AR092170A1 - Proceso para la fabricacion de benzoxazinonas - Google Patents
Proceso para la fabricacion de benzoxazinonasInfo
- Publication number
- AR092170A1 AR092170A1 ARP130102936A ARP130102936A AR092170A1 AR 092170 A1 AR092170 A1 AR 092170A1 AR P130102936 A ARP130102936 A AR P130102936A AR P130102936 A ARP130102936 A AR P130102936A AR 092170 A1 AR092170 A1 AR 092170A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- haloalkyl
- aryl
- formula
- alkoxy
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 9
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 5
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 3
- 125000003118 aryl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 2
- 125000006642 (C1-C6) cyanoalkyl group Chemical group 0.000 abstract 2
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 2
- 125000006570 (C5-C6) heteroaryl group Chemical group 0.000 abstract 2
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical compound O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 2
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- ORTFAQDWJHRMNX-UHFFFAOYSA-N hydroxidooxidocarbon(.) Chemical group O[C]=O ORTFAQDWJHRMNX-UHFFFAOYSA-N 0.000 abstract 2
- 125000004971 nitroalkyl group Chemical group 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- HQQTZCPKNZVLFF-UHFFFAOYSA-N 4h-1,2-benzoxazin-3-one Chemical class C1=CC=C2ONC(=O)CC2=C1 HQQTZCPKNZVLFF-UHFFFAOYSA-N 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 150000004657 carbamic acid derivatives Chemical class 0.000 abstract 1
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 1
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C335/04—Derivatives of thiourea
- C07C335/24—Derivatives of thiourea containing any of the groups, X being a hetero atom, Y being any atom
- C07C335/28—Y being a hetero atom, e.g. thiobiuret
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Reivindicación 1: Un proceso para la fabricación de benzoxazinonas caracterizado por la fórmula (1) en donde R¹ es H, halógeno o alquilo C₁₋₆; R² es H, halógeno o alquilo C₁₋₆; R³ es H, halógeno o alquilo C₁₋₆; R⁴ es H, alquilo C₁₋₆, haloalquilo C₁₋₆, cicloalquilo C₃₋₆, alquenilo C₃₋₆, haloalquenilo C₃₋₆, alquinilo C₃₋₆, haloalquinilo C₃₋₆, alcoxi C₁₋₆ o cicloalquil C₃₋₆-alquilo C₁₋₆; R⁵ es H o alquilo C₁₋₆; R⁶ es H o alquilo C₁₋₆; W es O ó S; y Z es O ó S; en donde los carbamatos de la fórmula (2), en donde R⁵ y R⁶ se definen como en la fórmula (1); y R⁷ es alquilo C₁₋₆, haloalquilo C₁₋₆, cianoalquilo C₁₋₆, nitroalquilo C₁₋₆, arilo, heteroarilo 5 ó 6 miembros o aril-alquilo C₁₋₆; en donde los anillos de arilo o heteroarilo son no sustituidos, parcial o totalmente halogenados, o sustituidos con 1 a 5 sustituyentes seleccionados del grupo que consiste en CN, NO₂, alquilo C₁₋₆, haloalquilo C₁₋₆, OH, alcoxi C₁₋₆, haloalcoxi C₁₋₆, formilo, alquilcarbonilo C₁₋₆, hidroxicarbonilo y alcoxicarbonilo C₁₋₆; se hacen reaccionar con carbamat-benzoxazinonas de la fórmula (3), en donde R¹, R², R³, R⁴ y W son como se definen en la fórmula (1); y R⁸ es haloalquilo C₁₋₆, cianoalquilo C₁₋₆, nitroalquilo C₁₋₆, arilo, heteroarilo de 5 ó 6 miembros o aril-alquilo C₁₋₆, en donde los anillos de arilo o heteroarilo son no sustituidos, parcial o totalmente halogenados, o sustituidos con 1 a 5 sustituyentes seleccionados del grupo que consiste en CN, NO₂, alquilo C₁₋₆, haloalquilo C₁₋₆, OH, alcoxi C₁₋₆, haloalcoxi C₁₋₆, formilo, alquilcarbonilo C₁₋₆, hidroxicarbonilo y alcoxicarbonilo C₁₋₆; en presencia de una base.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12180843 | 2012-08-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR092170A1 true AR092170A1 (es) | 2015-03-25 |
Family
ID=46940228
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP130102936A AR092170A1 (es) | 2012-08-17 | 2013-08-16 | Proceso para la fabricacion de benzoxazinonas |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US9518045B2 (es) |
| EP (1) | EP2885296B1 (es) |
| JP (1) | JP6273278B2 (es) |
| CN (1) | CN104583205B (es) |
| AR (1) | AR092170A1 (es) |
| AU (1) | AU2013304167B2 (es) |
| BR (1) | BR112015002912B1 (es) |
| CA (1) | CA2881026C (es) |
| DK (1) | DK2885296T3 (es) |
| EA (1) | EA029143B1 (es) |
| ES (1) | ES2594553T3 (es) |
| IL (1) | IL237027A (es) |
| MX (1) | MX349214B (es) |
| WO (1) | WO2014026928A1 (es) |
| ZA (1) | ZA201501764B (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2014026845A1 (en) | 2012-08-17 | 2014-02-20 | Basf Se | Carbamates |
| BR112016014018B8 (pt) | 2013-12-18 | 2021-10-26 | Basf Agro Bv | Processo para a preparação dos compostos de cetona (ia), e processo para a preparação dos compostos de triazol de fórmula (ic) |
| EP3131906B1 (en) | 2014-04-17 | 2018-06-13 | Basf Se | Substituted pyridine compounds having herbicidal activity |
| MX377942B (es) | 2014-07-08 | 2025-03-11 | Basf Agro Bv | Proceso para la preparacion de oxiranos y triazoles. |
| WO2016057931A1 (en) | 2014-10-10 | 2016-04-14 | The Research Foundation For The State University Of New York | Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration |
| CN107848922A (zh) | 2015-05-08 | 2018-03-27 | 巴斯夫农业公司 | 柠檬烯‑4‑醇的制备方法 |
| EP3294720B1 (en) | 2015-05-08 | 2020-12-02 | BASF Agro B.V. | A process for the preparation of terpinolene epoxide |
| EP3184515A1 (en) * | 2015-12-22 | 2017-06-28 | Basf Se | Process for manufacturing 1,4-benzoxazinones |
| ES2877169T3 (es) | 2016-06-15 | 2021-11-16 | Basf Agro Bv | Procedimiento para la epoxidación de un alqueno tetrasustituido |
| BR112018076043B1 (pt) | 2016-06-15 | 2023-09-26 | Basf Agro B.V | Processo de epoxidação de alqueno tetrassubstituído e uso de agente oxidante |
| WO2021088856A1 (zh) * | 2019-11-07 | 2021-05-14 | 青岛清原化合物有限公司 | 一种含取代异恶唑啉的芳香类化合物及其制备方法、除草组合物和应用 |
| CN111689922B (zh) * | 2020-07-17 | 2022-03-15 | 江西施美药业股份有限公司 | 一种苯磺酸左旋氨氯地平环合杂质的合成方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3392184A (en) | 1965-08-05 | 1968-07-09 | Upjohn Co | Allophanates and thiolallophanates |
| US3372180A (en) | 1965-10-22 | 1968-03-05 | Upjohn Co | Process for the production of hydrocarbyl 2, 4-dihydrocarbyl allophanates and thiolallophanates |
| DE3023675A1 (de) | 1980-06-25 | 1982-01-14 | Bayer Ag, 5090 Leverkusen | N-acylierte n-methyl-o-pyrazol(4)yl-carbaminsaeureester, verfahren zu ihrer herstellung und ihre verwendung in schaedlingsbekaempfungsmitteln |
| DE3106724A1 (de) * | 1981-02-24 | 1982-09-09 | Bayer Ag, 5090 Leverkusen | "verfahren zur herstellung von 1-amino-1,3,5-triazin-2,4 (1h, 3h)-dionen" |
| DE3145327A1 (de) * | 1981-11-14 | 1983-05-26 | Basf Ag, 6700 Ludwigshafen | Verfahren zur herstellung von n,n'-disubstituierten allophansaeureestern |
| DE3516632A1 (de) * | 1985-05-09 | 1986-11-13 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von 1,3,5-triazintrionen |
| JP2007533673A (ja) * | 2004-04-20 | 2007-11-22 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | バニロイド受容体（ｖｒ１）のアンタゴニストとしての尿素誘導体 |
| CL2008001003A1 (es) * | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
| BRPI1010081B8 (pt) * | 2009-06-19 | 2017-06-27 | Basf Se | benzoxazinonas, processo para preparar benzoxazinonas de fórmula i, compostos, acetamidas, composições herbicidas, composição para a dessecação/desfolhação de plantas, processos para preparar composições, método para controlar vegetação indesejada, método para a dessecação/desfolhação de plantas e uso das benzoxazinonas de fórmula i |
| DK2499136T3 (en) * | 2009-11-13 | 2014-03-03 | Basf Se | 3- (3,4-dihydro-2H-benzo [1,4] oxazin-6-yl) -1H-pyrimidine-2,4-dione COMPOUNDS AS HERBICIDES |
| EP2794599A1 (en) | 2011-12-23 | 2014-10-29 | Basf Se | Process for manufacturing triazinon-benzoxazinones |
| WO2014026845A1 (en) | 2012-08-17 | 2014-02-20 | Basf Se | Carbamates |
-
2013
- 2013-08-09 CN CN201380043755.3A patent/CN104583205B/zh active Active
- 2013-08-09 ES ES13747408.6T patent/ES2594553T3/es active Active
- 2013-08-09 BR BR112015002912A patent/BR112015002912B1/pt active IP Right Grant
- 2013-08-09 WO PCT/EP2013/066719 patent/WO2014026928A1/en not_active Ceased
- 2013-08-09 US US14/421,351 patent/US9518045B2/en active Active
- 2013-08-09 AU AU2013304167A patent/AU2013304167B2/en active Active
- 2013-08-09 MX MX2015002111A patent/MX349214B/es active IP Right Grant
- 2013-08-09 JP JP2015526945A patent/JP6273278B2/ja active Active
- 2013-08-09 EA EA201500234A patent/EA029143B1/ru not_active IP Right Cessation
- 2013-08-09 EP EP13747408.6A patent/EP2885296B1/en active Active
- 2013-08-09 CA CA2881026A patent/CA2881026C/en active Active
- 2013-08-09 DK DK13747408.6T patent/DK2885296T3/en active
- 2013-08-16 AR ARP130102936A patent/AR092170A1/es active IP Right Grant
-
2015
- 2015-02-01 IL IL237027A patent/IL237027A/en active IP Right Grant
- 2015-03-16 ZA ZA2015/01764A patent/ZA201501764B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2015002111A (es) | 2015-05-11 |
| EA201500234A1 (ru) | 2015-09-30 |
| US9518045B2 (en) | 2016-12-13 |
| CN104583205A (zh) | 2015-04-29 |
| CA2881026A1 (en) | 2014-02-20 |
| CA2881026C (en) | 2021-04-13 |
| JP6273278B2 (ja) | 2018-01-31 |
| AU2013304167A1 (en) | 2015-02-26 |
| DK2885296T3 (en) | 2016-10-03 |
| BR112015002912A2 (pt) | 2017-07-04 |
| MX349214B (es) | 2017-07-18 |
| EP2885296A1 (en) | 2015-06-24 |
| IL237027A (en) | 2016-12-29 |
| CN104583205B (zh) | 2017-03-08 |
| AU2013304167B2 (en) | 2017-09-07 |
| EP2885296B1 (en) | 2016-06-29 |
| ZA201501764B (en) | 2017-01-25 |
| BR112015002912B1 (pt) | 2020-02-04 |
| JP2015526437A (ja) | 2015-09-10 |
| US20150218140A1 (en) | 2015-08-06 |
| ES2594553T3 (es) | 2016-12-21 |
| WO2014026928A1 (en) | 2014-02-20 |
| EA029143B1 (ru) | 2018-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |