ATE213233T1 - Substituierte caprolactame und deren derivate verwendbar zur behandlung der hiv-krankheit - Google Patents
Substituierte caprolactame und deren derivate verwendbar zur behandlung der hiv-krankheitInfo
- Publication number
- ATE213233T1 ATE213233T1 AT94911704T AT94911704T ATE213233T1 AT E213233 T1 ATE213233 T1 AT E213233T1 AT 94911704 T AT94911704 T AT 94911704T AT 94911704 T AT94911704 T AT 94911704T AT E213233 T1 ATE213233 T1 AT E213233T1
- Authority
- AT
- Austria
- Prior art keywords
- treatment
- hiv disease
- substituted
- caprolactames
- derivatives usable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
- C07D245/02—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D255/00—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00
- C07D255/02—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00 not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D267/02—Seven-membered rings
- C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D267/10—Seven-membered rings having the hetero atoms in positions 1 and 4 not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/06—Seven-membered rings having the hetero atoms in positions 1 and 4 not condensed with other rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/040,324 US5663333A (en) | 1992-10-22 | 1993-03-30 | Substituted 1,4-diazapine caprolactams useful for treatment of HIV disease |
PCT/US1994/003224 WO1994022840A1 (en) | 1993-03-30 | 1994-03-28 | Substituted caprolactams and derivatives thereof useful for treatment of hiv disease |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE213233T1 true ATE213233T1 (de) | 2002-02-15 |
Family
ID=21910379
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT94911704T ATE213233T1 (de) | 1993-03-30 | 1994-03-28 | Substituierte caprolactame und deren derivate verwendbar zur behandlung der hiv-krankheit |
Country Status (7)
Country | Link |
---|---|
US (2) | US5663333A (de) |
EP (1) | EP0691961B1 (de) |
AT (1) | ATE213233T1 (de) |
AU (1) | AU6415994A (de) |
CA (1) | CA2159442A1 (de) |
DE (1) | DE69429856D1 (de) |
WO (1) | WO1994022840A1 (de) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5753652A (en) * | 1991-07-03 | 1998-05-19 | Novartis Corporation | Antiretroviral hydrazine derivatives |
US5663333A (en) * | 1992-10-22 | 1997-09-02 | The Dupont Merck Pharmaceutical Company | Substituted 1,4-diazapine caprolactams useful for treatment of HIV disease |
US5683999A (en) * | 1995-03-17 | 1997-11-04 | The Dupont Merck Pharmaceutical Company | Cyclic urea HIV protease inhibitors |
ZA966885B (en) * | 1995-08-22 | 1998-02-16 | Du Pont Merck Pharma | Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors. |
US5849911A (en) * | 1996-04-22 | 1998-12-15 | Novartis Finance Corporation | Antivirally active heterocyclic azahexane derivatives |
AU2003253992A1 (en) * | 2002-07-18 | 2004-02-09 | Robert P. Bennett | Viral vectors containing recombination sites |
EP2463268B1 (de) * | 2004-12-02 | 2013-08-28 | Daiichi Sankyo Company, Limited | 4-(Aminomethyl)benzoesäuren als Zwischenverbindungen für die Herstellung von Chymase-hemmende 1,4-Diazepan-2,5-dion-Verbindungen |
CA2635356C (en) * | 2005-12-29 | 2011-11-01 | Immupharma France Sa | Use of 1,3,5-triazepin-2,6-diones to treat malaria |
US20080031951A1 (en) | 2005-12-29 | 2008-02-07 | Gilles Guichard | Compositions and methods for the inhibition of phospholipase A2 |
CN107750247A (zh) | 2015-03-17 | 2018-03-02 | 里珍纳龙药品有限公司 | 氨基酸酰化试剂及其使用方法 |
US10189864B2 (en) | 2016-02-19 | 2019-01-29 | Lawrence Livermore National Security, Llc | Metal complexes based on a bis(2-pyridylmethyl)amine-based scaffold and methods of making the same |
US10112912B2 (en) * | 2016-03-02 | 2018-10-30 | Lawrence Livermore National Security, Llc | Homopiperazine-based catalysts for neutralization of organophosphorus-based compounds |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES436126A1 (es) * | 1974-11-29 | 1977-04-01 | Sandoz Ag | Un procedimiento para la produccion de derivados de 2, 3-di-hidro-1h-1, 4 diazepina. |
US4002612A (en) * | 1976-04-05 | 1977-01-11 | Morton-Norwich Products, Inc. | 1-(3,4-Dichlorobenzyl)hexahydro-1,3-diazepin-2(1H)-one |
US4190571A (en) * | 1977-09-21 | 1980-02-26 | The B. F. Goodrich Company | Substituted 2-keto-1,4-diazacycloalkanes and UV-light-stabilized compositions containing them |
US4466916A (en) * | 1979-10-26 | 1984-08-21 | The B. F. Goodrich Company | Substituted 2-keto-1,4-diazacycloalkanes |
US5438118A (en) * | 1990-11-30 | 1995-08-01 | Smithkline Beechman Corp. | HIV protease inhibitors |
US5663333A (en) * | 1992-10-22 | 1997-09-02 | The Dupont Merck Pharmaceutical Company | Substituted 1,4-diazapine caprolactams useful for treatment of HIV disease |
AU5359594A (en) * | 1992-10-22 | 1994-05-09 | Du Pont Merck Pharmaceutical Company, The | Substituted caprolactams and derivatives thereof useful for treatment of aids |
EP0708760A1 (de) * | 1993-07-14 | 1996-05-01 | Novartis AG | Cyclische hydrazin-verbindungen |
-
1993
- 1993-03-30 US US08/040,324 patent/US5663333A/en not_active Expired - Lifetime
-
1994
- 1994-03-28 AT AT94911704T patent/ATE213233T1/de not_active IP Right Cessation
- 1994-03-28 AU AU64159/94A patent/AU6415994A/en not_active Abandoned
- 1994-03-28 WO PCT/US1994/003224 patent/WO1994022840A1/en active IP Right Grant
- 1994-03-28 DE DE69429856T patent/DE69429856D1/de not_active Expired - Lifetime
- 1994-03-28 EP EP94911704A patent/EP0691961B1/de not_active Expired - Lifetime
- 1994-03-28 CA CA002159442A patent/CA2159442A1/en not_active Abandoned
-
1997
- 1997-05-23 US US08/862,560 patent/US5877170A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP0691961B1 (de) | 2002-02-13 |
CA2159442A1 (en) | 1994-10-13 |
EP0691961A1 (de) | 1996-01-17 |
US5663333A (en) | 1997-09-02 |
AU6415994A (en) | 1994-10-24 |
US5877170A (en) | 1999-03-02 |
WO1994022840A1 (en) | 1994-10-13 |
DE69429856D1 (de) | 2002-03-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |