AR071471A1 - Derivados de imidazol, procedimientos para su obtencion, una composicion fungicida que lo comprende, un metodo para el control de la infestacion de cultivos y su uso en la preparacion de un medicamento para el tratamiento del cancer. - Google Patents

Derivados de imidazol, procedimientos para su obtencion, una composicion fungicida que lo comprende, un metodo para el control de la infestacion de cultivos y su uso en la preparacion de un medicamento para el tratamiento del cancer.

Info

Publication number
AR071471A1
AR071471A1 ARP090101293A ARP090101293A AR071471A1 AR 071471 A1 AR071471 A1 AR 071471A1 AR P090101293 A ARP090101293 A AR P090101293A AR P090101293 A ARP090101293 A AR P090101293A AR 071471 A1 AR071471 A1 AR 071471A1
Authority
AR
Argentina
Prior art keywords
halogen
cancer
obtaining
preparation
treatment
Prior art date
Application number
ARP090101293A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR071471A1 publication Critical patent/AR071471A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/68—Halogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/60—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Derivados de imidazol de la formula (1) como ingredientes activos, que tienen actividad microbicida, en particular, actividad fungicida, donde R1 es halogeno, alquilo C1-4 o haloalquilo C1-4; R2 es un arilo opcionalmente sustituido; R3 es halogeno u OR7; R4 y R5 son, de manera independiente entre sí, hidrogeno, halogeno u OR7; R6 es halogeno o alquilo C1-4; y R7 es hidrogeno, alquilo C1-6, cicloalquilo C3-7, cicloalquilalquilo C3-10, haloalquilo C1-6, alquenilo C2-6, haloalquenilo C2-6, cicloalquenilo C3-7, alquinilo C2-6, haloalquinilo C2-6, alquiloxialquilo C2-6, dialquilaminoalquilo C3-8, cicloalquilaminoalquilo C4-10 o heterociclilalquilo C4-10; o una forma de sal agroquímicamente utilizable de dichos compuestos; siempre que: cuando R3 es halogeno, por lo menos uno de R4 o R5 es OR7; o cuando R3 es OR7, por lo menos uno de R4 o R5 es OR7 o halogeno. Métodos para su obtencion y su uso en métodos de control de infestacion de cultivos y en la preparacion de un medicamento para el tratamiento del cáncer.
ARP090101293A 2008-04-14 2009-04-13 Derivados de imidazol, procedimientos para su obtencion, una composicion fungicida que lo comprende, un metodo para el control de la infestacion de cultivos y su uso en la preparacion de un medicamento para el tratamiento del cancer. AR071471A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0806745.6A GB0806745D0 (en) 2008-04-14 2008-04-14 Novel imidazole derivatives

Publications (1)

Publication Number Publication Date
AR071471A1 true AR071471A1 (es) 2010-06-23

Family

ID=39433609

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090101293A AR071471A1 (es) 2008-04-14 2009-04-13 Derivados de imidazol, procedimientos para su obtencion, una composicion fungicida que lo comprende, un metodo para el control de la infestacion de cultivos y su uso en la preparacion de un medicamento para el tratamiento del cancer.

Country Status (6)

Country Link
EP (1) EP2279176A1 (es)
AR (1) AR071471A1 (es)
CL (1) CL2009000885A1 (es)
GB (1) GB0806745D0 (es)
TW (1) TW201002203A (es)
WO (1) WO2009127615A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201117722A (en) * 2009-11-04 2011-06-01 Du Pont Fungicidal mixtures
CN103153962A (zh) 2010-09-29 2013-06-12 纳幕尔杜邦公司 杀真菌咪唑
EP2841070B1 (en) 2012-04-24 2018-07-25 Board Of Trustees Of Northern Illinois University Design and synthesis of novel inhibitors of isoprenoid biosynthesis
US10155766B2 (en) 2016-06-14 2018-12-18 Board Of Trustees Of Northern Illinois University Pyrazolopyrimidine antibacterial agents
CN109810062B (zh) * 2019-01-24 2022-06-17 云南农业大学 一种苯基咪唑衍生物及其合成方法和在农药中的应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5223525A (en) * 1989-05-05 1993-06-29 Rhone-Poulenc Ag Company Pesticidal 1-arylimidazoles
EP0712847A4 (en) * 1993-08-11 1997-05-28 Nippon Soda Co IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION AND USE THEREOF AS A PEST CONTROL
AR024222A1 (es) * 1998-10-16 2002-09-25 Palau Pharma Sa Imidazoles con actividad antiinflamatoria un procedimiento para su preparacion y composiciones farmaceuticas que lo contienen
JP2001163861A (ja) * 1999-12-07 2001-06-19 Nippon Soda Co Ltd ジフェニルイミダゾール化合物および農園芸用殺菌剤
AU2003293376A1 (en) * 2002-12-10 2004-06-30 Imclone Systems Incorporated Anti-angiogenic compounds and their use in cancer treatment
EP2053044A1 (en) * 2007-10-26 2009-04-29 Syngenta Participations AG Novel imidazole derivatives

Also Published As

Publication number Publication date
GB0806745D0 (en) 2008-05-14
EP2279176A1 (en) 2011-02-02
WO2009127615A1 (en) 2009-10-22
CL2009000885A1 (es) 2009-10-09
TW201002203A (en) 2010-01-16

Similar Documents

Publication Publication Date Title
IL284913A (en) A multispecific antigen-binding molecule that has the function-changing activity of a cofactor for blood coagulation factor viii (fviii), and a pharmaceutical formulation containing the molecule as an active ingredient
CY1124519T1 (el) ΣΤΕΡΕΕΣ ΜΟΡΦΕΣ ΚΑΙ ΦΑΡΜΑΚΟΤΕΧΝΙΚΕΣ ΜΟΡΦΕΣ ΤΟΥ (S)-4-(8-ΑΜΙΝΟ-3-(1-(ΒΟΥΤ-2-ΥΝΟΫΛΟ)ΠΥΡΡΟΛΙΔΙΝ-2-ΥΛΟ) ΙΜΙΔΑΖΟ[1,5-α|ΠΥΡΑΖΙΝ-1-ΥΛΟ)-Ν-(ΠΥΡΙΔΙΝ-2-ΥΛΟ) ΒΕΝΖΑΜΙΔΙΟΥ
DK201470535A (en) Parasiticidal oral veterinary compositions comprising systemically-acting active agents, methods and uses thereof
NI201700011A (es) 2-(morfolin-4-il)-1,7-naftiridinas.
RU2017127135A (ru) Терапевтическое средство против рака желчных протоков
MX2015016416A (es) Derivados de la pirazolopirrolidina y su uso en el tratamiento de enfermedades.
EA201790094A1 (ru) Пестицидные композиции, содержащие изоксазолиновый активный ингредиент, и способы их применения
EA201591662A1 (ru) Липиды и липидные композиции для доставки активных агентов
CR20110270A (es) Piriloxi-indoles Inhibidores del VEGF-R2 y Uso de los Mismos para el Tratamiento de Enfermedades
CO6351786A2 (es) Inkibidores de la cinasa map p38
EA201201371A1 (ru) Паразитицидные композиции, содержащие несколько активных агентов, способы и их применения
EA201300869A1 (ru) Морфинановые соединения
EA201390541A1 (ru) Эмульсионные композиции клевидипина, содержащие противомикробные агенты
AR071471A1 (es) Derivados de imidazol, procedimientos para su obtencion, una composicion fungicida que lo comprende, un metodo para el control de la infestacion de cultivos y su uso en la preparacion de un medicamento para el tratamiento del cancer.
PH12014502366A1 (en) Injectable formulation
EA201291167A1 (ru) Замещенные гетероциклилбензилпиразолы и их применение
BR112014011981A8 (pt) Formulações farmacêuticas sólidas orais, seus processos de preparação e usos
ECSP099382A (es) Sulfonamidas heterocíclicos que tienen actividad antagonista edg-i
CL2013001390A1 (es) 1-[6-(morfolin-4-il)pirimidin-4-il]-4-(1h-1,2,3-triazol-1-il)-1h-pirazol-5-olato sodico; procedimiento de preparacion; composicion farmaceutica y uso en el tratamiento y/o profilaxis de enfermedades tales como insuficiencia cardiaca, anemia, insuficiencia renal y enf. cardiovasculares.
BR112012005194A2 (pt) uso de éteres de glicerol como agentes de ativação de efeitos biológicos de ao menos uma substância herbicida, fungicida ou inseticida , composição fitossanitária e processo de tratamento fitossanitário
CY1120727T1 (el) Συνδυασμοι με ενα πεπτιδιο κυκλοποιημενου σκελετου
AR071657A1 (es) DERIVADOS DE PIRAZOL, PROCEDIMIENTOS PARA SU OBTENCIoN Y LA DE SUS INTERMEDIARIOS DE S¡NTESIS, UNA COMPOSICIoN FUNGICIDA QUE LO COMPRENDE, UN MITODO PARA EL CONTROL DE LA INFESTACIoN DE CULTIVOS Y SU USO EN LA PREPARACIoN DE UN MEDICAMENTO PARA EL TRATAMIENTO DEL CµNCER
RU2010150718A (ru) Способ предпосевной обработки семян
ATE524180T1 (de) Mittel zur prophylaxe oder behandlung von alkoholabhängigkeit oder drogenabhängigkeit
GEP20125640B (en) Phenanthrenone compounds, compositions containing them and use thereof

Legal Events

Date Code Title Description
FB Suspension of granting procedure