AR199879A1 - PROCEDURE FOR THE PREPARATION OF 4-AZA-BENZIMIDAZOLES - Google Patents

PROCEDURE FOR THE PREPARATION OF 4-AZA-BENZIMIDAZOLES

Info

Publication number
AR199879A1
AR199879A1 AR243765A AR24376572A AR199879A1 AR 199879 A1 AR199879 A1 AR 199879A1 AR 243765 A AR243765 A AR 243765A AR 24376572 A AR24376572 A AR 24376572A AR 199879 A1 AR199879 A1 AR 199879A1
Authority
AR
Argentina
Prior art keywords
benzimidazoles
aza
procedure
preparation
Prior art date
Application number
AR243765A
Other languages
Spanish (es)
Original Assignee
Degussa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Degussa filed Critical Degussa
Application granted granted Critical
Publication of AR199879A1 publication Critical patent/AR199879A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
AR243765A 1971-08-26 1972-08-28 PROCEDURE FOR THE PREPARATION OF 4-AZA-BENZIMIDAZOLES AR199879A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
AT748871A AT315831B (en) 1971-08-26 1971-08-26 Process for the preparation of new 4-aza-benzimidazole derivatives and their salts

Publications (1)

Publication Number Publication Date
AR199879A1 true AR199879A1 (en) 1974-10-08

Family

ID=3596529

Family Applications (1)

Application Number Title Priority Date Filing Date
AR243765A AR199879A1 (en) 1971-08-26 1972-08-28 PROCEDURE FOR THE PREPARATION OF 4-AZA-BENZIMIDAZOLES

Country Status (19)

Country Link
JP (1) JPS4832898A (en)
AR (1) AR199879A1 (en)
AT (1) AT315831B (en)
AU (1) AU461671B2 (en)
BE (1) BE788065A (en)
BR (1) BR7205845A (en)
CA (1) CA979907A (en)
CH (1) CH592660A5 (en)
DD (1) DD99580A5 (en)
DE (1) DE2241575A1 (en)
ES (1) ES405982A1 (en)
FR (1) FR2150820B1 (en)
GB (1) GB1397645A (en)
HU (1) HU166382B (en)
IL (1) IL40080A (en)
NL (1) NL7211407A (en)
SU (1) SU557758A3 (en)
YU (1) YU34897B (en)
ZA (1) ZA725868B (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1140119A (en) * 1978-04-03 1983-01-25 Joseph Torremans N-heterocyclyl-4-piperidinamines
US4588722A (en) * 1984-01-09 1986-05-13 Janssen Pharmaceutica N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives
US4772600A (en) * 1986-06-09 1988-09-20 A. H. Robins Company, Inc. Fused imidazoheterocyclic compounds and pharmaceutical compositions
US5200407A (en) * 1989-06-29 1993-04-06 Meiji Seika Kaburhiki Kaisha Azole derivatives and anti-ulcerative composition containing same
JP2679745B2 (en) * 1989-06-29 1997-11-19 明治製菓株式会社 Azole derivatives and antiulcer agents containing them as active ingredients
PL191618B1 (en) 1997-09-26 2006-06-30 Zentaris Gmbh Azabenzimidazole-based compounds, pharmaceuticals containing such compounds and the method for their manufacture and application
US8227603B2 (en) 2006-08-01 2012-07-24 Cytokinetics, Inc. Modulating skeletal muscle
US8299248B2 (en) 2006-08-02 2012-10-30 Cytokinetics, Incorporated Certain 1H-imidazo[4,5-b]pyrazin-2(3H)-ones and 1H-imidazo[4,5-b]pyrazin-2-ols and methods for their use
EP2069352B9 (en) 2006-08-02 2017-03-15 Cytokinetics, Inc. Certain chemical entities, compositions and methods
WO2008121333A1 (en) * 2007-03-30 2008-10-09 Cytokinetics, Incorporated Certain chemical entities, compositions and methods
US20140113824A1 (en) 2011-05-10 2014-04-24 Bayer Intellectual Property Gmbh Bicyclic (thio)carbonylamidines
CN109316480A (en) 2011-07-13 2019-02-12 赛特凯恩蒂克公司 Combine ALS therapy
EP3495366A1 (en) * 2011-07-15 2019-06-12 Shionogi & Co., Ltd Azabenzimidazole derivative having ampk-activating activity

Also Published As

Publication number Publication date
HU166382B (en) 1975-03-28
CA979907A (en) 1975-12-16
IL40080A0 (en) 1972-10-29
YU34897B (en) 1980-04-30
ES405982A1 (en) 1975-09-16
DE2241575A1 (en) 1973-03-08
GB1397645A (en) 1975-06-11
DD99580A5 (en) 1973-08-12
JPS4832898A (en) 1973-05-02
AT315831B (en) 1974-06-10
ZA725868B (en) 1973-05-30
BR7205845A (en) 1976-05-04
BR7205845D0 (en) 1973-07-03
CH592660A5 (en) 1977-10-31
FR2150820A1 (en) 1973-04-13
SU557758A3 (en) 1977-05-05
NL7211407A (en) 1973-02-28
FR2150820B1 (en) 1975-10-17
IL40080A (en) 1975-12-31
AU4598172A (en) 1974-02-28
YU204172A (en) 1979-10-31
BE788065A (en) 1973-02-26
AU461671B2 (en) 1975-06-05

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