AR241136A1 - Procedimiento para preparar esteres de 6-hidroxi-2-benzotiazolsulfonamida para tratamiento topicode presion intraocular elevada" - Google Patents
Procedimiento para preparar esteres de 6-hidroxi-2-benzotiazolsulfonamida para tratamiento topicode presion intraocular elevada"Info
- Publication number
- AR241136A1 AR241136A1 AR289937A AR28993782A AR241136A1 AR 241136 A1 AR241136 A1 AR 241136A1 AR 289937 A AR289937 A AR 289937A AR 28993782 A AR28993782 A AR 28993782A AR 241136 A1 AR241136 A1 AR 241136A1
- Authority
- AR
- Argentina
- Prior art keywords
- topicode
- benzotiazolsulfonamide
- hydroxy
- esters
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
- C07D277/76—Sulfur atoms attached to a second hetero atom
- C07D277/80—Sulfur atoms attached to a second hetero atom to a nitrogen atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US28247081A | 1981-07-13 | 1981-07-13 | |
US35240082A | 1982-02-25 | 1982-02-25 |
Publications (2)
Publication Number | Publication Date |
---|---|
AR241136A2 AR241136A2 (es) | 1991-11-29 |
AR241136A1 true AR241136A1 (es) | 1991-11-29 |
Family
ID=26961471
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR289937A AR241136A1 (es) | 1981-07-13 | 1982-06-08 | Procedimiento para preparar esteres de 6-hidroxi-2-benzotiazolsulfonamida para tratamiento topicode presion intraocular elevada" |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0070239B1 (es) |
AR (1) | AR241136A1 (es) |
AU (1) | AU556363B2 (es) |
CA (1) | CA1185980A (es) |
DE (1) | DE3264033D1 (es) |
DK (1) | DK312082A (es) |
ES (1) | ES8400417A1 (es) |
FI (1) | FI78080C (es) |
GR (1) | GR76527B (es) |
IE (1) | IE53868B1 (es) |
IL (1) | IL66238A0 (es) |
NO (1) | NO157538C (es) |
NZ (1) | NZ201157A (es) |
PT (1) | PT75229B (es) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5095026A (en) * | 1983-02-04 | 1992-03-10 | University Of Iowa Research Foundation | Prodrugs of carbonic anhydrase inhibitors |
US4500538A (en) * | 1983-03-14 | 1985-02-19 | Merck & Co., Inc. | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure |
US4499103A (en) * | 1983-03-17 | 1985-02-12 | Merck & Co., Inc. | Benzothiazole-2-sulfonamide derivatives for the topical treatment of elevated intraocular pressure |
US4472418A (en) * | 1983-04-22 | 1984-09-18 | Merck & Co., Inc. | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure |
US4456599A (en) * | 1983-04-22 | 1984-06-26 | Merck & Co., Inc. | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure |
US4470991A (en) * | 1983-04-22 | 1984-09-11 | Merck & Co., Inc. | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure |
US4472417A (en) * | 1983-04-22 | 1984-09-18 | Merck & Co., Inc. | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure |
ES8600752A1 (es) * | 1983-06-20 | 1985-10-16 | Merck & Co Inc | Un procedimiento para la preparacion de nuevos derivados de tiosulfonamida. |
NZ208444A (en) * | 1983-06-20 | 1987-08-31 | Merck & Co Inc | 2-thiophene derivatives and pharmaceutical compositions |
US4544667A (en) * | 1984-02-09 | 1985-10-01 | Merck & Co., Inc. | 2-Sulfamoylbenzo[b]furan derivatives for the treatment of elevated intraocular pressure |
EP0155214B1 (en) * | 1984-03-14 | 1990-03-14 | Merck & Co. Inc. | 2-sulfamoyl-1h-indole derivatives for the treatment of elevated intraocular pressure |
US5059613A (en) * | 1990-03-19 | 1991-10-22 | Research Corporation Technologies, Inc. | Topically active ocular benzothiazole sulfonamide carbonic anhydrase inhibitors |
US5519040A (en) * | 1994-04-29 | 1996-05-21 | Allergan | Substituted thiazole sulfonamides as antiglaucoma agents |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2595334A (en) * | 1950-04-08 | 1952-05-06 | American Cyanamid Co | Benzothiazolesulfonamides and method of preparing the same |
US2868800A (en) * | 1954-10-13 | 1959-01-13 | Upjohn Co | 6-ethoxybenzothiazole-2-sulfonamide |
-
1982
- 1982-06-08 AR AR289937A patent/AR241136A1/es active
- 1982-07-05 NZ NZ201157A patent/NZ201157A/en unknown
- 1982-07-06 IL IL66238A patent/IL66238A0/xx not_active IP Right Cessation
- 1982-07-07 GR GR68682A patent/GR76527B/el unknown
- 1982-07-09 CA CA000407023A patent/CA1185980A/en not_active Expired
- 1982-07-09 FI FI822464A patent/FI78080C/fi not_active IP Right Cessation
- 1982-07-09 ES ES513831A patent/ES8400417A1/es not_active Expired
- 1982-07-09 EP EP82401299A patent/EP0070239B1/en not_active Expired
- 1982-07-09 DE DE8282401299T patent/DE3264033D1/de not_active Expired
- 1982-07-09 AU AU85775/82A patent/AU556363B2/en not_active Ceased
- 1982-07-12 IE IE1668/82A patent/IE53868B1/en unknown
- 1982-07-12 NO NO822410A patent/NO157538C/no unknown
- 1982-07-12 DK DK312082A patent/DK312082A/da not_active Application Discontinuation
- 1982-07-12 PT PT75229A patent/PT75229B/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NZ201157A (en) | 1985-02-28 |
IL66238A0 (en) | 1982-11-30 |
NO822410L (no) | 1983-01-14 |
AR241136A2 (es) | 1991-11-29 |
FI822464A0 (fi) | 1982-07-09 |
FI822464L (fi) | 1983-01-14 |
PT75229B (en) | 1985-10-04 |
DK312082A (da) | 1983-01-14 |
FI78080B (fi) | 1989-02-28 |
IE53868B1 (en) | 1989-03-29 |
DE3264033D1 (en) | 1985-07-11 |
GR76527B (es) | 1984-08-10 |
IE821668L (en) | 1983-01-13 |
NO157538B (no) | 1987-12-28 |
CA1185980A (en) | 1985-04-23 |
PT75229A (en) | 1982-08-01 |
NO157538C (no) | 1988-04-06 |
AU8577582A (en) | 1983-01-20 |
AU556363B2 (en) | 1986-10-30 |
FI78080C (fi) | 1989-06-12 |
ES513831A0 (es) | 1983-11-01 |
EP0070239A1 (en) | 1983-01-19 |
EP0070239B1 (en) | 1985-06-05 |
ES8400417A1 (es) | 1983-11-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE3364150D1 (en) | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure | |
ES525435A0 (es) | Procedimiento para la produccion de n-piridinsulfonil-n'-pirimidinil- y -triacinilureas | |
GB2091441B (en) | Applanation tonometer | |
ES518875A0 (es) | Procedimiento para la produccion de n-aril-sulfonil-n'-pirimidil-ureas. | |
ES489358A0 (es) | Procedimiento para la preparacion de un hidrolizado de pro- teinas purificado. | |
ES514868A0 (es) | "un procedimiento para la preparacion de un derivado de tiazol". | |
ES511835A0 (es) | "procedimiento para la preparacion de nuevas piriimidinonas". | |
ES515453A0 (es) | "procedimiento para la preparacion de esteres perfluoroalcohilicos". | |
AR241136A1 (es) | Procedimiento para preparar esteres de 6-hidroxi-2-benzotiazolsulfonamida para tratamiento topicode presion intraocular elevada" | |
ES512913A0 (es) | "procedimiento para la preparacion de nuevas fenilalcohilaminas". | |
ES510677A0 (es) | "procedimiento para la preparacion de acidos oxazafosforin-4-tio-alcansulfonicos". | |
EP0122831A3 (en) | Benzothiazole-2-sulfonamide derivatives for the topical treatment of elevated intraocular pressure | |
GB2061956B (en) | Process for the preparation of keratin hydrolysates | |
ES508811A0 (es) | "prodedimiento para la preparacion de derivados de fenoxi-aminipropanol" | |
ES530388A0 (es) | Procedimiento para preparar derivados del 2-azabiciclo-2.2.1-heptano. | |
ES525709A0 (es) | Procedimiento para formar un producto de polivinilpirrolidona o copolimero de vinilpirrolidona-acetato de vinilo | |
IT1110132B (it) | Procedimento per la fabbricazione di sigarette presentanti un filtro di estremita' | |
ZA842959B (en) | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure | |
ZA842665B (en) | Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure | |
ZA848451B (en) | Ethers of hydroxybenzothiazole-2-sulfonamide for the topical treatment of elevated intraocular pressure | |
ZA842958B (en) | Benzothiazolesulfonamide for the topical treatment of elevated intraocular pressure | |
ES514456A0 (es) | "un procedimiento para la preparacion de esteres de 2-tenoilmercaptopropionilglicina". | |
ES516605A0 (es) | "procedimiento para la produccion o tratamiento de ferrocromo". | |
ES512769A0 (es) | "procedimiento para la preparacion de esteres 2-metoxifenilicos de aminoacidos n-substituidos". | |
ZA844114B (en) | 6(or 5)-hydroxybenzothiazole-2-sulfonamide-o-sulfate salts for the topical treatment of elevated intraocular pressure |