ATA782177A - METHOD FOR PRODUCING NEW CIS-4A-ARYLOCTAHYDRO-1H-2-PYRINDINE COMPOUNDS AND THE NON-TOXIC PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF - Google Patents

METHOD FOR PRODUCING NEW CIS-4A-ARYLOCTAHYDRO-1H-2-PYRINDINE COMPOUNDS AND THE NON-TOXIC PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF

Info

Publication number
ATA782177A
ATA782177A AT0782177A AT782177A ATA782177A AT A782177 A ATA782177 A AT A782177A AT 0782177 A AT0782177 A AT 0782177A AT 782177 A AT782177 A AT 782177A AT A782177 A ATA782177 A AT A782177A
Authority
AT
Austria
Prior art keywords
aryloctahydro
pyrindine
compounds
pharmaceutically acceptable
acid addition
Prior art date
Application number
AT0782177A
Other languages
German (de)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of ATA782177A publication Critical patent/ATA782177A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/757Unsaturated compounds containing a keto groups being part of a ring containing —CHO groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/94Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
AT0782177A 1976-11-02 1977-11-02 METHOD FOR PRODUCING NEW CIS-4A-ARYLOCTAHYDRO-1H-2-PYRINDINE COMPOUNDS AND THE NON-TOXIC PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF ATA782177A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73795876A 1976-11-02 1976-11-02

Publications (1)

Publication Number Publication Date
ATA782177A true ATA782177A (en) 1981-10-15

Family

ID=24965981

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0782177A ATA782177A (en) 1976-11-02 1977-11-02 METHOD FOR PRODUCING NEW CIS-4A-ARYLOCTAHYDRO-1H-2-PYRINDINE COMPOUNDS AND THE NON-TOXIC PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF

Country Status (26)

Country Link
JP (1) JPS5356669A (en)
AR (1) AR223454A1 (en)
AT (1) ATA782177A (en)
AU (1) AU513679B2 (en)
BE (1) BE860314A (en)
CA (1) CA1100136A (en)
CS (1) CS211380B2 (en)
DD (1) DD133795A5 (en)
DE (1) DE2748466A1 (en)
DK (1) DK485277A (en)
ES (3) ES463784A1 (en)
FR (1) FR2369267A1 (en)
GB (1) GB1590155A (en)
GR (1) GR70053B (en)
HU (1) HU176231B (en)
IE (1) IE45901B1 (en)
IL (1) IL53236A0 (en)
NL (1) NL7712053A (en)
NZ (1) NZ185539A (en)
PH (1) PH12590A (en)
PL (3) PL108610B1 (en)
PT (1) PT67194B (en)
RO (3) RO77935A (en)
SE (3) SE7712218L (en)
SU (3) SU812174A3 (en)
ZA (1) ZA776497B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT68934A (en) * 1977-12-27 1979-01-01 Lilly Co Eli Process for preparing 4a-aryl-octahydro-1h-2-pyrindines
US4236009A (en) * 1979-06-21 1980-11-25 Eli Lilly And Company Method of preparing 4A-arylhexahydro-1H-2-pyrindines and 4A-aryloctahydroisoquinolines
US4277608A (en) * 1979-06-21 1981-07-07 Eli Lilly And Company Method of preparing 4a-arylhexahydro-1H-2-pyrindines and 4a-aryloctahydroisoquinolines
ZA9510829B (en) * 1994-12-23 1996-07-03 Smithkline Beecham Corp 3,3-(disubstituted)cyclohexan-1-one monomers and related compounds
EP2595989B1 (en) 2010-05-06 2016-07-13 Vertex Pharmaceuticals Incorporated Heterocyclic chromene-spirocyclic piperidine amides as modulators of ion channels
US8916565B2 (en) 2011-02-02 2014-12-23 Vertex Pharmaceuticals Incorporated Pyrrolopyrazine-spirocyclic piperidine amides as modulators of ion channels
US10385070B2 (en) 2011-02-18 2019-08-20 Vertex Pharmaceuticals Incorporated Chroman-spirocyclic piperidine amides as modulators of ion channels
US8828996B2 (en) 2011-03-14 2014-09-09 Vertex Pharmaceuticals Incorporated Morpholine-spirocyclic piperidine amides as modulators of ion channels

Also Published As

Publication number Publication date
NL7712053A (en) 1978-05-05
RO77935A (en) 1981-12-25
AU513679B2 (en) 1980-12-18
PL108466B1 (en) 1980-04-30
PL109690B1 (en) 1980-06-30
RO78300A (en) 1982-04-12
FR2369267A1 (en) 1978-05-26
GB1590155A (en) 1981-05-28
AR223454A1 (en) 1981-08-31
SE8103107L (en) 1981-05-18
DE2748466A1 (en) 1978-05-03
DD133795A5 (en) 1979-01-24
SE7712218L (en) 1978-05-02
ES463783A1 (en) 1979-07-16
HU176231B (en) 1981-01-28
NZ185539A (en) 1979-12-11
PL201885A1 (en) 1978-12-04
PH12590A (en) 1979-06-27
ZA776497B (en) 1979-06-27
IE45901B1 (en) 1982-12-29
DK485277A (en) 1978-05-03
PT67194B (en) 1979-03-23
SU812174A3 (en) 1981-03-07
JPS5356669A (en) 1978-05-23
ES463784A1 (en) 1978-06-16
PL108610B1 (en) 1980-04-30
SE8103106L (en) 1981-05-18
CA1100136A (en) 1981-04-28
AU3023577A (en) 1979-05-10
CS211380B2 (en) 1982-02-26
SU913941A3 (en) 1982-03-15
ES472276A1 (en) 1979-10-01
RO72900A (en) 1981-11-04
BE860314A (en) 1978-04-28
GR70053B (en) 1982-07-26
IE45901L (en) 1978-05-02
SU845777A3 (en) 1981-07-07
IL53236A0 (en) 1977-12-30
FR2369267B1 (en) 1980-05-16
PT67194A (en) 1977-11-01

Similar Documents

Publication Publication Date Title
AT359488B (en) METHOD FOR PRODUCING NEW PHTHALANE DERIVATIVES AND THEIR PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS
AT357143B (en) METHOD FOR PRODUCING NEW SUBSTITUTED 3-PHENOXY-2-HYDROXY-1-AMINOPROPANES AND THEIR ACID ADDITION SALTS
AT363465B (en) METHOD FOR PRODUCING NEW 5-AROYL-1,2-DIHYDRO-3H-PYRROLO- (1,2-A) -PYRROL-1-CARBONIC ACID ESTERS AND SALTS
AT367430B (en) METHOD FOR PRODUCING NEW HYDROXYLAMINO-HYDROCARBYLPHOSPHONIC ACID DERIVATIVES
AT358035B (en) METHOD FOR PRODUCING NEW INDOLICINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT360533B (en) METHOD FOR PRODUCING NEW TRANS- HEXAHYDROPYRIDO-INDOLES AND THEIR ACID ADDITION SALTS
AT359523B (en) METHOD FOR PRODUCING NEW 6-AMINO-ALKYLAMINOURACILES AND THEIR ACID ADDITION SALTS
AT354436B (en) METHOD FOR PRODUCING NEW 2-BROMO-6-FLUOR-N-2-IMIDAZOLIDINYLIDENE-BENZAMINE AND ITS ACID ADDITION SALTS
AT373580B (en) METHOD FOR PRODUCING NEW SUBSTITUTED 2-BENZYLPYRROLIDINES, THEIR QUATERIAL ALKYL COMPOUNDS AND THEIR ACID ADDITION SALTS
ATA782177A (en) METHOD FOR PRODUCING NEW CIS-4A-ARYLOCTAHYDRO-1H-2-PYRINDINE COMPOUNDS AND THE NON-TOXIC PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF
AT356110B (en) METHOD FOR PRODUCING NEW BENZYLISO-CHINOLINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT361904B (en) METHOD FOR PRODUCING NEW 3-ANILINO-AETHYLAMINO-2-HYDROXY-1-PHENOXYPROPANES AND THEIR ACID ADDITION SALTS
AT363928B (en) METHOD FOR PRODUCING NEW HYDRAZONE COMPOUNDS AND PHARMACOLOGICALLY COMPATIBLE ACID ADDITION SALTS AND QUATERNAUS AMMONIUM SALTS THEREOF
AT359521B (en) METHOD FOR PRODUCING NEW ISOTHIO-UREA AMINOALKYLAETHERS AND THEIR SALTS
AT353960B (en) METHOD FOR PRODUCING NEW BIS-PENI-CILLANOYLOXY ALKANS AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS
AT365170B (en) METHOD FOR PRODUCING NEW 13-THIAPROSTANIC ACID DERIVATIVES
AT360029B (en) METHOD FOR PRODUCING NEW 2,4-DIAMINO -5-THIOBENZYLPYRIMIDINES AND THEIR ACID ADDITION SALTS
AT358046B (en) METHOD FOR PRODUCING NEW TRANS-5A- ARYL DECAHYDROBENZAZEPINES AND THEIR ACID ADDITION SALTS
ATA392379A (en) METHOD FOR PRODUCING NEW BENZO (C) -QUINOLINES AND THEIR PHARMACEUTICALLY COMPATIBLE ACID ADDITION SALTS
ATA162476A (en) METHOD FOR PRODUCING NEW PHENOXY-PHENYLBUTTERIC ACID DERIVATIVES AND ITS SALTS
AT357692B (en) METHOD FOR PRODUCING 4-DESACETOXY- -VINBLASTIN AND ITS ACID ADDITION SALTS
AT360675B (en) METHOD FOR PRODUCING NEW TETRADECAPEPTIDES AND THEIR PHARMACEUTICAL ACCEPTABLE NON-TOXIC ACID ADDITION SALTS
ATA95279A (en) METHOD FOR PRODUCING NEW INDOLICINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA59280A (en) METHOD FOR PRODUCING NEW 3-ANILINOAETHYLAMINO-2-HYDROXY-1-PHENOXYPROPANES AND THEIR ACID ADDITION SALTS
AT363941B (en) METHOD FOR PRODUCING NEW AMINOALKYLHETEROCYCLES AND THEIR ACID ADDITION SALTS

Legal Events

Date Code Title Description
A1AW Revocation of published examined application