ATE417052T1 - Oxazaborolidine als bakterielle effektoren - Google Patents

Oxazaborolidine als bakterielle effektoren

Info

Publication number
ATE417052T1
ATE417052T1 AT04770462T AT04770462T ATE417052T1 AT E417052 T1 ATE417052 T1 AT E417052T1 AT 04770462 T AT04770462 T AT 04770462T AT 04770462 T AT04770462 T AT 04770462T AT E417052 T1 ATE417052 T1 AT E417052T1
Authority
AT
Austria
Prior art keywords
bacteria
composition
oxazaborolidines
decreasing
relates
Prior art date
Application number
AT04770462T
Other languages
English (en)
Inventor
Morris Srebnik
Adel Jabbour
Arik Moussaieff
Valery Dembitsky
Moshe Bronshteyn
Doron Steinberg
Original Assignee
Yissum Res Dev Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yissum Res Dev Co filed Critical Yissum Res Dev Co
Application granted granted Critical
Publication of ATE417052T1 publication Critical patent/ATE417052T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
AT04770462T 2003-09-02 2004-09-02 Oxazaborolidine als bakterielle effektoren ATE417052T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49900503P 2003-09-02 2003-09-02

Publications (1)

Publication Number Publication Date
ATE417052T1 true ATE417052T1 (de) 2008-12-15

Family

ID=34272757

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04770462T ATE417052T1 (de) 2003-09-02 2004-09-02 Oxazaborolidine als bakterielle effektoren

Country Status (7)

Country Link
US (1) US20070155698A1 (de)
EP (1) EP1664064B1 (de)
JP (1) JP5030590B2 (de)
AT (1) ATE417052T1 (de)
DE (1) DE602004018339D1 (de)
ES (1) ES2319197T3 (de)
WO (1) WO2005021559A2 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2654449A1 (en) * 2006-06-12 2007-12-21 Anacor Pharmaceuticals, Inc. Compounds for the treatment of periodontal disease
EP2136800A4 (de) * 2007-03-19 2011-10-05 Wisconsin Alumni Res Found Modulation der bakteriellen quorum-messung mit synthetischen liganden
EP2155705A4 (de) * 2007-06-08 2012-02-15 Univ Georgia State Res Found Zusammensetzungen zur regulierung oder modulierung eines quorum-sensings in bakterien, verfahren zur verwendung der verbindungen und verfahren zur regulierung oder modulierung eines quorum-sensings in bakterien
US8624063B2 (en) 2009-06-30 2014-01-07 Wisconsin Alumni Research Foundation Non-lactone carbocyclic and heterocyclic antagonists and agonists of bacterial quorum sensing
GB2472315B (en) * 2009-07-28 2012-01-18 Raymond Stanley Steggles Antibacterial compositions
WO2012137166A1 (en) 2011-04-07 2012-10-11 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. An oxoborolidine compound and uses thereof
WO2012137164A1 (en) 2011-04-07 2012-10-11 Biolinerx Ltd. Antimicrobial compositions, antibiofilm compositions and uses thereof
FR3029936B1 (fr) * 2014-12-15 2020-01-24 Biomerieux Procede et dispositif de caracterisation du pouvoir inhibiteur d'une molecule sur un microorganisme
US10526278B2 (en) 2017-10-19 2020-01-07 Wisconsin Alumni Research Foundation Inhibitors of quorum sensing receptor LasR
GB202111203D0 (en) 2021-08-03 2021-09-15 Pathway Intermediates Ltd Novel applications for oxazaborolidines and new methods of manufacture thereof.
GB202111761D0 (en) 2021-08-17 2021-09-29 Collins Mike Methods for preparing oxazoborolidines

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3137723A (en) * 1961-09-25 1964-06-16 Olin Mathieson Boron containing heterocyclic compounds and process for producing them
JP3498332B2 (ja) * 1993-10-07 2004-02-16 住友化学工業株式会社 不斉還元剤、および該不斉還元剤を用いる光学活性体の製造方法
US6458764B1 (en) * 1995-05-26 2002-10-01 Theratechnologies Inc. GRF analogs with increased biological potency
US5538829A (en) * 1995-09-05 1996-07-23 Xerox Corporation Toner compositions with zinc and boron charge enhancing additives
EP1282415A2 (de) * 2000-05-10 2003-02-12 Princeton University Office of Techology Licensing & I.P. Verbindungen und verfahren zur regulierung von bakteriellen wachstum und pathogenese
CA2455504A1 (en) * 2001-08-24 2003-03-06 Quorex Pharmaceuticals, Inc. Anti-bacterial agents based upon oxoanion binding
JP2003192596A (ja) * 2001-12-27 2003-07-09 Shionogi & Co Ltd 有機ホウ素化合物を含有する新規な抗コクシジウム剤

Also Published As

Publication number Publication date
JP5030590B2 (ja) 2012-09-19
JP2007504214A (ja) 2007-03-01
EP1664064A2 (de) 2006-06-07
ES2319197T3 (es) 2009-05-05
DE602004018339D1 (de) 2009-01-22
EP1664064B1 (de) 2008-12-10
WO2005021559A2 (en) 2005-03-10
US20070155698A1 (en) 2007-07-05
WO2005021559A3 (en) 2005-04-07

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties