AR132761A1 - Compuesto inhibidor de la quinasa inducible por sal y composición farmacéutica que lo incluye - Google Patents
Compuesto inhibidor de la quinasa inducible por sal y composición farmacéutica que lo incluyeInfo
- Publication number
- AR132761A1 AR132761A1 ARP240101301A ARP240101301A AR132761A1 AR 132761 A1 AR132761 A1 AR 132761A1 AR P240101301 A ARP240101301 A AR P240101301A AR P240101301 A ARP240101301 A AR P240101301A AR 132761 A1 AR132761 A1 AR 132761A1
- Authority
- AR
- Argentina
- Prior art keywords
- pharmaceutical composition
- salt
- kinase inhibitor
- inhibitor compound
- inducible kinase
- Prior art date
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Classifications
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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- A61K31/4192—1,2,3-Triazoles
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023085585 | 2023-05-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR132761A1 true AR132761A1 (es) | 2025-07-30 |
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| Application Number | Title | Priority Date | Filing Date |
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| ARP240101301A AR132761A1 (es) | 2023-05-24 | 2024-05-23 | Compuesto inhibidor de la quinasa inducible por sal y composición farmacéutica que lo incluye |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20260062387A1 (https=) |
| EP (1) | EP4737443A1 (https=) |
| JP (1) | JPWO2024242169A1 (https=) |
| KR (1) | KR20260015855A (https=) |
| CN (1) | CN121358713A (https=) |
| AR (1) | AR132761A1 (https=) |
| AU (1) | AU2024276075A1 (https=) |
| IL (1) | IL324835A (https=) |
| MX (1) | MX2025013981A (https=) |
| TW (1) | TW202509021A (https=) |
| WO (1) | WO2024242169A1 (https=) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US20240124450A1 (en) * | 2022-09-21 | 2024-04-18 | Pfizer Inc. | Novel SIK Inhibitors |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US7488745B2 (en) | 2004-07-16 | 2009-02-10 | Schering Corporation | Compounds for the treatment of inflammatory disorders |
| WO2013144191A1 (de) | 2012-03-29 | 2013-10-03 | Bayer Intellectual Property Gmbh | Substituierte 2 -amino - 3 - cyanopyridine als inhibitoren des natrium calcium austausches und ihre verwendung bei kardiovaskulären erkrankungen |
| US9688680B2 (en) | 2014-08-04 | 2017-06-27 | Blueprint Medicines Corporation | Compositions useful for treating disorders related to kit |
| EP3717471B1 (en) * | 2017-12-02 | 2022-01-05 | Galapagos NV | Novel compounds and pharmaceutical compositions thereof for the treatment of diseases |
| MA52873A (fr) * | 2018-06-15 | 2021-04-21 | Galapagos Nv | Nouveaux composés et compositions pharmaceutiques associées pour le traitement de maladies |
| CA3112326A1 (en) | 2018-09-12 | 2020-03-19 | Novartis Ag | Antiviral pyridopyrazinedione compounds |
| GB201907616D0 (en) * | 2019-05-29 | 2019-07-10 | Galapagos Nv | Novel compounds and pharmaceutical compositons thereof for the treatment of diseases |
| GB201907558D0 (en) | 2019-05-29 | 2019-07-10 | Galapagos Nv | Novel compounds and pharmaceutical compositions thereof for the treatment of diseases |
| US20240010652A1 (en) | 2020-10-14 | 2024-01-11 | Blueprint Medicines Corporation | Compositions and methods for treating kit- and pdgfra-mediated diseases |
| CN115448881A (zh) | 2021-06-09 | 2022-12-09 | 江苏恒瑞医药股份有限公司 | 杂芳基类化合物、其制备方法及其在医药上的应用 |
| JP7290703B1 (ja) | 2021-11-30 | 2023-06-13 | ハシダ技研工業株式会社 | 樹脂成形品の製造方法 |
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2024
- 2024-05-23 EP EP24811175.9A patent/EP4737443A1/en active Pending
- 2024-05-23 AR ARP240101301A patent/AR132761A1/es unknown
- 2024-05-23 AU AU2024276075A patent/AU2024276075A1/en active Pending
- 2024-05-23 WO PCT/JP2024/018995 patent/WO2024242169A1/ja not_active Ceased
- 2024-05-23 JP JP2025522449A patent/JPWO2024242169A1/ja active Pending
- 2024-05-23 KR KR1020257041596A patent/KR20260015855A/ko active Pending
- 2024-05-23 CN CN202480026705.2A patent/CN121358713A/zh active Pending
- 2024-05-23 TW TW113119171A patent/TW202509021A/zh unknown
- 2024-05-23 IL IL324835A patent/IL324835A/en unknown
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2025
- 2025-11-10 US US19/383,969 patent/US20260062387A1/en active Pending
- 2025-11-21 MX MX2025013981A patent/MX2025013981A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN121358713A (zh) | 2026-01-16 |
| WO2024242169A1 (ja) | 2024-11-28 |
| EP4737443A1 (en) | 2026-05-06 |
| IL324835A (en) | 2026-01-01 |
| KR20260015855A (ko) | 2026-02-03 |
| US20260062387A1 (en) | 2026-03-05 |
| MX2025013981A (es) | 2026-01-07 |
| JPWO2024242169A1 (https=) | 2024-11-28 |
| AU2024276075A1 (en) | 2026-01-22 |
| TW202509021A (zh) | 2025-03-01 |
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