AR065471A1 - Proceso para la preparacion de ciertas sulfiliminas sustituidas - Google Patents
Proceso para la preparacion de ciertas sulfiliminas sustituidasInfo
- Publication number
- AR065471A1 AR065471A1 ARP080100777A ARP080100777A AR065471A1 AR 065471 A1 AR065471 A1 AR 065471A1 AR P080100777 A ARP080100777 A AR P080100777A AR P080100777 A ARP080100777 A AR P080100777A AR 065471 A1 AR065471 A1 AR 065471A1
- Authority
- AR
- Argentina
- Prior art keywords
- haloalkenyl
- haloalkyl
- alkynyl
- alkenyl
- integer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/32—Sulfur atoms
- C07D213/34—Sulfur atoms to which a second hetero atom is attached
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se producen cianosulfiliminas sustituidas a partir de los correspondientes sulfuros, por reaccion con cianamida e hipoclorito. Reivindicacion 1: Un proceso para preparar sulfiliminas de la formula (1), en donde Het representa grupo de formulas (2),X representa halogeno, alquilo C1-4, haloalquilo C1-4, alquenilo C2-4, alquinilo C2-4, haloalquenilo C2-4, alcoxi C1-4, haloalcoxi C1-4, CN, NO2, SOmR6 en donde m es un entero entre 0-2, COOR4 o CONR4R5; Y representa hidrogeno, halogeno, alquilo C1-4, haloalquilo, C1-4, alquenilo C2-4, alquinilo C2-4, haloalquenilo C2-4, alcoxi C1-4, haloalcoxi C1-4, CN, NO2, SOmR1 en donde m es un entero entre 0-2, COOR4, CONR4R5, arilo o heteroarilo; n es un entero entre 0-3; L representa un enlace simple, -CH(CH2)p- en donde R1, S y L tomados juntos representan un anillo de 4, 5 o 6 miembros y p es un entero entre 1-3, -CH(CH2OCH2)- en donde R1, S y L tomados juntos representan un anillo de 6 miembros, o -CH- en donde L, R2 y el carbono comun al queestán conectados tomados juntos representan un anillo de 4, 5 o 6 miembros con hasta, pero no más de 1 heteroátomo; R1 representa alquilo C1-4, haloalquilo C1-4, alquenilo C3-6, alquinilo C3-6, haloalquenilo C3-6, arilalquilo, heteroarilalquilo, o -CH2- en los casos de que R1, S y L tomados juntos representan un anillo de 4, 5 o 6 miembros; R2 y R3 representan independientemente hidrogeno, halogeno, alquilo C1-4, haloalquilo C1-4, alquenilo C2-4, alquinilo C2-4, haloalquenilo C2-4, alcoxi C1-4, haloalcoxi C1-4, CN, SOmR6 en donde m es un entero entre 0-2, COOR4, CONR4R5, arilalquilo, heteroarilalquilo, o R2 y R3 y el anillo comun al que se unen forma un anillo de 3 a 6 miembros; R4 y R5 representan independientemente hidrogeno, alquiloC1-4, haloalquilo C1-4; alquenilo C3-6, alquinilo C3-6, haloalquenilo C3-6, arilo, heteroarilo, arilalquilo o heteroarilalquilo; y R6 representa alquilo C1-4, haloalquilo C1-4; alquenilo C3-6, alquinilo C3-6, haloalquenilo C3-6, arilalquilo oheteroarilalquilo; que comprende poner en contacto un solfuro de la formula (3) en donde R1, R2, R3, L, Het y n son como se definio con anterioridad con cianamida y solucion de hipoclorito a una temperatura de aproximadamente -40°C a aproximadamente30°C en un solvente orgánico adecuado que es esencialmente inerte en las condiciones de reaccion.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US90347107P | 2007-02-26 | 2007-02-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065471A1 true AR065471A1 (es) | 2009-06-10 |
Family
ID=39523499
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100777A AR065471A1 (es) | 2007-02-26 | 2008-02-25 | Proceso para la preparacion de ciertas sulfiliminas sustituidas |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US7868027B2 (es) |
| EP (1) | EP2114886B1 (es) |
| JP (1) | JP5302221B2 (es) |
| KR (1) | KR101437710B1 (es) |
| CN (1) | CN101641331B (es) |
| AR (1) | AR065471A1 (es) |
| AU (1) | AU2008219748B2 (es) |
| BR (1) | BRPI0807702B8 (es) |
| CA (1) | CA2678028C (es) |
| CL (1) | CL2008000564A1 (es) |
| DK (1) | DK2114886T3 (es) |
| HK (1) | HK1141013A1 (es) |
| IL (1) | IL200520A (es) |
| TW (1) | TWI393706B (es) |
| WO (1) | WO2008106006A1 (es) |
| ZA (1) | ZA200905012B (es) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8193222B1 (en) | 2007-02-26 | 2012-06-05 | Dow AgroSciences, L.L.C. | Process for the preparation of certain substituted sulfilimines |
| WO2010074747A1 (en) | 2008-12-26 | 2010-07-01 | Dow Agrosciences, Llc | Stable insecticide compositions and methods for producing same |
| RU2518251C2 (ru) * | 2008-12-26 | 2014-06-10 | ДАУ АГРОСАЙЕНСИЗ, ЭлЭлСи | Стабильная пестицидная композиция на основе сульфоксимина и способ борьбы с насекомыми |
| WO2010075966A1 (de) * | 2008-12-29 | 2010-07-08 | Bayer Cropscience Ag | Verfahren zur verbesserten nutzung des produktionspotentials genetisch modifizierter pflanzen |
| EP2223602A1 (de) | 2009-02-23 | 2010-09-01 | Bayer CropScience AG | Verfahren zur verbesserten Nutzung des Produktionspotentials genetisch modifizierter Pflanzen |
| EP2223598A1 (de) | 2009-02-23 | 2010-09-01 | Bayer CropScience AG | Insektizide Zusammensetzungen mit verbesserter Wirkung |
| US20110306643A1 (en) | 2010-04-23 | 2011-12-15 | Bayer Cropscience Ag | Triglyceride-containing dormancy sprays |
| EP2545964A1 (en) | 2011-07-13 | 2013-01-16 | Phenex Pharmaceuticals AG | Novel FXR (NR1H4) binding and activity modulating compounds |
| BR102013003576B8 (pt) * | 2012-02-16 | 2022-10-11 | Dow Agrosciences Llc | Método para produzir n-ciano-s-metil-s-[1-(6-tri-flúormetil-3-piridinil)etil]sulfilimina |
| US9156784B2 (en) | 2012-02-21 | 2015-10-13 | Bayer Intellectual Property Gmbh | Herbicidal sulfinimidoyl- and sulfonimidoyl benzoyl derivatives |
| WO2013124228A1 (de) | 2012-02-21 | 2013-08-29 | Bayer Intellectual Property Gmbh | Herbizid wirksame 3 - ( sulfin- /sulfonimidoyl) - benzamide |
| CN104602527B (zh) | 2012-06-30 | 2018-09-25 | 美国陶氏益农公司 | 吡啶n-氧化物及其制备方法 |
| KR102089479B1 (ko) | 2012-06-30 | 2020-03-17 | 다우 아그로사이언시즈 엘엘씨 | N-치환된 술폭시민 피리딘 n-옥시드의 제조 |
| CN105324365A (zh) * | 2012-12-11 | 2016-02-10 | 美国陶氏益农公司 | 用于制备n-氰基-s-[1-(吡啶-3-基)乙基]-s-甲基硫亚胺的改善方法 |
| EP2873668A1 (en) | 2013-11-13 | 2015-05-20 | Syngenta Participations AG. | Pesticidally active bicyclic heterocycles with sulphur containing substituents |
| EP3356343B1 (en) | 2015-09-28 | 2020-03-18 | Syngenta Participations AG | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| ES2921432T3 (es) | 2016-06-13 | 2022-08-25 | Gilead Sciences Inc | Derivados de azetidina como moduladores de FXR (NR1H4) |
| CA2968836A1 (en) | 2016-06-13 | 2017-12-13 | Gilead Sciences, Inc. | Fxr (nr1h4) modulating compounds |
| TWI735573B (zh) * | 2016-06-21 | 2021-08-11 | 美商陶氏農業科學公司 | 生產某些經取代硫亞胺之方法 |
| CA3030946A1 (en) | 2016-07-22 | 2018-01-25 | Sumitomo Chemical Company, Limited | Herbicide composition including [3-[2-chloro-4-fluoro-5-(1-methyl-6-trifluoromethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2-pyridyloxy]acetate and 2,4-d choline salt and method for controlling weeds |
| JP7282031B2 (ja) | 2016-12-01 | 2023-05-26 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
| ES2927019T3 (es) | 2017-03-28 | 2022-11-02 | Gilead Sciences Inc | Combinaciones terapéuticas para el tratamiento de enfermedades hepáticas |
| JP7309615B2 (ja) | 2017-05-02 | 2023-07-18 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な複素環式誘導体 |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CN112262140B (zh) | 2018-06-06 | 2024-05-28 | 先正达农作物保护股份公司 | 具有含亚砜亚胺取代基的杀有害生物活性杂环衍生物 |
| AR115495A1 (es) | 2018-06-06 | 2021-01-27 | Syngenta Crop Protection Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| DK3911647T3 (da) | 2019-01-15 | 2024-02-26 | Gilead Sciences Inc | Isoxazol-forbindelse som FXR-agonist og farmaceutiske sammensætninger, der omfatter en sådan |
| CN113439078B (zh) | 2019-02-19 | 2024-04-23 | 吉利德科学公司 | Fxr激动剂的固体形式 |
| MX2023006990A (es) | 2020-12-14 | 2023-06-26 | Basf Se | Plaguicidas de sulfoximina. |
| CA3221102A1 (en) | 2021-06-02 | 2022-12-08 | Michel Muehlebach | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7678920B2 (en) | 2004-04-08 | 2010-03-16 | Dow Agrosciences Llc | Insecticidal N-substituted sulfoximines |
| TWI398433B (zh) * | 2006-02-10 | 2013-06-11 | Dow Agrosciences Llc | 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺 |
-
2008
- 2008-02-12 CA CA2678028A patent/CA2678028C/en not_active Expired - Fee Related
- 2008-02-12 AU AU2008219748A patent/AU2008219748B2/en active Active
- 2008-02-12 CN CN2008800045382A patent/CN101641331B/zh active Active
- 2008-02-12 EP EP08725445.4A patent/EP2114886B1/en active Active
- 2008-02-12 JP JP2009550885A patent/JP5302221B2/ja active Active
- 2008-02-12 US US12/069,627 patent/US7868027B2/en active Active
- 2008-02-12 BR BRPI0807702A patent/BRPI0807702B8/pt active IP Right Grant
- 2008-02-12 DK DK08725445.4T patent/DK2114886T3/da active
- 2008-02-12 KR KR1020097017664A patent/KR101437710B1/ko active IP Right Grant
- 2008-02-12 ZA ZA200905012A patent/ZA200905012B/xx unknown
- 2008-02-12 WO PCT/US2008/001818 patent/WO2008106006A1/en active Application Filing
- 2008-02-21 TW TW097106047A patent/TWI393706B/zh not_active IP Right Cessation
- 2008-02-25 AR ARP080100777A patent/AR065471A1/es active IP Right Grant
- 2008-02-25 CL CL200800564A patent/CL2008000564A1/es unknown
-
2009
- 2009-08-20 IL IL200520A patent/IL200520A/en active IP Right Grant
-
2010
- 2010-07-31 HK HK10107320.4A patent/HK1141013A1/xx not_active IP Right Cessation
- 2010-11-18 US US12/949,213 patent/US20110077409A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0807702A2 (pt) | 2014-05-27 |
| JP5302221B2 (ja) | 2013-10-02 |
| WO2008106006A1 (en) | 2008-09-04 |
| DK2114886T3 (da) | 2014-06-30 |
| IL200520A0 (en) | 2010-04-29 |
| AU2008219748A1 (en) | 2008-09-04 |
| EP2114886B1 (en) | 2014-03-26 |
| TW200844097A (en) | 2008-11-16 |
| CL2008000564A1 (es) | 2008-08-29 |
| KR20090113870A (ko) | 2009-11-02 |
| AU2008219748B2 (en) | 2012-05-03 |
| CA2678028A1 (en) | 2008-09-04 |
| EP2114886A1 (en) | 2009-11-11 |
| US7868027B2 (en) | 2011-01-11 |
| TWI393706B (zh) | 2013-04-21 |
| IL200520A (en) | 2014-02-27 |
| CA2678028C (en) | 2015-02-03 |
| HK1141013A1 (en) | 2010-10-29 |
| KR101437710B1 (ko) | 2014-09-03 |
| US20080207910A1 (en) | 2008-08-28 |
| CN101641331A (zh) | 2010-02-03 |
| ZA200905012B (en) | 2010-10-27 |
| CN101641331B (zh) | 2012-06-27 |
| US20110077409A1 (en) | 2011-03-31 |
| BRPI0807702B1 (pt) | 2016-11-01 |
| BRPI0807702B8 (pt) | 2022-06-28 |
| JP2010519296A (ja) | 2010-06-03 |
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Legal Events
| Date | Code | Title | Description |
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| FG | Grant, registration |