AR215134A1 - Procedimiento para preparar nuevas 1-amidino-3-fenilureas - Google Patents

Procedimiento para preparar nuevas 1-amidino-3-fenilureas

Info

Publication number
AR215134A1
AR215134A1 AR266807A AR26680777A AR215134A1 AR 215134 A1 AR215134 A1 AR 215134A1 AR 266807 A AR266807 A AR 266807A AR 26680777 A AR26680777 A AR 26680777A AR 215134 A1 AR215134 A1 AR 215134A1
Authority
AR
Argentina
Prior art keywords
phenylureas
amidino
procedure
prepare new
prepare
Prior art date
Application number
AR266807A
Other languages
English (en)
Inventor
Julius Diamond
George Henry Douglas
Original Assignee
Rorer Inc William H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19762629756 external-priority patent/DE2629756A1/de
Application filed by Rorer Inc William H filed Critical Rorer Inc William H
Application granted granted Critical
Publication of AR215134A1 publication Critical patent/AR215134A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR266807A 1975-03-31 1977-03-10 Procedimiento para preparar nuevas 1-amidino-3-fenilureas AR215134A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/558,187 US4060635A (en) 1975-03-31 1975-03-31 Amidinoureas for treating diarrhea
DE19762629756 DE2629756A1 (de) 1973-07-16 1976-07-02 1-amidin-3-substituierte phenylharnstoffe und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
AR215134A1 true AR215134A1 (es) 1979-09-14

Family

ID=25770652

Family Applications (2)

Application Number Title Priority Date Filing Date
AR262513A AR216898A1 (es) 1975-03-31 1976-03-11 Procedimiento para preparar nuevas 1-amidino-3-fenilureas
AR266807A AR215134A1 (es) 1975-03-31 1977-03-10 Procedimiento para preparar nuevas 1-amidino-3-fenilureas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR262513A AR216898A1 (es) 1975-03-31 1976-03-11 Procedimiento para preparar nuevas 1-amidino-3-fenilureas

Country Status (8)

Country Link
US (1) US4060635A (es)
AR (2) AR216898A1 (es)
AU (1) AU504728B2 (es)
CA (1) CA1064934A (es)
CH (1) CH635823A5 (es)
EG (1) EG12773A (es)
GB (1) GB1538158A (es)
GR (1) GR59274B (es)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4488993A (en) * 1972-09-22 1984-12-18 William H. Rorer, Inc. Amidinoureas
US4326074A (en) * 1972-09-22 1982-04-20 William H. Rorer, Inc. Amidinoureas
US4204000A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Anti-ulcer amidinoureas
US4203920A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Amidinoureas
US4353842A (en) * 1978-09-14 1982-10-12 William H. Rorer, Inc. Amidinoureas
US4203985A (en) * 1978-11-13 1980-05-20 William H. Rorer, Inc. Antidiarrheal triazinones
US4241087A (en) * 1979-04-02 1980-12-23 William H. Rorer, Inc. Dysmenorrhea treatment
US4279928A (en) * 1979-04-02 1981-07-21 William H. Rorer, Inc. Method of lowering blood pressure
US4418209A (en) * 1980-04-14 1983-11-29 William H. Rorer, Inc. Amidinothioureas
US4443456A (en) * 1981-05-12 1984-04-17 William H. Rorer, Inc. Pyridyl alkylene amidinoureas
US4565826A (en) * 1981-05-12 1986-01-21 William H. Rorer, Inc. Heterocyclic amidinoureas
US4704401A (en) * 1981-07-06 1987-11-03 Rorer Pharmaceutical Corporation Substituted phenyl amidinoureas
US4487779A (en) * 1981-07-06 1984-12-11 William H. Rorer, Inc. Substituted phenyl amidinoureas
AU543834B2 (en) * 1981-08-24 1985-05-02 Rorer International (Overseas) Inc. Heterocyclic amidino substituted ureas and their pharmaceutical uses
US4562209A (en) * 1981-08-24 1985-12-31 William H. Rorer, Inc. Promotion of feed efficiency in animals
US4575514A (en) * 1982-12-20 1986-03-11 Mcneilab, Inc. Anxiety alleviating compositions containing loweralkyl-N-[amino(arylaminocarbonyl)-iminomethyl]-N-methylglycinates
US4714707A (en) * 1984-01-13 1987-12-22 Rorer Pharmaceutical Corporation Aryl substituted heterocycles for treating gastrointestinal motility dysfunction
JPS62501839A (ja) * 1985-02-15 1987-07-23 ロウラ−　インタ−ナシヨナル（オ−バ−シ−ズ）　インコ−ポレ−テツド アミジノ尿素の製造法および医薬用組成物
AU605584B2 (en) * 1987-04-10 1991-01-17 Reanal Finomvegyszergyar Method for the preparation of amidino-urea derivatives
US6190691B1 (en) 1994-04-12 2001-02-20 Adolor Corporation Methods for treating inflammatory conditions
US5962477A (en) * 1994-04-12 1999-10-05 Adolor Corporation Screening methods for cytokine inhibitors
US5849761A (en) * 1995-09-12 1998-12-15 Regents Of The University Of California Peripherally active anti-hyperalgesic opiates
US6573282B1 (en) 1995-09-12 2003-06-03 Adolor Corporation Peripherally active anti-hyperalgesic opiates
US5667773A (en) * 1996-03-12 1997-09-16 Adolor Corporation Film-forming compositions of antihyperalgesic opiates and method of treating hyperalgesic conditions therewith
US5888494A (en) * 1996-03-12 1999-03-30 Adolor Corporation Film-forming compositions of antihyperalgesic opiates and method of treating hyperalgesic and pruritic conditions therewith
US5849762A (en) * 1997-07-14 1998-12-15 Adolor Corporation Peripherally acting anti-pruritic opiates
US6353004B1 (en) 1997-07-14 2002-03-05 Adolor Coporation Peripherally acting anti-pruritic opiates
CN104383542B (zh) 2003-04-08 2017-09-26 普罗热尼奇制药公司 包含甲基纳曲酮的药物配方
AR057325A1 (es) 2005-05-25 2007-11-28 Progenics Pharm Inc Sintesis de (s)-n-metilnaltrexona, composiciones farmaceuticas y usos
AR057035A1 (es) 2005-05-25 2007-11-14 Progenics Pharm Inc SíNTESIS DE (R)-N-METILNALTREXONA, COMPOSICIONES FARMACÉUTICAS Y USOS
MX351611B (es) 2007-03-29 2017-10-20 Wyeth Llc Formas de cristal de bromuro de (r)-n-metilnaltrexona y uso de las mismas.
SI2139890T1 (sl) 2007-03-29 2014-12-31 Wyeth Llc Antagonisti perifernih opioidnih receptorjev in njih uporaba
PA8774201A1 (es) 2007-03-29 2009-06-23 Progenics Pharm Inc Antagonista del receptor
EP2730578A1 (en) 2008-02-06 2014-05-14 Progenics Pharmaceuticals, Inc. Preparation and use of (r),(r)-2,2'-bis-methylnal trexone
CA2676881C (en) 2008-09-30 2017-04-25 Wyeth Peripheral opioid receptor antagonists and uses thereof
KR101705446B1 (ko) * 2014-04-29 2017-02-09 가톨릭대학교 산학협력단 면역질환 치료효과를 갖는 신규한 화합물 및 이의 용도

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1194835A (en) * 1966-07-07 1970-06-10 Wellcome Found Novel 1-Amidino-3-Phenyl-Urea Derivatives, the preparation thereof and Compositions containing the same

Also Published As

Publication number Publication date
AR216898A1 (es) 1980-02-15
US4060635A (en) 1977-11-29
AU504728B2 (en) 1979-10-25
GR59274B (en) 1977-12-05
EG12773A (en) 1979-12-31
CH635823A5 (de) 1983-04-29
CA1064934A (en) 1979-10-23
GB1538158A (en) 1979-01-10
AU1230276A (en) 1977-09-29

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