AR221682A1 - PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2 (IMIDAZOL-4-IL, PIRIDIL-2-ILO OR TIAZOLIL-2-ILO-BUTIL OR METHYLTIO-ETILAMINO) -5- (1-NAFTIL-ALQUILENOXI; 1,3-BENZODIOXOLIL-ALQUILENOXI ; 1,4-BENZODIOXINILALQUILENOXI; 1-NAFTILALQUILEN; 1,3-BENZODIOXOLILALQUILEN; OR 1,4-BENZO DIOXINILALQUILEN) -4-PIRIMIDONA O 4-PIRIMIDINTIONA - Google Patents

PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2 (IMIDAZOL-4-IL, PIRIDIL-2-ILO OR TIAZOLIL-2-ILO-BUTIL OR METHYLTIO-ETILAMINO) -5- (1-NAFTIL-ALQUILENOXI; 1,3-BENZODIOXOLIL-ALQUILENOXI ; 1,4-BENZODIOXINILALQUILENOXI; 1-NAFTILALQUILEN; 1,3-BENZODIOXOLILALQUILEN; OR 1,4-BENZO DIOXINILALQUILEN) -4-PIRIMIDONA O 4-PIRIMIDINTIONA

Info

Publication number
AR221682A1
AR221682A1 AR264926A AR26492676A AR221682A1 AR 221682 A1 AR221682 A1 AR 221682A1 AR 264926 A AR264926 A AR 264926A AR 26492676 A AR26492676 A AR 26492676A AR 221682 A1 AR221682 A1 AR 221682A1
Authority
AR
Argentina
Prior art keywords
alquilenoxi
ilo
pirimidona
pirimidintiona
naftilalquilen
Prior art date
Application number
AR264926A
Other languages
Spanish (es)
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Application granted granted Critical
Publication of AR221682A1 publication Critical patent/AR221682A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60Three or more oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56One oxygen atom and one sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR264926A 1975-10-02 1976-09-30 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2 (IMIDAZOL-4-IL, PIRIDIL-2-ILO OR TIAZOLIL-2-ILO-BUTIL OR METHYLTIO-ETILAMINO) -5- (1-NAFTIL-ALQUILENOXI; 1,3-BENZODIOXOLIL-ALQUILENOXI ; 1,4-BENZODIOXINILALQUILENOXI; 1-NAFTILALQUILEN; 1,3-BENZODIOXOLILALQUILEN; OR 1,4-BENZO DIOXINILALQUILEN) -4-PIRIMIDONA O 4-PIRIMIDINTIONA AR221682A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4034175 1975-10-02

Publications (1)

Publication Number Publication Date
AR221682A1 true AR221682A1 (en) 1981-03-13

Family

ID=10414412

Family Applications (1)

Application Number Title Priority Date Filing Date
AR264926A AR221682A1 (en) 1975-10-02 1976-09-30 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 2 (IMIDAZOL-4-IL, PIRIDIL-2-ILO OR TIAZOLIL-2-ILO-BUTIL OR METHYLTIO-ETILAMINO) -5- (1-NAFTIL-ALQUILENOXI; 1,3-BENZODIOXOLIL-ALQUILENOXI ; 1,4-BENZODIOXINILALQUILENOXI; 1-NAFTILALQUILEN; 1,3-BENZODIOXOLILALQUILEN; OR 1,4-BENZO DIOXINILALQUILEN) -4-PIRIMIDONA O 4-PIRIMIDINTIONA

Country Status (36)

Country Link
JP (2) JPS5246087A (en)
AR (1) AR221682A1 (en)
AT (1) AT358045B (en)
AU (1) AU504897B2 (en)
BE (1) BE846452A (en)
BG (1) BG25224A3 (en)
CA (1) CA1067076A (en)
CH (1) CH625801A5 (en)
CS (1) CS203003B2 (en)
DD (1) DD126563A5 (en)
DE (1) DE2643670C2 (en)
DK (1) DK442476A (en)
ES (1) ES452060A1 (en)
FI (1) FI61701C (en)
FR (1) FR2326192A1 (en)
GR (1) GR61307B (en)
HU (1) HU175537B (en)
IE (1) IE44845B1 (en)
IL (1) IL50503A (en)
IN (1) IN146736B (en)
IT (2) IT1070839B (en)
LU (1) LU75922A1 (en)
MW (1) MW3476A1 (en)
MX (1) MX4614E (en)
NL (1) NL7609917A (en)
NO (1) NO145792C (en)
NZ (1) NZ181959A (en)
OA (1) OA05445A (en)
PH (1) PH13921A (en)
PL (1) PL105828B1 (en)
PT (1) PT65590B (en)
RO (1) RO73511A (en)
SE (1) SE431872B (en)
YU (1) YU237276A (en)
ZA (1) ZA765498B (en)
ZM (1) ZM12176A1 (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MW5076A1 (en) * 1975-12-29 1978-02-08 Smith Kline French Lab Pharmacologicalle active compounds
NZ186511A (en) 1977-03-19 1980-11-14 Smith Kline French Lab 3-substituted alkylamino-6-substituted alkyl-1,2,4-triazin-5-ones and pharmaceutical compositions 3-substituted thio-1,2,4-triazin-5-ones
US4165378A (en) 1977-04-20 1979-08-21 Ici Americas Inc. Guanidine derivatives of imidazoles and thiazoles
NZ186965A (en) 1977-04-20 1980-02-21 Ici Ltd Guanidino derivatives and pharmaceutical compositions
JPS54104816A (en) * 1978-01-27 1979-08-17 Memorex Corp Magnetic recorder tape reel
IN151188B (en) * 1978-02-13 1983-03-05 Smith Kline French Lab
IL57005A (en) * 1978-04-11 1983-11-30 Smith Kline French Lab Process for the preparation of 2-amino pyrimid-4-one derivatives and novel 2-nitroaminopyrimid-4-ones as intermediates therefor
IL57416A (en) * 1978-05-30 1983-03-31 Smith Kline French Lab Nitro compounds,processes for preparing them and compositions containing them
ZA793443B (en) * 1978-07-26 1980-12-31 Glaxo Group Ltd Heterocyclic derivatives
US4374836A (en) 1978-10-16 1983-02-22 Imperial Chemical Industries Ltd. Antisecretory heterocyclic derivatives, process for their manufacture and pharmaceutical compositions containing them
US4496567A (en) * 1978-11-13 1985-01-29 Smith Kline & French Laboratories Limited Phenyl alkylaminopyrimidones
US4521418A (en) * 1979-02-21 1985-06-04 Smith Kline & French Laboratories Limited Guanidinothiazolyl derivatives
JPS55145683A (en) * 1979-04-26 1980-11-13 Smith Kline French Lab Pyrimidone derivative
CA1155842A (en) * 1980-03-29 1983-10-25 Thomas H. Brown Compounds
ZW21281A1 (en) * 1980-10-01 1981-11-18 Smith Kline French Lab Amine derivatives
IE53068B1 (en) * 1981-06-15 1988-05-25 Merck & Co Inc Diamino isothiazole-1-oxides and -1,1-dioxides as gastic secretion inhibitors
PT75074B (en) * 1981-06-27 1986-02-26 Smith Kline French Lab Process for preparing certain pyrimidone derivatives and compositions containing them
NZ202797A (en) * 1981-12-28 1985-08-30 Lilly Co Eli Pyrimidine derivatives and pharmaceutical compositions
JPS5993074A (en) * 1982-10-01 1984-05-29 スミス・クライン・アンド・フレンチ・ラボラトリ−ス・リミテツド Pyrimidone derivative
DE8309239U1 (en) * 1983-03-29 1983-09-29 Basf Ag, 6700 Ludwigshafen TAPE REEL, IN PARTICULAR FOR MAGNETIC TAPES

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1397436A (en) * 1972-09-05 1975-06-11 Smith Kline French Lab Heterocyclic n-cyanoguinidines
GB1419994A (en) * 1973-05-03 1976-01-07 Smith Kline French Lab Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them

Also Published As

Publication number Publication date
FR2326192B1 (en) 1979-01-12
CS203003B2 (en) 1981-02-27
CH625801A5 (en) 1981-10-15
ZA765498B (en) 1977-08-31
RO73511A (en) 1981-04-30
BG25224A3 (en) 1978-08-10
IE44845B1 (en) 1982-04-21
FR2326192A1 (en) 1977-04-29
HU175537B (en) 1980-08-28
JPS609755B2 (en) 1985-03-12
PL105828B1 (en) 1979-11-30
GR61307B (en) 1978-10-19
ES452060A1 (en) 1977-10-01
PT65590A (en) 1976-10-01
AU1829576A (en) 1978-04-06
DE2643670A1 (en) 1977-04-14
IE44845L (en) 1977-04-02
ATA711976A (en) 1980-01-15
LU75922A1 (en) 1977-05-06
CA1067076A (en) 1979-11-27
NO145792C (en) 1982-06-02
YU237276A (en) 1983-01-21
IL50503A0 (en) 1976-11-30
JPS5246087A (en) 1977-04-12
FI61701C (en) 1982-09-10
DE2643670C2 (en) 1982-07-01
DD126563A5 (en) 1977-07-27
NO763371L (en) 1977-04-05
PH13921A (en) 1980-11-04
MW3476A1 (en) 1977-11-09
BE846452A (en) 1977-03-22
MX4614E (en) 1982-07-07
SE7610409L (en) 1977-04-03
JPS5695186A (en) 1981-08-01
JPS5635674B2 (en) 1981-08-19
AT358045B (en) 1980-08-11
NL7609917A (en) 1977-04-05
ZM12176A1 (en) 1977-07-21
FI762803A (en) 1977-04-03
DK442476A (en) 1977-04-03
IL50503A (en) 1980-12-31
NO145792B (en) 1982-02-22
SE431872B (en) 1984-03-05
FI61701B (en) 1982-05-31
AU504897B2 (en) 1979-11-01
PT65590B (en) 1978-03-28
IN146736B (en) 1979-08-25
IT1070839B (en) 1985-04-02
NZ181959A (en) 1978-07-28
IT7830708A0 (en) 1978-12-11
OA05445A (en) 1981-03-31

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