ATA649276A - PROCESS FOR THE PREPARATION OF NEW 2,4-DIAMINO-5-BENZYLPYRIMIDINES AND THEIR ACID ADDITIONAL SALTS - Google Patents

PROCESS FOR THE PREPARATION OF NEW 2,4-DIAMINO-5-BENZYLPYRIMIDINES AND THEIR ACID ADDITIONAL SALTS

Info

Publication number
ATA649276A
ATA649276A AT649276A AT649276A ATA649276A AT A649276 A ATA649276 A AT A649276A AT 649276 A AT649276 A AT 649276A AT 649276 A AT649276 A AT 649276A AT A649276 A ATA649276 A AT A649276A
Authority
AT
Austria
Prior art keywords
benzylpyrimidines
diamino
preparation
new
additional salts
Prior art date
Application number
AT649276A
Other languages
German (de)
Other versions
AT352735B (en
Original Assignee
Heumann Ludwig & Co Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Heumann Ludwig & Co Gmbh filed Critical Heumann Ludwig & Co Gmbh
Publication of ATA649276A publication Critical patent/ATA649276A/en
Application granted granted Critical
Publication of AT352735B publication Critical patent/AT352735B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT649276A 1975-10-17 1976-09-01 PROCESS FOR THE PREPARATION OF NEW 2,4-DIAMINO-5-BENZYLPYRIMIDINES AND THEIR ACID ADDITIONAL SALTS AT352735B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2546667A DE2546667C3 (en) 1975-10-17 1975-10-17 2,4-DiamuH »-5- (3-methoxy-4-hydroxy-5-halobenzyl) -pyrimidines, and medicinal products containing these compounds

Publications (2)

Publication Number Publication Date
ATA649276A true ATA649276A (en) 1979-03-15
AT352735B AT352735B (en) 1979-10-10

Family

ID=5959437

Family Applications (1)

Application Number Title Priority Date Filing Date
AT649276A AT352735B (en) 1975-10-17 1976-09-01 PROCESS FOR THE PREPARATION OF NEW 2,4-DIAMINO-5-BENZYLPYRIMIDINES AND THEIR ACID ADDITIONAL SALTS

Country Status (17)

Country Link
JP (1) JPS5251376A (en)
AR (1) AR210905A1 (en)
AT (1) AT352735B (en)
AU (1) AU1724576A (en)
BE (1) BE846397A (en)
CA (1) CA1055498A (en)
CH (1) CH623313A5 (en)
DE (1) DE2546667C3 (en)
ES (1) ES451375A1 (en)
FR (1) FR2327786A1 (en)
GB (1) GB1522537A (en)
GR (1) GR60352B (en)
HU (1) HU174155B (en)
IL (1) IL50430A0 (en)
MX (1) MX4485E (en)
NL (1) NL7609652A (en)
PT (1) PT65482B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2720771C3 (en) 1977-05-09 1979-11-29 Ludwig Heumann & Co Gmbh, 8500 Nuernberg 2,4-Diamino-5- (33-dimethoxy-4thioalkyl-benzyD-pyrimidines, process for their preparation and pharmaceuticals containing these compounds
ZW9979A1 (en) * 1978-05-24 1980-12-24 Wellcome Found Benzylpyrimidine compositions
HU188588B (en) * 1982-08-13 1986-04-28 Egyt Gyogyszervegyeszeti Gyar Process for the production of 2,4-diamino-5-benzyl-pyrimidine-derivatives

Also Published As

Publication number Publication date
MX4485E (en) 1982-05-21
NL7609652A (en) 1977-04-19
ES451375A1 (en) 1981-10-16
CA1055498A (en) 1979-05-29
GR60352B (en) 1978-05-18
DE2546667A1 (en) 1977-04-28
GB1522537A (en) 1978-08-23
BE846397A (en) 1977-01-17
DE2546667B2 (en) 1978-02-09
DE2546667C3 (en) 1978-10-12
PT65482B (en) 1978-02-13
FR2327786A1 (en) 1977-05-13
AR210905A1 (en) 1977-09-30
JPS5251376A (en) 1977-04-25
IL50430A0 (en) 1976-11-30
AT352735B (en) 1979-10-10
AU1724576A (en) 1978-03-02
PT65482A (en) 1976-09-01
HU174155B (en) 1979-11-28
FR2327786B1 (en) 1980-04-18
CH623313A5 (en) 1981-05-29

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Legal Events

Date Code Title Description
EIH Change in the person of patent owner
ELJ Ceased due to non-payment of the annual fee