ATE349457T1 - Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen - Google Patents

Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen

Info

Publication number
ATE349457T1
ATE349457T1 AT04706638T AT04706638T ATE349457T1 AT E349457 T1 ATE349457 T1 AT E349457T1 AT 04706638 T AT04706638 T AT 04706638T AT 04706638 T AT04706638 T AT 04706638T AT E349457 T1 ATE349457 T1 AT E349457T1
Authority
AT
Austria
Prior art keywords
avermectin
derivatives substituted
pesticidal properties
monosaccharide derivatives
exhibit pesticidal
Prior art date
Application number
AT04706638T
Other languages
English (en)
Inventor
Thomas Pitterna
Kessabi Fiona Murphy
Peter Maienfisch
Jerome Cassayre
Laura Quaranta
Pierre Jung
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Application granted granted Critical
Publication of ATE349457T1 publication Critical patent/ATE349457T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Environmental Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AT04706638T 2003-01-31 2004-01-30 Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen ATE349457T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0302308.2A GB0302308D0 (en) 2003-01-31 2003-01-31 Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties

Publications (1)

Publication Number Publication Date
ATE349457T1 true ATE349457T1 (de) 2007-01-15

Family

ID=9952239

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04706638T ATE349457T1 (de) 2003-01-31 2004-01-30 Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen

Country Status (15)

Country Link
US (1) US7678740B2 (de)
EP (1) EP1592699B1 (de)
JP (1) JP2006516584A (de)
AR (1) AR042966A1 (de)
AT (1) ATE349457T1 (de)
CL (1) CL2004000148A1 (de)
CY (1) CY1108005T1 (de)
DE (1) DE602004003907T2 (de)
DK (1) DK1592699T3 (de)
ES (1) ES2280022T3 (de)
GB (1) GB0302308D0 (de)
PT (1) PT1592699E (de)
SI (1) SI1592699T1 (de)
TW (1) TW200510443A (de)
WO (1) WO2004067543A1 (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) * 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
GB0129267D0 (en) * 2001-12-06 2002-01-23 Syngenta Ltd Fungicides
TW200407330A (en) * 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0227556D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227558D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227555D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227554D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0312864D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0312863D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
HUE028600T2 (en) 2010-05-12 2016-12-28 Merial Inc Injectable parasiticidal formulations of levamisole and macrocyclic lactones
NZ612185A (en) 2010-12-07 2015-10-30 Merial Inc Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN109485683A (zh) * 2018-11-27 2019-03-19 齐鲁晟华制药有限公司 一种含氟系列阿维菌素衍生物及其制备方法
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN115403644B (zh) * 2022-09-01 2024-04-05 石家庄学院 一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

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NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
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US4662313A (en) * 1985-10-23 1987-05-05 Xerox Corporation Image density controller
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US5169839A (en) 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
IL98599A (en) 1990-06-28 1995-06-29 Merck & Co Inc Stable salts of 4"-deoxy-4"-epi-methylamino avermectin b1a/b1b and insecticidal compositions containing them
US5346698A (en) 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
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CA2418975C (en) 2000-08-09 2012-01-17 Satoshi Omura Avermectin derivatives
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
TW200301079A (en) 2001-12-21 2003-07-01 Syngenta Participations Ag Avermectin B1 derivatives having an aminosulfonyloxy substituent in the 4"-position
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302548D0 (en) 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
AR042966A1 (es) 2005-07-13
PT1592699E (pt) 2007-04-30
SI1592699T1 (sl) 2007-08-31
CL2004000148A1 (es) 2005-01-14
EP1592699B1 (de) 2006-12-27
GB0302308D0 (en) 2003-03-05
CY1108005T1 (el) 2013-09-04
US7678740B2 (en) 2010-03-16
ES2280022T3 (es) 2007-09-01
DE602004003907D1 (de) 2007-02-08
US20060140997A1 (en) 2006-06-29
TW200510443A (en) 2005-03-16
WO2004067543A1 (en) 2004-08-12
DE602004003907T2 (de) 2007-10-25
JP2006516584A (ja) 2006-07-06
EP1592699A1 (de) 2005-11-09
DK1592699T3 (da) 2007-05-07

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