ATE192650T1 - Verwendung von efaroxan und dessen derivaten zur herstellung eines arzneimittels zur behandlung parkinsonscher krankheit - Google Patents
Verwendung von efaroxan und dessen derivaten zur herstellung eines arzneimittels zur behandlung parkinsonscher krankheitInfo
- Publication number
- ATE192650T1 ATE192650T1 AT94919712T AT94919712T ATE192650T1 AT E192650 T1 ATE192650 T1 AT E192650T1 AT 94919712 T AT94919712 T AT 94919712T AT 94919712 T AT94919712 T AT 94919712T AT E192650 T1 ATE192650 T1 AT E192650T1
- Authority
- AT
- Austria
- Prior art keywords
- efaroxan
- parkinson
- disease
- derivatives
- treatment
- Prior art date
Links
- RATZLMXRALDSJW-UHFFFAOYSA-N 2-(2-ethyl-3H-benzofuran-2-yl)-4,5-dihydro-1H-imidazole Chemical compound C1C2=CC=CC=C2OC1(CC)C1=NCCN1 RATZLMXRALDSJW-UHFFFAOYSA-N 0.000 title abstract 2
- 208000018737 Parkinson disease Diseases 0.000 title abstract 2
- 229950001765 efaroxan Drugs 0.000 title abstract 2
- 229940126601 medicinal product Drugs 0.000 title abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Psychology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9307379A FR2706303B1 (fr) | 1993-06-18 | 1993-06-18 | Utilisation de l'Efaroxan et de ses dérivés pour la préparation d'un médicament destiné au traitement de la maladie de Parkinson. |
| PCT/FR1994/000715 WO1995000145A1 (fr) | 1993-06-18 | 1994-06-15 | Utilisation de l'efaroxan et de ses derives pour la preparation d'un medicament destine au traitement de la maladie de parkinson |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE192650T1 true ATE192650T1 (de) | 2000-05-15 |
Family
ID=9448287
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT94919712T ATE192650T1 (de) | 1993-06-18 | 1994-06-15 | Verwendung von efaroxan und dessen derivaten zur herstellung eines arzneimittels zur behandlung parkinsonscher krankheit |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US5948806A (de) |
| EP (1) | EP0703781B1 (de) |
| JP (1) | JP3394257B2 (de) |
| AT (1) | ATE192650T1 (de) |
| AU (1) | AU689783B2 (de) |
| CA (1) | CA2165437A1 (de) |
| DE (1) | DE69424415T2 (de) |
| DK (1) | DK0703781T3 (de) |
| ES (1) | ES2147576T3 (de) |
| FR (1) | FR2706303B1 (de) |
| GR (1) | GR3034062T3 (de) |
| NZ (1) | NZ268039A (de) |
| PT (1) | PT703781E (de) |
| WO (1) | WO1995000145A1 (de) |
| ZA (1) | ZA944281B (de) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6281207B1 (en) * | 1999-09-15 | 2001-08-28 | Reed Richter | Treatment of movement disorders by administration of mirtazapine |
| FR2814368B1 (fr) * | 2000-09-26 | 2004-05-07 | Pf Medicament | Preparation pharmaceutique a base d'oxans |
| US20040039041A1 (en) * | 2000-11-14 | 2004-02-26 | Antti Haapalinna | Prevention of development of dyskinesias |
| US8188126B2 (en) | 2002-05-16 | 2012-05-29 | Pierre Fabre Medicament | Imidazolic compounds and use thereof as alpha-2 adrenergic receptors |
| US9463186B2 (en) | 2013-04-15 | 2016-10-11 | Northwestern University | Treatment for dopaminergic disorders |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZW13782A1 (en) * | 1981-07-28 | 1982-10-06 | Reckitt & Colmann Prod Ltd | Imidazoline derivatives |
| FR2669030B1 (fr) * | 1990-11-14 | 1992-12-31 | Adir | Nouveaux derives d'imidazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US5281607B1 (en) * | 1992-10-08 | 1998-05-19 | Univ New York | Method of using alpha 2-antagonists for the treatment of neurodegenerative diseases |
-
1993
- 1993-06-18 FR FR9307379A patent/FR2706303B1/fr not_active Expired - Lifetime
-
1994
- 1994-06-15 WO PCT/FR1994/000715 patent/WO1995000145A1/fr not_active Ceased
- 1994-06-15 CA CA002165437A patent/CA2165437A1/fr not_active Abandoned
- 1994-06-15 AU AU70764/94A patent/AU689783B2/en not_active Ceased
- 1994-06-15 JP JP50249995A patent/JP3394257B2/ja not_active Expired - Fee Related
- 1994-06-15 DE DE69424415T patent/DE69424415T2/de not_active Expired - Fee Related
- 1994-06-15 EP EP94919712A patent/EP0703781B1/de not_active Expired - Lifetime
- 1994-06-15 NZ NZ268039A patent/NZ268039A/xx unknown
- 1994-06-15 ES ES94919712T patent/ES2147576T3/es not_active Expired - Lifetime
- 1994-06-15 AT AT94919712T patent/ATE192650T1/de not_active IP Right Cessation
- 1994-06-15 DK DK94919712T patent/DK0703781T3/da active
- 1994-06-15 PT PT94919712T patent/PT703781E/pt unknown
- 1994-06-16 ZA ZA944281A patent/ZA944281B/xx unknown
-
1997
- 1997-03-26 US US08/825,414 patent/US5948806A/en not_active Expired - Fee Related
-
2000
- 2000-07-28 GR GR20000401754T patent/GR3034062T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DK0703781T3 (da) | 2000-10-02 |
| FR2706303B1 (fr) | 1995-09-08 |
| EP0703781B1 (de) | 2000-05-10 |
| NZ268039A (en) | 1999-06-29 |
| CA2165437A1 (fr) | 1994-12-19 |
| JP3394257B2 (ja) | 2003-04-07 |
| WO1995000145A1 (fr) | 1995-01-05 |
| JPH09500375A (ja) | 1997-01-14 |
| EP0703781A1 (de) | 1996-04-03 |
| PT703781E (pt) | 2000-10-31 |
| DE69424415T2 (de) | 2000-12-21 |
| FR2706303A1 (fr) | 1994-12-23 |
| US5948806A (en) | 1999-09-07 |
| ZA944281B (en) | 1995-02-10 |
| ES2147576T3 (es) | 2000-09-16 |
| GR3034062T3 (en) | 2000-11-30 |
| DE69424415D1 (de) | 2000-06-15 |
| AU7076494A (en) | 1995-01-17 |
| AU689783B2 (en) | 1998-04-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |