AR204003A1 - Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables - Google Patents

Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables

Info

Publication number
AR204003A1
AR204003A1 AR253060A AR25306074A AR204003A1 AR 204003 A1 AR204003 A1 AR 204003A1 AR 253060 A AR253060 A AR 253060A AR 25306074 A AR25306074 A AR 25306074A AR 204003 A1 AR204003 A1 AR 204003A1
Authority
AR
Argentina
Prior art keywords
oxopyride
piperazinyl
pyrimidine
procedure
pharmaceutically acceptable
Prior art date
Application number
AR253060A
Other languages
English (en)
Spanish (es)
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Application granted granted Critical
Publication of AR204003A1 publication Critical patent/AR204003A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR253060A 1973-04-03 1974-01-01 Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables AR204003A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (nl) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (nl) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (nl) 1973-06-07 1973-06-07

Publications (1)

Publication Number Publication Date
AR204003A1 true AR204003A1 (es) 1975-11-12

Family

ID=27289838

Family Applications (2)

Application Number Title Priority Date Filing Date
AR253060A AR204003A1 (es) 1973-04-03 1974-01-01 Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables
AR258571A AR204660A1 (es) 1973-04-03 1975-01-01 Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR258571A AR204660A1 (es) 1973-04-03 1975-01-01 Procedimiento para preparar compuestos derivados del acido 2(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico

Country Status (11)

Country Link
AR (2) AR204003A1 (nl)
AT (1) AT340931B (nl)
CA (1) CA1066701A (nl)
CH (1) CH593281A5 (nl)
ES (1) ES424851A1 (nl)
FI (1) FI56011C (nl)
IE (1) IE39102B1 (nl)
NL (1) NL186087C (nl)
NO (1) NO142221C (nl)
PH (2) PH10529A (nl)
SE (1) SE416051B (nl)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (it) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti.
PL2448938T3 (pl) 2009-06-29 2014-11-28 Incyte Holdings Corp Pirymidynony jako inhibitory PI3K
AR079529A1 (es) 2009-12-18 2012-02-01 Incyte Corp Derivados arilo y heteroarilo sustituidos y fundidos como inhibidores de la pi3k
WO2011075643A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted heteroaryl fused derivatives as pi3k inhibitors
TW201249844A (en) 2010-12-20 2012-12-16 Incyte Corp N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
KR102131612B1 (ko) 2011-09-02 2020-07-08 인사이트 홀딩스 코포레이션 Pi3k 억제제로서 헤테로시클릴아민
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
MA41607B1 (fr) 2015-02-27 2021-01-29 Incyte Corp Sels d'un inhibiteur de pi3k et procédés de préparation de ces sels
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor

Also Published As

Publication number Publication date
SE416051B (sv) 1980-11-24
NO142221B (no) 1980-04-08
NO740349L (no) 1974-10-04
IE39102B1 (en) 1978-08-02
NO142221C (no) 1980-07-16
FI56011B (fi) 1979-07-31
IE39102L (en) 1974-10-03
ES424851A1 (es) 1976-06-01
ATA277774A (de) 1977-05-15
PH10984A (en) 1977-10-18
CH593281A5 (en) 1977-11-30
FI56011C (fi) 1979-11-12
CA1066701A (en) 1979-11-20
NL186087C (nl) 1990-09-17
PH10529A (en) 1977-05-30
NL186087B (nl) 1990-04-17
NL7401509A (nl) 1974-10-07
AR204660A1 (es) 1976-02-20
AT340931B (de) 1978-01-10

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