ATE396177T1 - Neue kristalline formen eines faktor xa inhibitors - Google Patents
Neue kristalline formen eines faktor xa inhibitorsInfo
- Publication number
- ATE396177T1 ATE396177T1 AT01979459T AT01979459T ATE396177T1 AT E396177 T1 ATE396177 T1 AT E396177T1 AT 01979459 T AT01979459 T AT 01979459T AT 01979459 T AT01979459 T AT 01979459T AT E396177 T1 ATE396177 T1 AT E396177T1
- Authority
- AT
- Austria
- Prior art keywords
- inhibitor
- factor
- crystalline forms
- new crystalline
- new
- Prior art date
Links
- 229940123583 Factor Xa inhibitor Drugs 0.000 title 1
- 108010074860 Factor Xa Proteins 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Liquid Crystal Substances (AREA)
- Compounds Of Unknown Constitution (AREA)
- Medicinal Preparation (AREA)
- Pyridine Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23831600P | 2000-10-05 | 2000-10-05 | |
| GBGB0108903.6A GB0108903D0 (en) | 2000-10-05 | 2001-04-10 | Novel crystalline forms of a factor Xa inhibitor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE396177T1 true ATE396177T1 (de) | 2008-06-15 |
Family
ID=22897372
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01979459T ATE396177T1 (de) | 2000-10-05 | 2001-10-04 | Neue kristalline formen eines faktor xa inhibitors |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7034160B2 (de) |
| EP (1) | EP1326838B1 (de) |
| JP (1) | JP4177663B2 (de) |
| AT (1) | ATE396177T1 (de) |
| AU (2) | AU1142502A (de) |
| CA (1) | CA2424565C (de) |
| CY (1) | CY1108224T1 (de) |
| DK (1) | DK1326838T3 (de) |
| ES (1) | ES2304396T3 (de) |
| GB (1) | GB0108903D0 (de) |
| IL (1) | IL155189A (de) |
| MX (1) | MXPA03002067A (de) |
| PT (1) | PT1326838E (de) |
| WO (1) | WO2002028836A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6964784B2 (en) * | 2002-03-07 | 2005-11-15 | Optigenex, Inc. | Method of preparation and composition of a water soluble extract of the bioactive component of the plant species uncaria for enhancing immune, anti-inflammatory, anti-tumor and dna repair processes of warm blooded animals |
| SG193612A1 (en) * | 2011-03-29 | 2013-11-29 | Sanofi Sa | Benzoic acid salt of otamixaban |
| TWI551289B (zh) * | 2011-03-29 | 2016-10-01 | 賽諾菲公司 | 具有改良之安定性之奧米沙班調配物 |
| EA025572B1 (ru) * | 2011-03-29 | 2017-01-30 | Санофи | Лекарственные формы отамиксабана с улучшенной стабильностью |
| CA3218491A1 (en) | 2012-06-04 | 2013-12-12 | Pharmacyclics Llc | Crystalline forms of a bruton's tyrosine kinase inhibitor |
| MX2017001671A (es) | 2014-08-07 | 2017-07-04 | Pharmacyclics Llc | Formulaciones novedosas de un inhibidor de la tirosina cinasa de bruton. |
| IL315294A (en) | 2015-03-03 | 2024-10-01 | Pharmacyclics Llc | Pharmaceutical formulations of bruton's tyrosine kinase inhibitor |
| MA41827A (fr) * | 2015-03-27 | 2018-01-30 | Pharmacyclics Llc | Formes solvatées d'un inhibiteur de la tyrosine kinase de bruton |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CZ297544B6 (cs) * | 1996-01-02 | 2007-02-07 | Aventis Pharmaceuticals Inc. | Substituované N-[(aminoiminomethyl)-fenyl]propylamidy nebo N-[(aminomethyl)fenyl]propylamidy |
| US6080767A (en) * | 1996-01-02 | 2000-06-27 | Aventis Pharmaceuticals Products Inc. | Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides |
-
2001
- 2001-04-10 GB GBGB0108903.6A patent/GB0108903D0/en not_active Ceased
- 2001-10-04 AU AU1142502A patent/AU1142502A/xx active Pending
- 2001-10-04 CA CA2424565A patent/CA2424565C/en not_active Expired - Fee Related
- 2001-10-04 MX MXPA03002067A patent/MXPA03002067A/es active IP Right Grant
- 2001-10-04 ES ES01979459T patent/ES2304396T3/es not_active Expired - Lifetime
- 2001-10-04 AU AU2002211425A patent/AU2002211425B2/en not_active Ceased
- 2001-10-04 DK DK01979459T patent/DK1326838T3/da active
- 2001-10-04 PT PT01979459T patent/PT1326838E/pt unknown
- 2001-10-04 JP JP2002532422A patent/JP4177663B2/ja not_active Expired - Fee Related
- 2001-10-04 AT AT01979459T patent/ATE396177T1/de active
- 2001-10-04 EP EP01979459A patent/EP1326838B1/de not_active Expired - Lifetime
- 2001-10-04 WO PCT/US2001/031087 patent/WO2002028836A1/en not_active Ceased
-
2003
- 2003-04-01 IL IL155189A patent/IL155189A/en not_active IP Right Cessation
- 2003-04-01 US US10/404,678 patent/US7034160B2/en not_active Expired - Lifetime
-
2008
- 2008-07-29 CY CY20081100790T patent/CY1108224T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PT1326838E (pt) | 2008-07-08 |
| US20030225144A1 (en) | 2003-12-04 |
| US7034160B2 (en) | 2006-04-25 |
| JP2004521082A (ja) | 2004-07-15 |
| ES2304396T3 (es) | 2008-10-16 |
| AU2002211425B2 (en) | 2006-03-02 |
| JP4177663B2 (ja) | 2008-11-05 |
| IL155189A (en) | 2011-11-30 |
| CA2424565C (en) | 2011-04-26 |
| EP1326838B1 (de) | 2008-05-21 |
| AU1142502A (en) | 2002-04-15 |
| WO2002028836A1 (en) | 2002-04-11 |
| MXPA03002067A (es) | 2003-06-24 |
| WO2002028836A9 (en) | 2003-11-20 |
| GB0108903D0 (en) | 2001-05-30 |
| DK1326838T3 (da) | 2008-09-22 |
| CY1108224T1 (el) | 2014-02-12 |
| EP1326838A1 (de) | 2003-07-16 |
| CA2424565A1 (en) | 2002-04-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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