AR096433A1 - Método de tratamiento del cáncer y uso - Google Patents

Método de tratamiento del cáncer y uso

Info

Publication number
AR096433A1
AR096433A1 ARP140102081A ARP140102081A AR096433A1 AR 096433 A1 AR096433 A1 AR 096433A1 AR P140102081 A ARP140102081 A AR P140102081A AR P140102081 A ARP140102081 A AR P140102081A AR 096433 A1 AR096433 A1 AR 096433A1
Authority
AR
Argentina
Prior art keywords
cancer treatment
human
trioxo
pyrido
phenylamino
Prior art date
Application number
ARP140102081A
Other languages
English (en)
Inventor
Michael Richards Eric
R Hamid Mohammed
Behbahani Roya
R W Streit Michael
A Patel Kiran
Ouellet Daniele
Ann Rogan Debra
Original Assignee
Glaxosmithkline Intellectual Property (No 2) Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Intellectual Property (No 2) Ltd filed Critical Glaxosmithkline Intellectual Property (No 2) Ltd
Publication of AR096433A1 publication Critical patent/AR096433A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Reivindicación 1: Un método para tratar el cáncer en un ser humano que lo necesite, que comprende la administración in vivo de una cantidad terapéuticamente eficaz de un compuesto seleccionado de N-{3-[3-ciclopropil-5-(2-fluoro-4-yodo-fenilamino)-6,8-dimetil-2,4,7-trioxo-3,4,6,7-tetrahidro-2H-pirido[4,3-d]pirimidin-1-iI]fenil}acetamida, o una de sus sales o solvatos farmacéuticamente aceptables, a dicho ser humano.
ARP140102081A 2013-05-28 2014-05-26 Método de tratamiento del cáncer y uso AR096433A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361827940P 2013-05-28 2013-05-28

Publications (1)

Publication Number Publication Date
AR096433A1 true AR096433A1 (es) 2015-12-30

Family

ID=50884976

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP140102081A AR096433A1 (es) 2013-05-28 2014-05-26 Método de tratamiento del cáncer y uso

Country Status (4)

Country Link
AR (1) AR096433A1 (es)
TW (1) TW201536292A (es)
UY (1) UY35587A (es)
WO (1) WO2014191920A1 (es)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7378423B2 (en) 2004-06-11 2008-05-27 Japan Tobacco Inc. Pyrimidine compound and medical use thereof
RS50569B (sr) 2004-06-11 2010-05-07 Japan Tobacco Inc. Derivati 5-amino-2,4,7-triokso-3,4,7,8-tetrahidro-2h-pirido (2,3-d)pirimidina i slična jedinjenja za lečenje raka

Also Published As

Publication number Publication date
TW201536292A (zh) 2015-10-01
WO2014191920A1 (en) 2014-12-04
UY35587A (es) 2014-12-31

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