AR076494A1 - Arilpirrolidinas plaguicidas - Google Patents

Arilpirrolidinas plaguicidas

Info

Publication number
AR076494A1
AR076494A1 ARP100101449A ARP100101449A AR076494A1 AR 076494 A1 AR076494 A1 AR 076494A1 AR P100101449 A ARP100101449 A AR P100101449A AR P100101449 A ARP100101449 A AR P100101449A AR 076494 A1 AR076494 A1 AR 076494A1
Authority
AR
Argentina
Prior art keywords
alkyl
haloalkyl
cyano
represents hydrogen
alkylcarbonyl
Prior art date
Application number
ARP100101449A
Other languages
English (en)
Inventor
Kei Domon
Tetsuya Murata
Yasushi Yoneta
Koichi Araki
Norio Sasaki
Mamoru Hatazawa
Ulrico Gorgens
Katsuhiko Shibuya
Eiichi Shimojo
Teruyuki Ichihara
Masashi Ataka
Jun Mihara
Daiei Yamazaki
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2009111390A external-priority patent/JP2010116389A/ja
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of AR076494A1 publication Critical patent/AR076494A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se refiere a compuestos de arilpirrolidina que muestran una eficacia insecticida excelente y que pueden usarse tanto en el campo agroquímico como en el campo de la medicina veterinaria. Reivindicacion 1: Compuestos arilpirrolidina de formula (1) en la que: R representa alquilo C1-12 o haloalquilo C1-12 opcionalmente sustituido: Q representa un grupo seleccionado entre los grupos Q-1 a Q-12 en los que W1 representa un enlace sencillo o metileno (es decir, un grupo -CH2-), pudiendo estar dicho grupo opcionalmente sustituido con al menos un sustituyente Y1, mientras que el sustituyente está conectado preferentemente a un átomo de carbono; B1, B2, B3 y B4, cada uno independientemente, representa C-X2 o nitrogeno, y si cualquiera de B1 y B2, o B2 y B3, o B3 y B4 representa C-X2, entonces los sustituyentes X2 pueden formar, junto con los átomos de carbono a los que están unidos, un anillo heterocíclico o un anillo hidrocarburo de 5 o 6 miembros, saturado o insaturado; X1, X2, cada uno independientemente, representa hidrogeno, halogeno, nitro, ciano, hidroxilo, mercapto, amino, alquilo, haloalquilo, alcoxi, haloalcoxi, alquilsulfanilo, alquilsulfinilo, alquilsulfonilo, haloalquilsulfanilo, haloalquilsulfinilo, haloalquilsulfonilo. acilamino, alcoxicarbonilamino, haloalcoxicarbonilamino, alcoxiimino, haloalcoxiimino, alquilsulfonilamino o pentafluorosulfuro; Y1 representa cada uno independientemente hidrogeno, halogeno, nitro, ciano, hidroxilo, mercapto, amino, alquilo, haloalquilo, cicloalquilo, ciclohaloalquilo, alquenilo, alquinilo, alcoxi, haloalcoxi, alquilsulfanilo, alquilsulfinilo, alquilsulfonilo, haloalquiIsuIfanilo, haloalquilsuIfinilo, haloaIquiIsuIfonilo, alquiIsuIfoniloxi, haloalquilsulfoniloxi, alquilaminosulfonilo, haloalquilaminosulfonilo, dialquilaminosulfonilo, di(haloalquil)aminosulfonilo, alquilamino, dialquilamino, acilamino, alcoxicarbonilamino, haloalcoxicarbonilamino, alquilsulfonilamino, haloalquilsulfonilamino, trialquilsililo, alcoxiimino, haloalcoxiimino, alcoxiiminoalquilo, haloalcoxiiminoalquilo, alquilsulfinilimino, alquilsulfiniliminoalquilo, alquilsulfiniliminoalquilcarbonilo, alquilsulfoxiimino, alquilsulfoxiiminoalquilo, alcoxicarbonilo, alquilcarbonilo, aminocarbonilo, alquilaminocarbonilo, aminotiocarbonilo, alquilaminotiocarbonilo, dialquilaminocarbonilo o dialquilaminotiocarbonilo; R3 representa hidrogeno, ciano, alquilo, alquenilo, alquinilo, cicloalquilo o alcoxicarbonilo; R5 representa hidrogeno, amino, hidroxilo, ciano, alquilo, haloalquilo, cicloalquilo, alquenilo, alquinilo, alcoxi, aminocarbonilalquilo, iminoalquilo, alquilcarbonilo, alquilcarbonilamino, alquilimino, arilo, aralquilo, un heterociclo, alquilo sustituido con un anillo heterocíclico, R7-C(=O)- o R7-C(=S)-; R6 representa hidrogeno, ciano, carbonilo, tiocarbonilo, alquilcarbonilo, alquiltiocarbonilo, haloalquilcarbonilo, haloalquiltiocarbonilo, alquilaminocarbonilo, alquilaminotiocarbonilo, dialquilaminocarbonilo, dialquilaminotiocarbonilo, alcoxiaminocarbonilo, alcoxiaminotiocarbonilo, alcoxicarbonilo, alcoxitiocarbonilo, alquilsulfanilcarbonilo, alquilsulfaniltiocarbonilo, alquilsulfonilo, haloalquilsulfonilo, cicloalquilcarbonilo, alquenilcarbonilo, alquinilcarbonilo, cicloalquilalquilcarbonilo, alquilsulfanilalquilcarbonilo, alquilsulfinilalquilcarbonilo, alquilsulfonilalquilcarbonilo, alquilcarbonilalquilcarbonilo, cicloalquilaminocarbonilo, alquenilaminocarbonilo, alquinilaminocarbonilo, alquilaminosulfonilo, dialquilaminosulfonilo, alcoxialquilcarbonilo, alquilcarbonilaminoalquilcarbonilo, haloalquilcarbonilaminoalquilcarbonilo, alquilsulfanilalquilcarbonilaminoalquilcarbonilo, alquilsulfinilalquilcarbonilaminoalquilcarbonilo, alquilsulfonilalquilcarbonilaminoalquilcarbonilo, aralquilcarbonilo, alquilcarbonilo heterocíclicamente sustituido, R7-C(=O) o R7-C(S)-, o R5 y R6 pueden formar un anillo heterocíclico de 3 a 6 miembros, junto con el átomo de nitrogeno al que están unidos, y dicho anillo puede estar sustituido con ceto, tioceto o un grupo nitroimino o R7 representa un fenilo opcionalmente sustituido o un heterociclo opcionalmente sustituido.
ARP100101449A 2009-04-30 2010-04-29 Arilpirrolidinas plaguicidas AR076494A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2009111390A JP2010116389A (ja) 2008-10-17 2009-04-30 殺虫性アリールピロリジン類

Publications (1)

Publication Number Publication Date
AR076494A1 true AR076494A1 (es) 2011-06-15

Family

ID=42227127

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100101449A AR076494A1 (es) 2009-04-30 2010-04-29 Arilpirrolidinas plaguicidas

Country Status (7)

Country Link
US (1) US20120129854A1 (es)
EP (1) EP2424838A1 (es)
CN (1) CN102414175A (es)
AR (1) AR076494A1 (es)
BR (1) BRPI1014641A2 (es)
TW (1) TW201103903A (es)
WO (1) WO2010124845A1 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5508400B2 (ja) * 2008-06-05 2014-05-28 グラクソ グループ リミテッド Ｐｉ３キナーゼの阻害剤としてのベンズピラゾール誘導体
EP2280705B1 (en) 2008-06-05 2014-10-08 Glaxo Group Limited Novel compounds
US8765743B2 (en) * 2008-06-05 2014-07-01 Glaxosmithkline Intellectual Property Development Limited Compounds
JP5656880B2 (ja) 2009-03-09 2015-01-21 グラクソ グループ リミテッドＧｌａｘｏ Ｇｒｏｕｐ Ｌｉｍｉｔｅｄ Ｐｉ３キナーゼの阻害剤としての４−オキサジアゾール−２−イル−インダゾール
MA33304B1 (fr) * 2009-04-30 2012-05-02 Glaxo Group Ltd Indazoles substitués par oxazole comme inhibiteurs de pi3-kinase
TWI487486B (zh) 2009-12-01 2015-06-11 Syngenta Participations Ag 以異唑啉衍生物為主之殺蟲化合物
JP2011136928A (ja) 2009-12-28 2011-07-14 Bayer Cropscience Ag 殺虫性アリールピロリジン類
GB201018124D0 (en) 2010-10-27 2010-12-08 Glaxo Group Ltd Polymorphs and salts
BR112015006825A2 (pt) 2012-09-27 2017-08-08 Bayer Cropscience Ag processo para a preparação de fenil e piridil pirrolidinas opcionalmente substituídas.
US11034669B2 (en) 2018-11-30 2021-06-15 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10205862A1 (de) * 2002-02-13 2003-08-21 Bayer Cropscience Ag DELTA1-Pyrroline
WO2006101828A1 (en) * 2005-03-15 2006-09-28 Bayer Cropscience Ag Insecticidal alkylamino phenyl sulfonamide derivatives
BRPI0707091B8 (pt) * 2006-03-10 2018-02-14 Nissan Chemical Ind Ltd composto de isoxalina e benzaldoxima substituído ou um sal do mesmo; pesticida, agroquímico, endo- ou ecto-parasiticidapara mamíferos ou pássaros, inseticida e acaricida contendo como um ou mais ingredientes ativos selecionados a partir do composto de isoxalina substituído e o sal do mesmo
JP5164510B2 (ja) * 2006-10-06 2013-03-21 日本曹達株式会社 含窒素複素環化合物および有害生物防除剤
JP2010116389A (ja) * 2008-10-17 2010-05-27 Bayer Cropscience Ag 殺虫性アリールピロリジン類
JP2008266230A (ja) * 2007-04-23 2008-11-06 Bayer Cropscience Ag 殺虫性アリールピロリジン類

Also Published As

Publication number Publication date
EP2424838A1 (en) 2012-03-07
TW201103903A (en) 2011-02-01
US20120129854A1 (en) 2012-05-24
BRPI1014641A2 (pt) 2019-09-24
WO2010124845A1 (en) 2010-11-04
CN102414175A (zh) 2012-04-11

Similar Documents

Publication Publication Date Title
AR076494A1 (es) Arilpirrolidinas plaguicidas
AR073764A1 (es) Arilpirrolidinas plaguicidas
AR070582A1 (es) Arilpirrolinas insecticidas y procedimiento para prepararlos
AR071644A1 (es) Plaguicidas mesoionicos
CO6231032A2 (es) Dderivados de aril isoxazolina insecticidas
AR066144A1 (es) Derivados de aril pirrolidinas utiles como insecticidas y/o acaricidas y composiciones insecticidas que los contienen.
AR116978A1 (es) Fungicidas de tolilo sustituido
AR104202A1 (es) Derivados heterocíclicos bicíclicos condensados como pesticidas
AR107397A1 (es) Derivados de heterociclos bicíclicos condensados como pesticidas
AR109677A1 (es) Derivados heterocíclicos bicíclicos fusionados como plaguicidas
AR106165A1 (es) Derivados heterocíclicos condensados sustituidos por 2-(het)arilo como pesticidas
AR114330A1 (es) Derivados de heterociclos bicíclicos condensados como pesticidas
TW200602056A (en) Substituted 2-quinolyl-oxazoles useful as PDE4 inhibitors
AR071769A1 (es) Azoles sustituidos como fungicidas, una composicion fungicida que comprende el compuesto y un metodo para controlar enfermedades de las plantas
PE20090151A1 (es) Derivados de pirimidinona y metodos para su uso
AR069368A1 (es) Mezclas fungicidas
AR057688A1 (es) CARBOXAMIDAS HETEROCíCLICAS Y SU USO EN COMPOSICIONES FUNGICIDAS.
ES2531256T3 (es) Amidas fungicidas
AR081653A1 (es) Inhibidores del virus de la hepatitis c
AR070866A1 (es) Compuestos pesticidas de arilo de anillo condensado
AR072576A1 (es) Metodo para la represion de malezas en un cesped
RU2010107171A (ru) Фунгицидные n-циклоалкилбензилтиокарбоксамиды или n-циклоалкилбензил-n, -замещенные амидиновые производные
AR070680A1 (es) Derivados herbicidas de piridazinona
AR105322A1 (es) Heterociclos nitrogenados como pesticidas
JP2012522056A5 (es)

Legal Events

Date Code Title Description
FB Suspension of granting procedure