AR127700A1 - Prueba de disolución - Google Patents
Prueba de disoluciónInfo
- Publication number
- AR127700A1 AR127700A1 ARP220103162A ARP220103162A AR127700A1 AR 127700 A1 AR127700 A1 AR 127700A1 AR P220103162 A ARP220103162 A AR P220103162A AR P220103162 A ARP220103162 A AR P220103162A AR 127700 A1 AR127700 A1 AR 127700A1
- Authority
- AR
- Argentina
- Prior art keywords
- samples
- evaluation
- relates
- present
- dissolution test
- Prior art date
Links
- 238000007922 dissolution test Methods 0.000 title 1
- 238000011156 evaluation Methods 0.000 abstract 3
- 238000004090 dissolution Methods 0.000 abstract 2
- YIBOMRUWOWDFLG-ONEGZZNKSA-N rilpivirine Chemical compound CC1=CC(\C=C\C#N)=CC(C)=C1NC1=CC=NC(NC=2C=CC(=CC=2)C#N)=N1 YIBOMRUWOWDFLG-ONEGZZNKSA-N 0.000 abstract 2
- 229960002814 rilpivirine Drugs 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000012736 aqueous medium Substances 0.000 abstract 1
- 238000005259 measurement Methods 0.000 abstract 1
- 239000011859 microparticle Substances 0.000 abstract 1
- 239000002105 nanoparticle Substances 0.000 abstract 1
- 238000003908 quality control method Methods 0.000 abstract 1
- 239000000725 suspension Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Sampling And Sample Adjustment (AREA)
- Dermatology (AREA)
- Physics & Mathematics (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- General Physics & Mathematics (AREA)
- Immunology (AREA)
- Pathology (AREA)
- Food Science & Technology (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
Abstract
La presente invención se refiere a la evaluación de muestras que comprenden rilpivirina o una sal farmacéuticamente aceptable de esta en forma de micro- o nanopartículas, tales como suspensiones, y a la medición de la disolución de la rilpivirina o una sal farmacéuticamente aceptable de esta en un medio acuoso. La presente invención también se refiere a la evaluación del control de calidad de dichas muestras y a la entrega de lotes que comprenden dichas muestras para uso farmacéutico. La presente invención también se refiere a un medio para su uso en la evaluación de la disolución.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US2021/072453 WO2022109555A1 (en) | 2020-11-17 | 2021-11-17 | Treatment or prevention of hiv infection |
US202263342834P | 2022-05-17 | 2022-05-17 | |
EP22173914 | 2022-05-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR127700A1 true AR127700A1 (es) | 2024-02-21 |
Family
ID=84421043
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP220103162A AR127700A1 (es) | 2021-11-17 | 2022-11-16 | Prueba de disolución |
Country Status (7)
Country | Link |
---|---|
KR (1) | KR20240095514A (es) |
AR (1) | AR127700A1 (es) |
AU (1) | AU2022394742A1 (es) |
CA (1) | CA3234763A1 (es) |
IL (1) | IL312784A (es) |
TW (1) | TW202333725A (es) |
WO (1) | WO2023088964A1 (es) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JO3429B1 (ar) | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
MX2009000158A (es) | 2006-06-23 | 2009-01-23 | Tibotec Pharm Ltd | Suspensiones acuosas de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil ]-amino]-2-pirimidinil]-amino]-benzonitrilo. |
-
2022
- 2022-11-16 WO PCT/EP2022/082130 patent/WO2023088964A1/en active Application Filing
- 2022-11-16 TW TW111143802A patent/TW202333725A/zh unknown
- 2022-11-16 KR KR1020247015777A patent/KR20240095514A/ko unknown
- 2022-11-16 AR ARP220103162A patent/AR127700A1/es unknown
- 2022-11-16 CA CA3234763A patent/CA3234763A1/en active Pending
- 2022-11-16 AU AU2022394742A patent/AU2022394742A1/en active Pending
-
2024
- 2024-05-12 IL IL312784A patent/IL312784A/en unknown
Also Published As
Publication number | Publication date |
---|---|
TW202333725A (zh) | 2023-09-01 |
WO2023088964A1 (en) | 2023-05-25 |
CA3234763A1 (en) | 2023-05-25 |
KR20240095514A (ko) | 2024-06-25 |
IL312784A (en) | 2024-07-01 |
AU2022394742A1 (en) | 2024-07-04 |
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