapeutiche o cosmetiche
ITPI20090151A1 (it) 2009-11-27 2011-05-28 Giovanni Barco Estensione degli usi specifici della deina, di cui al brevetto d'invenzione pct/ib 2008 002562 "derivati dell'idrocortisone e loro usi per indicazioni terapeutiche o cosmetiche"
CN106632559B (zh) * 2016-12-11 2018-10-30 湖北竹溪人福药业有限责任公司 一种利用黄体酮母液物制备雄甾-3-酮-4-烯-17β羧酸的方法
EP3875464A1 (de) 2020-03-06 2021-09-08 F.I.S.- Fabbrica Italiana Sintetici S.p.A. Verfahren zur reinigung von etiocholensäure
CN113624898B (zh) * 2021-08-23 2023-08-25 成都诺和晟泰生物科技有限公司 一种手性镇痛类多肽药物的纯化方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE178795T1 (de) * 1993-11-04 1999-04-15 Merck & Co Inc 7-substituierte-4-aza-steroid-derivate als 5- alpha-reductase-hemmer
CN1121409C (zh) * 2001-01-18 2003-09-17 湖南正清制药集团股份有限公司 一种药物的生产方法

Also Published As

Publication number Publication date
JP2008505147A (ja) 2008-02-21
EP1619200A1 (de) 2006-01-25
CA2570468C (en) 2012-06-19
DE602005012508D1 (de) 2009-03-12
EA200700068A1 (ru) 2007-08-31
US20120226044A1 (en) 2012-09-06
KR20070028527A (ko) 2007-03-12
CA2570468A1 (en) 2006-01-12
CN1980950A (zh) 2007-06-13
EA014871B1 (ru) 2011-02-28
ES2321423T3 (es) 2009-06-05
IL180085A0 (en) 2007-05-15
EP1765848B1 (de) 2009-01-21
HK1106535A1 (en) 2008-03-14
BRPI0513039A (pt) 2008-04-22
CN1980950B (zh) 2011-07-20
EP1765848B8 (de) 2009-04-15
JP4981668B2 (ja) 2012-07-25
EP1765848A1 (de) 2007-03-28
WO2006002966A1 (en) 2006-01-12
IL180085A (en) 2012-01-31

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Legal Events

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