ATE194988T1 - Bicyclische nonan-und decanverbindungen mit dopamine-rezeptor-affinitaet - Google Patents

Bicyclische nonan-und decanverbindungen mit dopamine-rezeptor-affinitaet

Info

Publication number
ATE194988T1
ATE194988T1 AT95937148T AT95937148T ATE194988T1 AT E194988 T1 ATE194988 T1 AT E194988T1 AT 95937148 T AT95937148 T AT 95937148T AT 95937148 T AT95937148 T AT 95937148T AT E194988 T1 ATE194988 T1 AT E194988T1
Authority
AT
Austria
Prior art keywords
4alkyl
dopamine receptor
compounds
nonanene
decanene
Prior art date
Application number
AT95937148T
Other languages
English (en)
Inventor
Patricia L Power
Sumanas Rakhit
Original Assignee
Allelix Biopharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allelix Biopharma filed Critical Allelix Biopharma
Application granted granted Critical
Publication of ATE194988T1 publication Critical patent/ATE194988T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT95937148T 1994-12-12 1995-12-08 Bicyclische nonan-und decanverbindungen mit dopamine-rezeptor-affinitaet ATE194988T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/354,906 US5576314A (en) 1994-12-12 1994-12-12 Bicyclic nonane and decane compounds having dopamine receptor affinity
PCT/IB1995/001110 WO1996018630A1 (en) 1994-12-12 1995-12-08 Bicyclic nonane and decane compounds having dopamine receptor affinity

Publications (1)

Publication Number Publication Date
ATE194988T1 true ATE194988T1 (de) 2000-08-15

Family

ID=23395404

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95937148T ATE194988T1 (de) 1994-12-12 1995-12-08 Bicyclische nonan-und decanverbindungen mit dopamine-rezeptor-affinitaet

Country Status (7)

Country Link
US (2) US5576314A (de)
EP (1) EP0797577B1 (de)
AT (1) ATE194988T1 (de)
AU (1) AU3934795A (de)
CA (1) CA2207546A1 (de)
DE (1) DE69518165T2 (de)
WO (1) WO1996018630A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5576314A (en) * 1994-12-12 1996-11-19 Allelix Biopharmaceuticals Inc. Bicyclic nonane and decane compounds having dopamine receptor affinity
HUP0003718A3 (en) 1997-09-02 2002-11-28 Welfide Corp Fused thiophene derivatives, use thereof and pharmaceutical compositions containing them
US6251893B1 (en) * 1998-06-15 2001-06-26 Nps Allelix Corp. Bicyclic piperidine and piperazine compounds having 5-HT6 receptor affinity
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
GB9926303D0 (en) * 1999-11-05 2000-01-12 Smithkline Beecham Plc Novel compounds
US6890919B2 (en) * 2001-06-26 2005-05-10 Shitij Kapur Atypical antipsychotic agents having low affinity for the D2 receptor
FR2928150A1 (fr) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens
EP2145891A1 (de) * 2008-07-09 2010-01-20 Vetoquinol S.A. 9-substierte 5-Carboxy-Oxadiazin-Chinolon-Derivate, ihre Herstellung und ihre Anwendung als antibakterielle Mittel

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA772160A (en) * 1967-11-21 Schmutz Jean Diazepine and thiazepine derivatives
NL140242B (nl) * 1963-03-01 1973-11-15 Wander Ag Dr A Werkwijze voor het bereiden van op de 11-plaats door een basische groep gesubstitueerde dibenz (b.f.)(1.4) oxazepinen.
US3908010A (en) * 1967-03-22 1975-09-23 Wander Ag Dr A Basically substituted heterocycles as anti-emetics
US3751415A (en) * 1967-03-22 1973-08-07 Sandoz Ag 2-nitro-11-(1-piperazinyl)-dibenz(b,f)(1,4)oxazepines
US3758479A (en) * 1967-03-22 1973-09-11 Sandoz Ag Nitro and sulphamoyl substituted dibenzodiazepines
US3539573A (en) * 1967-03-22 1970-11-10 Jean Schmutz 11-basic substituted dibenzodiazepines and dibenzothiazepines
US3983234A (en) * 1974-07-04 1976-09-28 Sandoz Ltd. Treatment of dyskinesias
US4096261A (en) * 1977-02-23 1978-06-20 Abbott Laboratories Dibenzodiazepines
DD151166A1 (de) * 1979-11-05 1981-10-08 Carla Rueger Verfahren zur herstellung von in 11-stellung substituierten 5h-dibenzo eckige klammer auf b,e eckige klammer zu eckige klammer auf 1,4 eckige klammer zu diazepinen
SU1015618A1 (ru) * 1980-01-28 1986-12-15 Научно-исследовательский институт фармакологии АМН СССР 11- @ -(Диазабицикло (4. @ . @ )алканил) @ -5 @ -дибензо-( @ , @ ) (1,4)диазепины,обладающие нейролиптическим действием
CS224988B1 (cs) * 1982-08-17 1984-02-13 Jilek Jiri Derivát oktahydropyrrolo(l,2-a)pyrazinu a jeho methansulfonát
US5393752A (en) * 1992-05-26 1995-02-28 Therabel Research S.A./N.V. Methylpiperazinoazepine compounds, preparation and use thereof
US5354747A (en) * 1993-06-16 1994-10-11 G. D. Searle & Co. 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- and/or 10-substituted dibenzoxazepine and dibenzthiazepine compounds, pharmaceutical compositions and methods of use
US5576314A (en) * 1994-12-12 1996-11-19 Allelix Biopharmaceuticals Inc. Bicyclic nonane and decane compounds having dopamine receptor affinity

Also Published As

Publication number Publication date
US5703072A (en) 1997-12-30
AU3934795A (en) 1996-07-03
DE69518165D1 (de) 2000-08-31
CA2207546A1 (en) 1996-06-20
EP0797577B1 (de) 2000-07-26
WO1996018630A1 (en) 1996-06-20
EP0797577A1 (de) 1997-10-01
DE69518165T2 (de) 2001-06-07
US5576314A (en) 1996-11-19

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