AR099137A2 - FORMULATION FOR DIRECT COMPRESSION AND PROCESS - Google Patents
FORMULATION FOR DIRECT COMPRESSION AND PROCESSInfo
- Publication number
- AR099137A2 AR099137A2 ARP150100149A ARP150100149A AR099137A2 AR 099137 A2 AR099137 A2 AR 099137A2 AR P150100149 A ARP150100149 A AR P150100149A AR P150100149 A ARP150100149 A AR P150100149A AR 099137 A2 AR099137 A2 AR 099137A2
- Authority
- AR
- Argentina
- Prior art keywords
- percent
- dry weight
- pharmaceutically acceptable
- weight
- weight basis
- Prior art date
Links
Landscapes
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Reivindicación 1: Una composición farmacéutica, la cual comprende: (a) del 5 al 60 por ciento en peso, sobre una base de peso seco, de un inhibidor de dipeptidil-peptidasa IV en forma libre o en forma de sal de adición de ácido; (b) del 40 al 95 por ciento en peso, sobre una base de peso seco, de un diluyente farmacéuticamente aceptable; (c) del 0 al 20 por ciento en peso, sobre una base de peso seco, de un desintegrante farmacéuticamente aceptable; (d) del 0.1 al 10 por ciento en peso, sobre una base de peso seco, de un lubricante farmacéuticamente aceptable. Reivindicación 14: Una composición de acuerdo con cualquiera de las reivindicaciones 1 a 12, en donde el inhibidor de dipeptidil-peptidasa IV es 1-[3-hidroxi-adamant-1-il-amino)-acetil]-pirrolidin-2(S)-carbonitrilo.Claim 1: A pharmaceutical composition, which comprises: (a) 5 to 60 percent by weight, on a dry weight basis, of a dipeptidyl peptidase IV inhibitor in free form or in the form of acid addition salt ; (b) from 40 to 95 percent by weight, on a dry weight basis, of a pharmaceutically acceptable diluent; (c) from 0 to 20 percent by weight, on a dry weight basis, of a pharmaceutically acceptable disintegrant; (d) 0.1 to 10 percent by weight, on a dry weight basis, of a pharmaceutically acceptable lubricant. Claim 14: A composition according to any one of claims 1 to 12, wherein the dipeptidyl peptidase IV inhibitor is 1- [3-hydroxy-adamant-1-yl-amino) -acetyl] -pyrrolidin-2 (S ) -carbonitrile.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53770604P | 2004-01-20 | 2004-01-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR099137A2 true AR099137A2 (en) | 2016-06-29 |
Family
ID=39962907
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP150100149A AR099137A2 (en) | 2004-01-20 | 2015-01-20 | FORMULATION FOR DIRECT COMPRESSION AND PROCESS |
Country Status (4)
Country | Link |
---|---|
CN (2) | CN101618216B (en) |
AR (1) | AR099137A2 (en) |
TN (1) | TNSN06223A1 (en) |
ZA (1) | ZA200605513B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104856970B (en) * | 2015-06-23 | 2017-08-25 | 张磊 | A kind of vildagliptin tablet for treating type II diabetes |
CN105233300B (en) * | 2015-11-05 | 2019-10-25 | 北京泰德制药股份有限公司 | A kind of stable vildagliptin composition and preparation method thereof |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3131402A1 (en) * | 1981-08-07 | 1983-02-24 | Kilian & Co GmbH, 5000 Köln | METHOD AND TABLET PRESS FOR THE SUCCESSFUL PRODUCTION OF A VARIETY OF TABLETS OF THE SAME WEIGHT |
DE19823831A1 (en) * | 1998-05-28 | 1999-12-02 | Probiodrug Ges Fuer Arzneim | New pharmaceutical use of isoleucyl thiazolidide and its salts |
FR2822826B1 (en) * | 2001-03-28 | 2003-05-09 | Servier Lab | NOVEL ALPHA-AMINO ACID SULPHONYL DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR2824825B1 (en) * | 2001-05-15 | 2005-05-06 | Servier Lab | NOVEL ALPHA-AMINOACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
JP2005519052A (en) * | 2002-01-11 | 2005-06-30 | アスファルマ リミテッド | Pravastatin pharmaceutical preparation and method of use thereof |
JP2003327532A (en) * | 2002-05-10 | 2003-11-19 | Takeda Chem Ind Ltd | Peptidase inhibitor |
-
2005
- 2005-01-17 CN CN200910164779XA patent/CN101618216B/en active Active
- 2005-01-17 CN CNA2005800056665A patent/CN101262851A/en active Pending
-
2006
- 2006-07-04 ZA ZA200605513A patent/ZA200605513B/en unknown
- 2006-07-19 TN TNP2006000223A patent/TNSN06223A1/en unknown
-
2015
- 2015-01-20 AR ARP150100149A patent/AR099137A2/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CN101262851A (en) | 2008-09-10 |
CN101618216A (en) | 2010-01-06 |
TNSN06223A1 (en) | 2007-12-03 |
CN101618216B (en) | 2012-01-04 |
ZA200605513B (en) | 2007-11-28 |
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