AR204003A1 - Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables - Google Patents
Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptablesInfo
- Publication number
- AR204003A1 AR204003A1 AR253060A AR25306074A AR204003A1 AR 204003 A1 AR204003 A1 AR 204003A1 AR 253060 A AR253060 A AR 253060A AR 25306074 A AR25306074 A AR 25306074A AR 204003 A1 AR204003 A1 AR 204003A1
- Authority
- AR
- Argentina
- Prior art keywords
- oxopyride
- piperazinyl
- pyrimidine
- procedure
- pharmaceutically acceptable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3845373A JPS5546400B2 (nl) | 1973-04-03 | 1973-04-03 | |
JP5654473A JPS565753B2 (nl) | 1973-05-21 | 1973-05-21 | |
JP6446473A JPS565755B2 (nl) | 1973-06-07 | 1973-06-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR204003A1 true AR204003A1 (es) | 1975-11-12 |
Family
ID=27289838
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR253060A AR204003A1 (es) | 1973-04-03 | 1974-01-01 | Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables |
AR258571A AR204660A1 (es) | 1973-04-03 | 1975-01-01 | Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR258571A AR204660A1 (es) | 1973-04-03 | 1975-01-01 | Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico |
Country Status (11)
Country | Link |
---|---|
AR (2) | AR204003A1 (nl) |
AT (1) | AT340931B (nl) |
CA (1) | CA1066701A (nl) |
CH (1) | CH593281A5 (nl) |
ES (1) | ES424851A1 (nl) |
FI (1) | FI56011C (nl) |
IE (1) | IE39102B1 (nl) |
NL (1) | NL186087C (nl) |
NO (1) | NO142221C (nl) |
PH (2) | PH10529A (nl) |
SE (1) | SE416051B (nl) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1209163B (it) * | 1979-12-21 | 1989-07-10 | Unibios S P A Trecate Novara | Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti. |
PL2448938T3 (pl) | 2009-06-29 | 2014-11-28 | Incyte Holdings Corp | Pirymidynony jako inhibitory PI3K |
AR079529A1 (es) | 2009-12-18 | 2012-02-01 | Incyte Corp | Derivados arilo y heteroarilo sustituidos y fundidos como inhibidores de la pi3k |
WO2011075643A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
TW201249844A (en) | 2010-12-20 | 2012-12-16 | Incyte Corp | N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors |
KR102131612B1 (ko) | 2011-09-02 | 2020-07-08 | 인사이트 홀딩스 코포레이션 | Pi3k 억제제로서 헤테로시클릴아민 |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
WO2015191677A1 (en) | 2014-06-11 | 2015-12-17 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors |
MA41607B1 (fr) | 2015-02-27 | 2021-01-29 | Incyte Corp | Sels d'un inhibiteur de pi3k et procédés de préparation de ces sels |
WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
WO2016183063A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Crystalline forms of a pi3k inhibitor |
-
1974
- 1974-01-01 AR AR253060A patent/AR204003A1/es active
- 1974-01-30 CA CA191,286A patent/CA1066701A/en not_active Expired
- 1974-02-01 SE SE7401361A patent/SE416051B/xx not_active IP Right Cessation
- 1974-02-04 FI FI298/74A patent/FI56011C/fi active
- 1974-02-04 NL NLAANVRAGE7401509,A patent/NL186087C/nl not_active IP Right Cessation
- 1974-02-04 NO NO740349A patent/NO142221C/no unknown
- 1974-02-14 CH CH205474A patent/CH593281A5/de not_active IP Right Cessation
- 1974-03-25 IE IE00650/74A patent/IE39102B1/xx unknown
- 1974-04-02 ES ES424851A patent/ES424851A1/es not_active Expired
- 1974-04-03 AT AT277774A patent/AT340931B/de not_active IP Right Cessation
- 1974-04-03 PH PH15698A patent/PH10529A/en unknown
-
1975
- 1975-01-01 AR AR258571A patent/AR204660A1/es active
- 1975-09-05 PH PH17546A patent/PH10984A/en unknown
Also Published As
Publication number | Publication date |
---|---|
SE416051B (sv) | 1980-11-24 |
NO142221B (no) | 1980-04-08 |
NO740349L (no) | 1974-10-04 |
IE39102B1 (en) | 1978-08-02 |
NO142221C (no) | 1980-07-16 |
FI56011B (fi) | 1979-07-31 |
IE39102L (en) | 1974-10-03 |
ES424851A1 (es) | 1976-06-01 |
ATA277774A (de) | 1977-05-15 |
PH10984A (en) | 1977-10-18 |
CH593281A5 (en) | 1977-11-30 |
FI56011C (fi) | 1979-11-12 |
CA1066701A (en) | 1979-11-20 |
NL186087C (nl) | 1990-09-17 |
PH10529A (en) | 1977-05-30 |
NL186087B (nl) | 1990-04-17 |
NL7401509A (nl) | 1974-10-07 |
AR204660A1 (es) | 1976-02-20 |
AT340931B (de) | 1978-01-10 |
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