AR230422A1 - Procedimiento para preparar el acido(2',4'-difluoro-4-bifenil)-oxipropionico de accion analgesica y anti-inflamatoria - Google Patents

Procedimiento para preparar el acido(2',4'-difluoro-4-bifenil)-oxipropionico de accion analgesica y anti-inflamatoria

Info

Publication number
AR230422A1
AR230422A1 AR289467A AR28946782A AR230422A1 AR 230422 A1 AR230422 A1 AR 230422A1 AR 289467 A AR289467 A AR 289467A AR 28946782 A AR28946782 A AR 28946782A AR 230422 A1 AR230422 A1 AR 230422A1
Authority
AR
Argentina
Prior art keywords
oxipropionico
analgesic
difluoro
biphenyl
procedure
Prior art date
Application number
AR289467A
Other languages
English (en)
Original Assignee
Ausonia Farma Srl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ausonia Farma Srl filed Critical Ausonia Farma Srl
Application granted granted Critical
Publication of AR230422A1 publication Critical patent/AR230422A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/58Unsaturated compounds containing ether groups, groups, groups, or groups
    • C07C59/64Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
    • C07C59/66Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings
    • C07C59/68Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR289467A 1981-11-24 1982-05-20 Procedimiento para preparar el acido(2',4'-difluoro-4-bifenil)-oxipropionico de accion analgesica y anti-inflamatoria AR230422A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8125243A IT1211135B (it) 1981-11-24 1981-11-24 Composti ad attivita'analgesica e antiinfiammatoria, processo per la loro preparazione e relative composizioni farmaceutiche.

Publications (1)

Publication Number Publication Date
AR230422A1 true AR230422A1 (es) 1984-04-30

Family

ID=11216107

Family Applications (1)

Application Number Title Priority Date Filing Date
AR289467A AR230422A1 (es) 1981-11-24 1982-05-20 Procedimiento para preparar el acido(2',4'-difluoro-4-bifenil)-oxipropionico de accion analgesica y anti-inflamatoria

Country Status (13)

Country Link
US (1) US4440787A (es)
EP (1) EP0080010B1 (es)
JP (1) JPS5892636A (es)
KR (1) KR830010038A (es)
AR (1) AR230422A1 (es)
AT (1) ATE14720T1 (es)
CA (1) CA1185617A (es)
DE (1) DE3265210D1 (es)
ES (1) ES8302623A1 (es)
GR (1) GR75481B (es)
IT (1) IT1211135B (es)
PT (1) PT74937A (es)
ZA (1) ZA823487B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL83109A (en) * 1986-07-11 1992-06-21 Ciba Geigy Ag Guanidinium aspartates,their preparation and pharmaceutical compositions containing them
US4883818A (en) * 1987-11-17 1989-11-28 Analgesic Associates Onset-hastened/enhanced analgesia
US4927854A (en) * 1987-12-24 1990-05-22 Analgesic Associates Sustained/enhanced analgesia
US5286751A (en) * 1987-12-24 1994-02-15 Analgesic Associates Sustained/enhanced antipyretic response
ES2079997A1 (es) * 1993-06-15 1996-01-16 Lilly Co Eli Compuestos de fenil fenol sustituidos antagonistas de leucotrieno, procedimiento para su obtencion y formulaciones farmaceuticas de los mismos.
MX2015016543A (es) * 2013-06-27 2017-07-27 Lg Chemical Ltd Derivados de biarilo como agonistas de gpr120.
CN115925679A (zh) * 2014-12-24 2023-04-07 株式会社Lg化学 作为gpr120激动剂的联芳基衍生物

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1121722A (en) * 1966-03-31 1968-07-31 Ici Ltd New carboxylic acid derivatives
US3755603A (en) * 1970-07-01 1973-08-28 Syntex Corp Biphenylyloxyacetic acids in pharmaceutical compositions
US4021479A (en) * 1971-03-17 1977-05-03 Boehringer Ingelheim Gmbh Derivatives of 4-(4-biphenylyl)-butyric acid
US3948973A (en) * 1972-08-29 1976-04-06 Sterling Drug Inc. Halocyclopropyl substituted phenoxyalkanoic acids
GB1459084A (en) * 1973-05-24 1976-12-22 Boots Co Ltd Preparation of arylalkanoic acid
US4188491A (en) * 1975-04-04 1980-02-12 The Boots Company Limited Preparation of therapeutic compounds
US4151302A (en) * 1975-06-28 1979-04-24 Merck Patent Gesellschaft Mit Beschrankter Haftung Araliphatic dihalogen compounds composition and method of use
US4189499A (en) * 1977-03-16 1980-02-19 Biochefarm S.A. Lysine 4-allyloxy-3-chlorophenylacetate and method of its preparation
US4225730A (en) * 1978-05-11 1980-09-30 Merck & Co., Inc. Process for preparing 4-(2,4-difluorophenyl)-salicyclic acid
JPS5576840A (en) * 1978-12-01 1980-06-10 Kaken Pharmaceut Co Ltd New oxyacetic acid derivative, its preparation and blood- lipid depressor containing it as active principle
IT1141655B (it) * 1980-02-12 1986-10-08 Schiapparelli Spa Nuovi derivati dell'acido propanoico ad attivita' ipolipidemica e ipocolesterolemica

Also Published As

Publication number Publication date
ATE14720T1 (de) 1985-08-15
IT1211135B (it) 1989-09-29
ZA823487B (en) 1983-04-27
IT8125243A0 (it) 1981-11-24
DE3265210D1 (en) 1985-09-12
EP0080010A1 (en) 1983-06-01
CA1185617A (en) 1985-04-16
JPS6124374B2 (es) 1986-06-10
JPS5892636A (ja) 1983-06-02
US4440787A (en) 1984-04-03
GR75481B (es) 1984-07-23
KR830010038A (ko) 1983-12-24
ES512387A0 (es) 1983-02-01
ES8302623A1 (es) 1983-02-01
PT74937A (en) 1982-06-01
EP0080010B1 (en) 1985-08-07

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