ATA5962001A - Hydrophobisierte teilchen von k-clavulanat - Google Patents

Hydrophobisierte teilchen von k-clavulanat

Info

Publication number
ATA5962001A
ATA5962001A AT5962001A AT5962001A ATA5962001A AT A5962001 A ATA5962001 A AT A5962001A AT 5962001 A AT5962001 A AT 5962001A AT 5962001 A AT5962001 A AT 5962001A AT A5962001 A ATA5962001 A AT A5962001A
Authority
AT
Austria
Prior art keywords
clavulanat
hydrophobized particles
hydrophobized
particles
Prior art date
Application number
AT5962001A
Other languages
English (en)
Other versions
AT412344B (de
Inventor
Otto Ing Daemon
Herwig Dr Jennewein
Thomas Lentner
Franz Xaver Ing Schwarz
Robert Veigl
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Priority to AT5962001A priority Critical patent/AT412344B/de
Priority to PCT/EP2002/004062 priority patent/WO2002083129A2/en
Priority to AU2002315287A priority patent/AU2002315287A1/en
Priority to US10/474,480 priority patent/US20040132712A1/en
Priority to EP02740465A priority patent/EP1381362A2/de
Publication of ATA5962001A publication Critical patent/ATA5962001A/de
Application granted granted Critical
Publication of AT412344B publication Critical patent/AT412344B/de
Priority to US11/449,041 priority patent/US20060263424A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
AT5962001A 2001-04-12 2001-04-12 Hydrophobisierte teilchen von k-clavulanat AT412344B (de)

Priority Applications (6)

Application Number Priority Date Filing Date Title
AT5962001A AT412344B (de) 2001-04-12 2001-04-12 Hydrophobisierte teilchen von k-clavulanat
PCT/EP2002/004062 WO2002083129A2 (en) 2001-04-12 2002-04-11 Pharmaceutical composition comprising clavulanic acid
AU2002315287A AU2002315287A1 (en) 2001-04-12 2002-04-11 Pharmaceutical composition comprising clavulanic acid
US10/474,480 US20040132712A1 (en) 2001-04-12 2002-04-11 Pharmaceutical compositions comprising clavulanic acid
EP02740465A EP1381362A2 (de) 2001-04-12 2002-04-11 Pharmazeutische zusammensetzung entahaltend clavulansäure
US11/449,041 US20060263424A1 (en) 2001-04-12 2006-06-07 Pharmaceutical compositions comprising clavulanic acid

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
AT5962001A AT412344B (de) 2001-04-12 2001-04-12 Hydrophobisierte teilchen von k-clavulanat

Publications (2)

Publication Number Publication Date
ATA5962001A true ATA5962001A (de) 2004-06-15
AT412344B AT412344B (de) 2005-01-25

Family

ID=32398592

Family Applications (1)

Application Number Title Priority Date Filing Date
AT5962001A AT412344B (de) 2001-04-12 2001-04-12 Hydrophobisierte teilchen von k-clavulanat

Country Status (1)

Country Link
AT (1) AT412344B (de)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57171918A (en) * 1981-04-17 1982-10-22 Eisai Co Ltd Theophyllin gradually releasing composition
EP0080862B1 (de) * 1981-12-02 1985-09-25 Beecham Group Plc Pharmazeutische Zubereitung die Beta-Lactam Antibiotika enthält
GB9109862D0 (en) * 1991-05-08 1991-07-03 Beecham Lab Sa Pharmaceutical formulations
GB9405856D0 (en) * 1994-03-24 1994-05-11 Smithkline Beecham Plc Pharmaceutical formulation
PL334976A1 (en) * 1997-02-14 2000-03-27 Smithkline Beecham Lab Pharmaceutic preparations containing amoxycyclin and clavulate
TR200000529T2 (tr) * 1997-08-29 2000-08-21 Dsm N.V. İçinde eksipiyan olmayan granüller
BR9806280A (pt) * 1997-11-17 2000-02-15 Gist Brocades Bv Grânulos compreendendo clavulaneto e um ou mais excipientes

Also Published As

Publication number Publication date
AT412344B (de) 2005-01-25

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee