ATE338046T1 - 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza- cyclopenta(a)naphthalenyl derivate mit antipsychotischer aktivität - Google Patents
2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza- cyclopenta(a)naphthalenyl derivate mit antipsychotischer aktivitätInfo
- Publication number
- ATE338046T1 ATE338046T1 AT02756528T AT02756528T ATE338046T1 AT E338046 T1 ATE338046 T1 AT E338046T1 AT 02756528 T AT02756528 T AT 02756528T AT 02756528 T AT02756528 T AT 02756528T AT E338046 T1 ATE338046 T1 AT E338046T1
- Authority
- AT
- Austria
- Prior art keywords
- diaza
- cyclopenta
- oxa
- aminomethyl
- tetrahydro
- Prior art date
Links
- -1 2-(AMINOMETHYL)-TETRAHYDRO-9-OXA-1,3-DIAZA-CYCLOPENTA(A)NAPHTHALENYL Chemical class 0.000 title 1
- 230000000561 anti-psychotic effect Effects 0.000 title 1
- VYFYYTLLBUKUHU-UHFFFAOYSA-N dopamine Chemical compound NCCC1=CC=C(O)C(O)=C1 VYFYYTLLBUKUHU-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 229960003638 dopamine Drugs 0.000 abstract 1
- 230000008482 dysregulation Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30693101P | 2001-07-20 | 2001-07-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE338046T1 true ATE338046T1 (de) | 2006-09-15 |
Family
ID=23187510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02756528T ATE338046T1 (de) | 2001-07-20 | 2002-07-19 | 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza- cyclopenta(a)naphthalenyl derivate mit antipsychotischer aktivität |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US6541502B1 (de) |
| EP (1) | EP1421086B1 (de) |
| JP (1) | JP2004537556A (de) |
| CN (1) | CN100369916C (de) |
| AT (1) | ATE338046T1 (de) |
| BR (1) | BR0211207A (de) |
| CA (1) | CA2454543A1 (de) |
| DE (1) | DE60214397T2 (de) |
| DK (1) | DK1421086T3 (de) |
| ES (1) | ES2271314T3 (de) |
| MX (1) | MXPA04000581A (de) |
| WO (1) | WO2003008419A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200640931A (en) | 2005-02-17 | 2006-12-01 | Wyeth Corp | Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives |
| TW201412727A (zh) * | 2012-08-24 | 2014-04-01 | Daiichi Sankyo Co Ltd | 具有鏈狀側鏈之色酮衍生物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4135474A1 (de) | 1991-10-28 | 1993-04-29 | Bayer Ag | 2-aminomethyl-chromane |
| DE4140540A1 (de) | 1991-12-09 | 1993-06-17 | Bayer Ag | Neue azaheterocyclylmethyl-chromane |
| US5756532A (en) | 1995-11-06 | 1998-05-26 | American Home Products Corporation | Aminomethyl-2 3 8 9-tetrahydro-7H-1 4-dioxino 2 3-E!-indol-8-ones and derivatives |
| AR004523A1 (es) * | 1995-11-06 | 1998-12-16 | American Home Prod | 2-(AMINOMETIL)-3,4,7,9-TETRAHIDRO-2H-PIRANO-[2,3e] INDOL-8-ONAS Y COMPOSICIONES FARMACEUTICAS QUE LAS COMPRENDEN |
| US5750556A (en) | 1996-10-30 | 1998-05-12 | American Home Products Corporation | 2-(aminomethyl)-3,4,7,9-tetrahydro-2H-pyrano- 2,3-E!indol-8-ones and derivatives |
| AU746717B2 (en) | 1997-02-18 | 2002-05-02 | Wyeth | 4-aminoalkoxy-1H-benzimidazole derivatives, their preparation and their use as dopamine autoreceptor (D2) agonists |
-
2002
- 2002-07-18 US US10/197,797 patent/US6541502B1/en not_active Expired - Fee Related
- 2002-07-19 CA CA002454543A patent/CA2454543A1/en not_active Abandoned
- 2002-07-19 BR BR0211207-8A patent/BR0211207A/pt not_active IP Right Cessation
- 2002-07-19 CN CNB028180232A patent/CN100369916C/zh not_active Expired - Fee Related
- 2002-07-19 AT AT02756528T patent/ATE338046T1/de not_active IP Right Cessation
- 2002-07-19 DK DK02756528T patent/DK1421086T3/da active
- 2002-07-19 EP EP02756528A patent/EP1421086B1/de not_active Expired - Lifetime
- 2002-07-19 JP JP2003513978A patent/JP2004537556A/ja active Pending
- 2002-07-19 DE DE60214397T patent/DE60214397T2/de not_active Expired - Fee Related
- 2002-07-19 WO PCT/US2002/022981 patent/WO2003008419A1/en not_active Ceased
- 2002-07-19 ES ES02756528T patent/ES2271314T3/es not_active Expired - Lifetime
- 2002-07-19 MX MXPA04000581A patent/MXPA04000581A/es active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EP1421086A1 (de) | 2004-05-26 |
| EP1421086B1 (de) | 2006-08-30 |
| MXPA04000581A (es) | 2004-04-20 |
| CA2454543A1 (en) | 2003-01-30 |
| ES2271314T3 (es) | 2007-04-16 |
| DK1421086T3 (da) | 2006-12-11 |
| JP2004537556A (ja) | 2004-12-16 |
| CN1555377A (zh) | 2004-12-15 |
| BR0211207A (pt) | 2004-07-13 |
| DE60214397T2 (de) | 2007-10-11 |
| US6541502B1 (en) | 2003-04-01 |
| DE60214397D1 (en) | 2006-10-12 |
| CN100369916C (zh) | 2008-02-20 |
| WO2003008419A1 (en) | 2003-01-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |