AR205402A1 - Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazina - Google Patents
Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazinaInfo
- Publication number
- AR205402A1 AR205402A1 AR260094A AR26009475A AR205402A1 AR 205402 A1 AR205402 A1 AR 205402A1 AR 260094 A AR260094 A AR 260094A AR 26009475 A AR26009475 A AR 26009475A AR 205402 A1 AR205402 A1 AR 205402A1
- Authority
- AR
- Argentina
- Prior art keywords
- antraniloil
- sulfamoil
- elaboration
- piperazine
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH764373 | 1973-05-28 | ||
CH450774 | 1974-04-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR205402A1 true AR205402A1 (es) | 1976-04-30 |
Family
ID=25695649
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR260094A AR205402A1 (es) | 1973-05-28 | 1975-01-01 | Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazina |
Country Status (10)
Country | Link |
---|---|
US (1) | US3933802A (es) |
JP (1) | JPS5019760A (es) |
AR (1) | AR205402A1 (es) |
AU (1) | AU6939974A (es) |
DE (1) | DE2423847A1 (es) |
DK (1) | DK285974A (es) |
FR (1) | FR2231381A1 (es) |
IL (1) | IL44864A0 (es) |
LU (1) | LU70158A1 (es) |
NL (1) | NL7406684A (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2611705A1 (de) * | 1976-03-18 | 1977-09-22 | Josef Dipl Chem Dr Rer N Klosa | N-5-(nitrofurfuryliden-)-1-amino- hydantoin enthaltende kristalloesungsmittel |
US4268536A (en) * | 1978-12-07 | 1981-05-19 | Western Electric Company, Inc. | Method for depositing a metal on a surface |
JPS56124740A (en) * | 1980-02-29 | 1981-09-30 | Mitsubishi Electric Corp | Bushing |
GB8823775D0 (en) * | 1988-10-11 | 1988-11-16 | Scras | New 2-carbonyl substituted n n'-di-(trimethoxybenzoyl)piperazines |
GB0030710D0 (en) * | 2000-12-15 | 2001-01-31 | Hoffmann La Roche | Piperazine derivatives |
CA2537292C (en) * | 2003-09-09 | 2013-04-02 | F. Hoffmann-La Roche Ag | 1- (2-amino-benzol) -piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses |
KR100880093B1 (ko) * | 2004-12-09 | 2009-01-23 | 에프. 호프만-라 로슈 아게 | 페닐-피페라진 메탄온 유도체 |
JP4709849B2 (ja) * | 2004-12-15 | 2011-06-29 | エフ.ホフマン−ラ ロシュ アーゲー | アルツハイマー病治療のためのグリシントランスポーターi(glyt−1)インヒビターとしての二環式及び三環式置換フェニルメタノン類 |
US7485637B2 (en) * | 2005-01-04 | 2009-02-03 | Hoffmann-La Roche Inc. | Benzoyl-tetrahydropiperidine derivatives |
CA2593453A1 (en) * | 2005-01-06 | 2006-07-13 | F. Hoffmann-La Roche Ag | Sulfanyl substituted phenyl methanones as glycine transporter 1 (glyt-1) inhibitors for the treatment of neurological and neuropsychiatric disorders |
CA2593463C (en) * | 2005-01-07 | 2013-10-08 | F. Hoffmann-La Roche Ag | [4-(heteroaryl) piperazin-1-yl]-(2,5-substituted -phenyl)methanone derivatives as glycine transporter 1 (glyt-1) inhibitors for the treatment of neurological and neuropsychiatric disorders |
AU2006207650B2 (en) * | 2005-01-18 | 2011-01-27 | F. Hoffmann-La Roche Ag | 2, 5-disubstituted phenyl methanone derivatives as glycine transporter 1 (GlyT-I) inhibitors for the treatment of neurological and neuropsychiatry disorders |
EP1844045B1 (en) * | 2005-01-26 | 2009-11-04 | F.Hoffmann-La Roche Ag | Phenyl methanone derivatives and their use as glycine transporter 1 inhibitors |
MX2007009342A (es) * | 2005-02-07 | 2007-09-21 | Hoffmann La Roche | Fenil-metanonas sustituidas por heterociclo como inhibidor del transportador 1 de glicina. |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2598E (fr) * | 1903-05-19 | 1904-05-20 | Joseph Francois Antoine Franci | Renforceur du bois pour cannes à peche, mats, vergues, manches et articles d'utilité et de jeux |
US2910488A (en) * | 1958-01-22 | 1959-10-27 | Merck & Co Inc | Aniline derivatives |
CH433378A (de) * | 1962-03-09 | 1967-04-15 | Ciba Geigy | Verfahren zur Herstellung neuer Anthranilsäurederivate |
-
1974
- 1974-05-16 DE DE2423847A patent/DE2423847A1/de active Pending
- 1974-05-17 NL NL7406684A patent/NL7406684A/xx unknown
- 1974-05-20 IL IL44864A patent/IL44864A0/xx unknown
- 1974-05-22 US US05/472,333 patent/US3933802A/en not_active Expired - Lifetime
- 1974-05-27 FR FR7418225A patent/FR2231381A1/fr not_active Withdrawn
- 1974-05-27 AU AU69399/74A patent/AU6939974A/en not_active Expired
- 1974-05-27 DK DK285974A patent/DK285974A/da unknown
- 1974-05-27 LU LU70158*A patent/LU70158A1/xx unknown
- 1974-05-28 JP JP49059409A patent/JPS5019760A/ja active Pending
-
1975
- 1975-01-01 AR AR260094A patent/AR205402A1/es active
Also Published As
Publication number | Publication date |
---|---|
DE2423847A1 (de) | 1975-01-02 |
JPS5019760A (es) | 1975-03-01 |
NL7406684A (es) | 1974-12-02 |
AU6939974A (en) | 1975-11-27 |
IL44864A0 (en) | 1975-02-10 |
FR2231381A1 (es) | 1974-12-27 |
US3933802A (en) | 1976-01-20 |
DK285974A (es) | 1975-01-20 |
LU70158A1 (es) | 1976-04-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR206801A1 (es) | Procedimiento para la elaboracion de derivados del 1-pirid loxi-2-hidroxi-3-amino-propano | |
AR206339A1 (es) | Procedimiento para la preparacion de derivados de 1-(metoxifenil)-4-(3-(naft-1-il-oxi)-2-hidroxi-propil)-piperazina | |
AR202618A1 (es) | Procedimiento para la preparacion de metiltioalquilguanidinas heterociclicas | |
AR205402A1 (es) | Procedimiento para la elaboracion de compuestos de 1-(5-sulfamoil - antraniloil) - piperazina | |
AR206315A1 (es) | Procedimiento para la preparacion de compuestos de cefalosporina | |
AR205619A1 (es) | Procedimiento para la elaboracion de nuevos derivados (2-benzo-furanil)-piperidina | |
AR203222A1 (es) | Procedimiento para la preparacion de compuestos arilacetileno | |
IT995115B (it) | Procedimento per la vinilazione catalitica di composti aromatici | |
AR196775A1 (es) | Procedimiento para la preparacion de derivados de 1-(3-(5,6,7,8-tetrahidronaft-1-ii-oxi)-propil)- piperazina | |
AR205618A1 (es) | Procedimiento para la elaboracion de derivados del 1-(4-alquiltio-alcoxi)-fenoxi - 2 - hidroxi-3-alquilaminopropano | |
AR208184A1 (es) | Procedimiento para la fabricacion de derivados de 2-(aminocarbonil-aza-alcanamido)-benzofenoma | |
AR201343A1 (es) | Procedimiento para la preparacion de compuestos de quinoxalindiona sustituidos | |
AR197989A1 (es) | Procedimiento para la elaboracion de nuevos derivados de diazepina | |
AR200772A1 (es) | Procedimiento para la preparacion de compuestos 1-amino-4-feniltetralinicos | |
AR202476A1 (es) | Procedimiento para la elaboracion de compuestos del 2-hidroxi-3-amino-propoxi- 9,10-dihidroantraceno y sus sales | |
AR202966A1 (es) | Procedimiento para la preparacion de derivados de 1-(3-(naft-1-il-oxi)-propil)-piperazina | |
AR206796A1 (es) | Procedimiento para la elaboracion de nuevos compuestos derivados de cicloalquil-fenilalcanoilpiridinas | |
AR208063A1 (es) | Procedimiento para la elaboracion de nuevos derivados de la 4-anhidrofuranosa | |
AR200519A1 (es) | Procedimiento de preparacion de nuevos derivados de la piperazina | |
AR211695A1 (es) | Procedimiento para la preparacion de derivados de aminoscilanilidas primarias | |
AR207463A1 (es) | Procedimiento para la elaboracion de nuevos derivados de 1-(2-hidroxi-3-fenoxipropil)-piperidina-4-sustituida | |
AR201133A1 (es) | Procedimiento para la fabricacion de fibrillas discontinuas | |
MX3642E (es) | Procedimiento para la preparacion de compuestos de 4-(m-bromofenil)-pirazolodiazepina | |
AR197267A1 (es) | Procedimiento para la fabricacion de 1-(3-hidroxifenil)-2-aminopropanos | |
AR203844A1 (es) | Procedimiento para la elaboracion de nuevos derivados de la anhidrofuranosa |