AT368994B - METHOD FOR PRODUCING NEW N-PHENYL-N- (4-PIPERIDINYL) AMIDES AND THEIR ACID ADDITION SALTS - Google Patents

METHOD FOR PRODUCING NEW N-PHENYL-N- (4-PIPERIDINYL) AMIDES AND THEIR ACID ADDITION SALTS

Info

Publication number
AT368994B
AT368994B AT0322078A AT322078A AT368994B AT 368994 B AT368994 B AT 368994B AT 0322078 A AT0322078 A AT 0322078A AT 322078 A AT322078 A AT 322078A AT 368994 B AT368994 B AT 368994B
Authority
AT
Austria
Prior art keywords
piperidinyl
amides
phenyl
acid addition
addition salts
Prior art date
Application number
AT0322078A
Other languages
German (de)
Other versions
ATA322078A (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ATA322078A publication Critical patent/ATA322078A/en
Application granted granted Critical
Publication of AT368994B publication Critical patent/AT368994B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
AT0322078A 1977-05-05 1978-05-03 METHOD FOR PRODUCING NEW N-PHENYL-N- (4-PIPERIDINYL) AMIDES AND THEIR ACID ADDITION SALTS AT368994B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79381477A 1977-05-05 1977-05-05
US88618878A 1978-03-13 1978-03-13

Publications (2)

Publication Number Publication Date
ATA322078A ATA322078A (en) 1982-04-15
AT368994B true AT368994B (en) 1982-11-25

Family

ID=27121432

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0322078A AT368994B (en) 1977-05-05 1978-05-03 METHOD FOR PRODUCING NEW N-PHENYL-N- (4-PIPERIDINYL) AMIDES AND THEIR ACID ADDITION SALTS

Country Status (26)

Country Link
JP (1) JPS53149980A (en)
AT (1) AT368994B (en)
AU (1) AU514360B2 (en)
CA (1) CA1105464A (en)
CH (1) CH635585A5 (en)
CY (1) CY1253A (en)
DE (1) DE2819873A1 (en)
DK (1) DK152211C (en)
ES (1) ES469473A1 (en)
FI (1) FI64364C (en)
FR (1) FR2389622B1 (en)
GB (1) GB1598872A (en)
HK (1) HK72585A (en)
HU (1) HU179204B (en)
IE (1) IE46836B1 (en)
IL (1) IL54639A (en)
IT (1) IT1105288B (en)
KE (1) KE3429A (en)
LU (1) LU79575A1 (en)
NL (1) NL186861C (en)
NO (1) NO148747C (en)
NZ (1) NZ187164A (en)
PH (1) PH12831A (en)
SE (1) SE437516B (en)
SU (1) SU867304A3 (en)
YU (1) YU40703B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6144294A (en) * 1984-08-07 1986-03-03 Nippon Denso Co Ltd Heat exchanger
US5053411A (en) * 1989-04-20 1991-10-01 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
USRE34201E (en) * 1989-04-20 1993-03-23 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
JPH08193074A (en) * 1994-11-18 1996-07-30 Nippon Bayeragrochem Kk Herbicidal 1-cyclopropyltetrazolinones
JP2000327668A (en) * 1999-05-21 2000-11-28 Nippon Bayer Agrochem Co Ltd Tetrazolinone derivative
JP2003515588A (en) * 1999-12-06 2003-05-07 マリンクロッド・インコーポレイテッド New synthetic route to alfentanil, sufentanil and remifentanil
WO2006030931A1 (en) * 2004-09-14 2006-03-23 Nippon Chemiphar Co., Ltd. N-substituted n-(4-piperidinyl)amide derivative

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3998834A (en) * 1975-03-14 1976-12-21 Janssen Pharmaceutica N.V. N-(4-piperidinyl)-n-phenylamides and -carbamates

Also Published As

Publication number Publication date
DK193778A (en) 1978-11-06
SU867304A3 (en) 1981-09-23
CY1253A (en) 1984-08-31
YU40703B (en) 1986-04-30
AU514360B2 (en) 1981-02-05
KE3429A (en) 1984-08-10
JPS6324995B2 (en) 1988-05-23
NZ187164A (en) 1981-03-16
PH12831A (en) 1979-09-05
CA1105464A (en) 1981-07-21
SE7805110L (en) 1978-11-06
ES469473A1 (en) 1979-09-16
FI64364B (en) 1983-07-29
NO781559L (en) 1978-11-07
NO148747C (en) 1983-12-07
NL186861B (en) 1990-10-16
DE2819873A1 (en) 1978-11-09
DK152211C (en) 1988-08-08
FI781398A (en) 1978-11-06
DE2819873C2 (en) 1989-05-03
HU179204B (en) 1982-09-28
IT7849203A0 (en) 1978-05-04
ATA322078A (en) 1982-04-15
FR2389622B1 (en) 1982-05-21
NL186861C (en) 1991-03-18
HK72585A (en) 1985-10-04
FR2389622A1 (en) 1978-12-01
IL54639A (en) 1982-02-28
CH635585A5 (en) 1983-04-15
GB1598872A (en) 1981-09-23
AU3552278A (en) 1979-11-01
NO148747B (en) 1983-08-29
NL7804844A (en) 1978-11-07
YU108578A (en) 1983-01-21
IL54639A0 (en) 1978-07-31
FI64364C (en) 1983-11-10
DK152211B (en) 1988-02-08
SE437516B (en) 1985-03-04
IE46836B1 (en) 1983-10-05
IT1105288B (en) 1985-10-28
LU79575A1 (en) 1978-11-03
IE780901L (en) 1978-11-05
JPS53149980A (en) 1978-12-27

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee
ELA Expired due to lapse of time