ATE417052T1 - Oxazaborolidine als bakterielle effektoren - Google Patents

Oxazaborolidine als bakterielle effektoren

Info

Publication number
ATE417052T1
ATE417052T1 AT04770462T AT04770462T ATE417052T1 AT E417052 T1 ATE417052 T1 AT E417052T1 AT 04770462 T AT04770462 T AT 04770462T AT 04770462 T AT04770462 T AT 04770462T AT E417052 T1 ATE417052 T1 AT E417052T1
Authority
AT
Austria
Prior art keywords
bacteria
composition
oxazaborolidines
decreasing
relates
Prior art date
Application number
AT04770462T
Other languages
English (en)
Inventor
Morris Srebnik
Adel Jabbour
Arik Moussaieff
Valery Dembitsky
Moshe Bronshteyn
Doron Steinberg
Original Assignee
Yissum Res Dev Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yissum Res Dev Co filed Critical Yissum Res Dev Co
Application granted granted Critical
Publication of ATE417052T1 publication Critical patent/ATE417052T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT04770462T 2003-09-02 2004-09-02 Oxazaborolidine als bakterielle effektoren ATE417052T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49900503P 2003-09-02 2003-09-02

Publications (1)

Publication Number Publication Date
ATE417052T1 true ATE417052T1 (de) 2008-12-15

Family

ID=34272757

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04770462T ATE417052T1 (de) 2003-09-02 2004-09-02 Oxazaborolidine als bakterielle effektoren

Country Status (7)

Country Link
US (1) US20070155698A1 (de)
EP (1) EP1664064B1 (de)
JP (1) JP5030590B2 (de)
AT (1) ATE417052T1 (de)
DE (1) DE602004018339D1 (de)
ES (1) ES2319197T3 (de)
WO (1) WO2005021559A2 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2654449A1 (en) * 2006-06-12 2007-12-21 Anacor Pharmaceuticals, Inc. Compounds for the treatment of periodontal disease
EP2136800A4 (de) * 2007-03-19 2011-10-05 Wisconsin Alumni Res Found Modulation der bakteriellen quorum-messung mit synthetischen liganden
EP2529793B1 (de) * 2007-06-08 2016-08-10 Georgia State University Research Foundation, Inc. Zusammensetzungen zur Regulierung oder Modulierung von Quorum-Sensing in Bakterien, Verfahren zur Verwendung der Verbindungen sowie Verfahren zur Regulierung oder Modulierung von Quorum-Sensing in Bakterien
US8624063B2 (en) 2009-06-30 2014-01-07 Wisconsin Alumni Research Foundation Non-lactone carbocyclic and heterocyclic antagonists and agonists of bacterial quorum sensing
EP2459149A2 (de) * 2009-07-28 2012-06-06 QSlant Limited Antibakterielle kombinationen mit einem knoblauchextrakt oder einem s-allyl-zystein
WO2012137166A1 (en) 2011-04-07 2012-10-11 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. An oxoborolidine compound and uses thereof
WO2012137164A1 (en) 2011-04-07 2012-10-11 Biolinerx Ltd. Antimicrobial compositions, antibiofilm compositions and uses thereof
FR3029936B1 (fr) 2014-12-15 2020-01-24 Biomerieux Procede et dispositif de caracterisation du pouvoir inhibiteur d'une molecule sur un microorganisme
US10526278B2 (en) 2017-10-19 2020-01-07 Wisconsin Alumni Research Foundation Inhibitors of quorum sensing receptor LasR
GB202111203D0 (en) 2021-08-03 2021-09-15 Pathway Intermediates Ltd Novel applications for oxazaborolidines and new methods of manufacture thereof.
GB202111761D0 (en) 2021-08-17 2021-09-29 Collins Mike Methods for preparing oxazoborolidines

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3137723A (en) * 1961-09-25 1964-06-16 Olin Mathieson Boron containing heterocyclic compounds and process for producing them
JP3498332B2 (ja) * 1993-10-07 2004-02-16 住友化学工業株式会社 不斉還元剤、および該不斉還元剤を用いる光学活性体の製造方法
US6458764B1 (en) * 1995-05-26 2002-10-01 Theratechnologies Inc. GRF analogs with increased biological potency
US5538829A (en) * 1995-09-05 1996-07-23 Xerox Corporation Toner compositions with zinc and boron charge enhancing additives
JP2003532698A (ja) * 2000-05-10 2003-11-05 プリンストン ユニバーシティ 細菌の増殖および病理発生を調節するための化合物ならびに方法
US6737415B2 (en) * 2001-08-24 2004-05-18 Quorex Pharmaceuticals, Inc. Anti-bacterial agents based upon oxoanion binding
JP2003192596A (ja) * 2001-12-27 2003-07-09 Shionogi & Co Ltd 有機ホウ素化合物を含有する新規な抗コクシジウム剤

Also Published As

Publication number Publication date
JP2007504214A (ja) 2007-03-01
DE602004018339D1 (de) 2009-01-22
JP5030590B2 (ja) 2012-09-19
WO2005021559A3 (en) 2005-04-07
ES2319197T3 (es) 2009-05-05
EP1664064B1 (de) 2008-12-10
WO2005021559A2 (en) 2005-03-10
EP1664064A2 (de) 2006-06-07
US20070155698A1 (en) 2007-07-05

Similar Documents

Publication Publication Date Title
IL189017A0 (en) 8-methoxy-9h-isothiazolo[5,4-b]quinoline-3,4-diones and related compounds as anti-effective agents
MXPA06000675A (es) Derivado de quinolona o sal del mismo.
MY150630A (en) Amide derivative and insecticide containing the same
EA200200072A1 (ru) Пресервированные фармацевтические составы
EA200801083A1 (ru) Новые производные дигидропсевдоэритромицина
BRPI0510262A (pt) composição herbicida, e, método de combater ervas danihas e gramìneas daninhas em colheitas de plantas úteis
MX2007000392A (es) Derivados de 2-pirrolidona sustituida como fungicidas e insecticidas.
WO2007067559A3 (en) Antibacterial agents
ATE417052T1 (de) Oxazaborolidine als bakterielle effektoren
TW200734344A (en) Antibacterial agents
ATE420639T1 (de) Antimykotische mittel
BG108498A (en) New derivatives of oxazolidinones as antibacterial agents
UA84879C2 (ru) Изотиазолохинолоны и родственные соединения с противомикробным действием
BRPI0411534A (pt) derivados de lincomicina com atividade antimicrobiana
WO2005054234A3 (en) Substituted piperidino phenyloxazolidinones having antimicriobial activity with improved in vivo efficacy
TW200602295A (en) Organic compounds
SE0300105D0 (sv) Diarylmethylidene piperdine derivatives, preparations thereof and uses thereof
EA200900640A1 (ru) Пиримидилметилсульфонамидные соединения
TW200613251A (en) Organic compounds
UA101954C2 (ru) Замещенные ароматические гетероциклические соединения как фунгициды
CY1110156T1 (el) Υποκατεστημενες ενωσεις 4,5,6,7-τετραϋδρο-βενζοθειαζολ-2-υλαμινης
IL183153A0 (en) 8a, 9-DIHYDRO-4a-H-ISOTHIAZOLO[5,4-b]QUINOLINE-3,4-DIONES AND RELATED COMPOUNDS AS ANTI-INFECTIVE AGENTS
DK1439840T3 (da) Antibakterielle monobactam-forbindelser og fremgangsmåder til anvendelse heraf
WO2007027878A3 (en) 4-substituted 2-aryloxyphenol derivatives as antibacterial agents
UA91549C2 (ru) Производные хинолина как антибактериальные агенты

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties