AR099137A2 - FORMULATION FOR DIRECT COMPRESSION AND PROCESS - Google Patents

FORMULATION FOR DIRECT COMPRESSION AND PROCESS

Info

Publication number
AR099137A2
AR099137A2 ARP150100149A ARP150100149A AR099137A2 AR 099137 A2 AR099137 A2 AR 099137A2 AR P150100149 A ARP150100149 A AR P150100149A AR P150100149 A ARP150100149 A AR P150100149A AR 099137 A2 AR099137 A2 AR 099137A2
Authority
AR
Argentina
Prior art keywords
percent
dry weight
pharmaceutically acceptable
weight
weight basis
Prior art date
Application number
ARP150100149A
Other languages
Spanish (es)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39962907&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR099137(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR099137A2 publication Critical patent/AR099137A2/en

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  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Reivindicación 1: Una composición farmacéutica, la cual comprende: (a) del 5 al 60 por ciento en peso, sobre una base de peso seco, de un inhibidor de dipeptidil-peptidasa IV en forma libre o en forma de sal de adición de ácido; (b) del 40 al 95 por ciento en peso, sobre una base de peso seco, de un diluyente farmacéuticamente aceptable; (c) del 0 al 20 por ciento en peso, sobre una base de peso seco, de un desintegrante farmacéuticamente aceptable; (d) del 0.1 al 10 por ciento en peso, sobre una base de peso seco, de un lubricante farmacéuticamente aceptable. Reivindicación 14: Una composición de acuerdo con cualquiera de las reivindicaciones 1 a 12, en donde el inhibidor de dipeptidil-peptidasa IV es 1-[3-hidroxi-adamant-1-il-amino)-acetil]-pirrolidin-2(S)-carbonitrilo.Claim 1: A pharmaceutical composition, which comprises: (a) 5 to 60 percent by weight, on a dry weight basis, of a dipeptidyl peptidase IV inhibitor in free form or in the form of acid addition salt ; (b) from 40 to 95 percent by weight, on a dry weight basis, of a pharmaceutically acceptable diluent; (c) from 0 to 20 percent by weight, on a dry weight basis, of a pharmaceutically acceptable disintegrant; (d) 0.1 to 10 percent by weight, on a dry weight basis, of a pharmaceutically acceptable lubricant. Claim 14: A composition according to any one of claims 1 to 12, wherein the dipeptidyl peptidase IV inhibitor is 1- [3-hydroxy-adamant-1-yl-amino) -acetyl] -pyrrolidin-2 (S ) -carbonitrile.

ARP150100149A 2004-01-20 2015-01-20 FORMULATION FOR DIRECT COMPRESSION AND PROCESS AR099137A2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US53770604P 2004-01-20 2004-01-20

Publications (1)

Publication Number Publication Date
AR099137A2 true AR099137A2 (en) 2016-06-29

Family

ID=39962907

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150100149A AR099137A2 (en) 2004-01-20 2015-01-20 FORMULATION FOR DIRECT COMPRESSION AND PROCESS

Country Status (4)

Country Link
CN (2) CN101618216B (en)
AR (1) AR099137A2 (en)
TN (1) TNSN06223A1 (en)
ZA (1) ZA200605513B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104856970B (en) * 2015-06-23 2017-08-25 张磊 A kind of vildagliptin tablet for treating type II diabetes
CN105233300B (en) * 2015-11-05 2019-10-25 北京泰德制药股份有限公司 A kind of stable vildagliptin composition and preparation method thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3131402A1 (en) * 1981-08-07 1983-02-24 Kilian & Co GmbH, 5000 Köln METHOD AND TABLET PRESS FOR THE SUCCESSFUL PRODUCTION OF A VARIETY OF TABLETS OF THE SAME WEIGHT
DE19823831A1 (en) * 1998-05-28 1999-12-02 Probiodrug Ges Fuer Arzneim New pharmaceutical use of isoleucyl thiazolidide and its salts
FR2822826B1 (en) * 2001-03-28 2003-05-09 Servier Lab NOVEL ALPHA-AMINO ACID SULPHONYL DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
FR2824825B1 (en) * 2001-05-15 2005-05-06 Servier Lab NOVEL ALPHA-AMINOACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
JP2005519052A (en) * 2002-01-11 2005-06-30 アスファルマ リミテッド Pravastatin pharmaceutical preparation and method of use thereof
JP2003327532A (en) * 2002-05-10 2003-11-19 Takeda Chem Ind Ltd Peptidase inhibitor

Also Published As

Publication number Publication date
CN101262851A (en) 2008-09-10
CN101618216A (en) 2010-01-06
TNSN06223A1 (en) 2007-12-03
CN101618216B (en) 2012-01-04
ZA200605513B (en) 2007-11-28

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