AR054554A1 - COMPOUNDS OF 7- AMINO-6- TRIAZOLIL-1,2,4-TRIAZOLO (1,5-A) PYRIMIDINE AND ITS USE FOR THE COMBAT OF DANINE FUNGES - Google Patents

COMPOUNDS OF 7- AMINO-6- TRIAZOLIL-1,2,4-TRIAZOLO (1,5-A) PYRIMIDINE AND ITS USE FOR THE COMBAT OF DANINE FUNGES

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Publication number
AR054554A1
AR054554A1 ARP060103001A ARP060103001A AR054554A1 AR 054554 A1 AR054554 A1 AR 054554A1 AR P060103001 A ARP060103001 A AR P060103001A AR P060103001 A ARP060103001 A AR P060103001A AR 054554 A1 AR054554 A1 AR 054554A1
Authority
AR
Argentina
Prior art keywords
alkyl
alkynyl
alkenyl
partially
radicals
Prior art date
Application number
ARP060103001A
Other languages
Spanish (es)
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of AR054554A1 publication Critical patent/AR054554A1/en

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

Compuestos de 7-amino-6-triazolil-1,2,4-triazolo[1,5-a]pirimidina de la formula (1) y sus sales de tolerancia en agricultura, así como a su uso para el combate de hongos daninos, así como a agentes fitopatogenos que contienen por lo menos un compuesto de este tipo como componente eficaz. Reivindicacion 1: 7-amino-6-triazolil-1,2,4-triazolo[1,5-a]pirimidina caracterizada porque tiene la formula general (1) en donde los sustituyentes Het, R1, R2, X e Y presentan los siguientes significados: Het es 1 ,2,3-triazolilo o 1 ,2,4-triazolilo, en donde Het presenta dos sustituyentes L iguales o diferentes; R1 es hidrogeno, alquilo C1-8, cicloalquilo C3-8, bicicloalquilo C5-10, alquenilo C2-8, alcadienilo C4-10, cicloalquenilo C3- 8, alquinilo C2-8, fenilo, naftilo, o un heterociclo saturado, parcialmente insaturado o aromático de cinco o seis miembros, que contiene uno, dos, tres o cuatro heteroátomos del grupo O, N o S; R2 son los sustituyentes mencionados en R1, así como además alcoxi G1-8, cicloalcoxi C3-8, alquenil C2-8-oxi, alquinil C2-8-oxi, amino, R1 y R2 también pueden formar junto con el átomo de nitrogeno al que están unidos un heterociclo saturado, parcialmente insaturado o aromático de cinco o seis miembros, que puede contener como miembro del anillo uno, dos o tres heteroátomos más del grupo O, N y S; R1 y/o R2 o el heterociclo formado por R1 y R2 pueden estar sustituidos en si; X es hidrogeno, hidroxi, halogeno, ciano, NH2, NR3R4, en donde R3 y R4 presentan, de modo independiente entre si, los significados indicados para R1 o R2; o es alquilo C1-8, alcoxi C1-8, alquil C1-8-tio, alquil C1-8-sulfinilo, alquil C1-8-sulfonilo, alquenilo C2-8, alquinilo C2-8, alcoxi C1-4-alquilo C1-4 o ciano-alquilo C1-4, en donde estos radicales pueden estar parcial o totalmente halogenados; Y es hidrogeno, halogeno, ciano; o alquilo C1-8, cicloalquilo C3-6, alcoxi C1-8, alquil C1-8-tio, alquil C1-8-sulfinilo, alquil C1-8-sulfonilo, alquenilo C2- 8 o alquinilo C2-8, en donde estos radicales pueden estar parcial o totalmente halogenados; L es hidrogeno; o siempre que L sea el sustituyente de un nitrogeno de anillo de Het C(=O)A2, C(=S)A2; o alquilo C1-8, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-8, cicloalquenilo C3-8, alcoximino C1-8-alquilo, alquenil C2-8- oximinoalquilo, alquinil C2-8-oximinoalquilo, en donde estos radicales pueden estar parcial o totalmente halogenados; o, siempre que L sea sustituyente de un carbono del anillo de Het, los compuestos mencionados en el caso de la sustitucion de un nitrogeno de anillo de Het, así como además halogeno, ciano, hidroxi, nitro, NR5R6, NR5-(C=O)-R6, S(=O)nA1, o alcoxi C1-8 alquenil C2-C8-oxi, alquinil C2-8-oxi, cicloalcoxi C3-8, en donde estos radicales pueden estar parcial o totalmente halogenados; y donde A1 es alquilo C1-6, alquil C1-6-amino o di-(alquil C1-6) amino, en donde estos radicales pueden estar parcial o totalmente halogenados; n es 0,1 o 2; A2 es uno de los grupos mencionados en A1; o alquenilo C2-8, alquinilo C2-8, alcoxi C1-6, alquenil C2-8-oxi, alquinil C2-8-oxi, cicloalcoxi C3-8, en donde estos radicales pueden estar parcial o totalmente halogenados; R5, R6 son, de modo independiente entre si, hidrogeno; o alquilo C1-6, alquenilo C2-8, alquinilo C2-8, cicloalquilo C3-8 o cicloalquenilo C3-8, en donde estos radicales pueden estar parcial o totalmente halogenados; y sus sales de tolerancia en agricultura.Compounds of 7-amino-6-triazolyl-1,2,4-triazolo [1,5-a] pyrimidine of the formula (1) and its tolerance salts in agriculture, as well as its use for combating harmful fungi , as well as to phytopathogenic agents that contain at least one such compound as an effective component. Claim 1: 7-amino-6-triazolyl-1,2,4-triazolo [1,5-a] pyrimidine characterized in that it has the general formula (1) wherein the substituents Het, R1, R2, X and Y present the following meanings: Het is 1, 2,3-triazolyl or 1, 2,4-triazolyl, wherein Het has two identical or different L substituents; R 1 is hydrogen, C 1-8 alkyl, C 3-8 cycloalkyl, C 5-10 bicycloalkyl, C 2-8 alkenyl, C 4-10 alkynyl, C 3-8 cycloalkenyl, C 2-8 alkynyl, phenyl, naphthyl, or a saturated, partially unsaturated heterocycle or aromatic of five or six members, which contains one, two, three or four heteroatoms of the group O, N or S; R2 are the substituents mentioned in R1, as well as in addition G1-8 alkoxy, C3-8 cycloalkoxy, C2-8-oxy alkenyl, C2-8-oxy alkynyl, amino, R1 and R2 may also form together with the nitrogen atom at that a saturated, partially unsaturated or aromatic heterocycle of five or six members is attached, which may contain as a member of the ring one, two or three more heteroatoms of the group O, N and S; R1 and / or R2 or the heterocycle formed by R1 and R2 may be substituted per se; X is hydrogen, hydroxy, halogen, cyano, NH2, NR3R4, where R3 and R4 have, independently of each other, the meanings indicated for R1 or R2; or is C1-8 alkyl, C1-8 alkoxy, C1-8-thio alkyl, C1-8 alkyl sulfinyl, C1-8 alkyl sulfonyl, C2-8 alkenyl, C2-8 alkynyl, C1-4 alkoxy-C1 alkyl -4 or cyano-C1-4 alkyl, wherein these radicals may be partially or totally halogenated; And it is hydrogen, halogen, cyano; or C1-8 alkyl, C3-6 cycloalkyl, C1-8 alkoxy, C1-8-thio alkyl, C1-8-sulfinyl alkyl, C1-8-sulfonyl alkyl, C2-8 alkenyl or C2-8 alkynyl, wherein these radicals can be partially or totally halogenated; L is hydrogen; or whenever L is the substituent of a ring nitrogen of Het C (= O) A2, C (= S) A2; or C 1-8 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 3-8 cycloalkyl, C 3-8 cycloalkenyl, C 1-8 alkoxy alkyl, C 2-8 alkynyl alkynyl, C 2-8 alkynyl alkynyl alkyl, wherein these radicals can be partially or totally halogenated; or, provided that L is a Het ring carbon substituent, the compounds mentioned in the case of the replacement of a Het ring nitrogen, as well as halogen, cyano, hydroxy, nitro, NR5R6, NR5- (C = O) -R6, S (= O) nA1, or C1-8 alkoxyC2-C8-oxy alkenyl, C2-8-oxy alkynyl, C3-8 cycloalkoxy, wherein these radicals may be partially or totally halogenated; and where A1 is C1-6 alkyl, C1-6-amino alkyl or di- (C1-6 alkyl) amino, wherein these radicals may be partially or totally halogenated; n is 0.1 or 2; A2 is one of the groups mentioned in A1; or C2-8 alkenyl, C2-8 alkynyl, C1-6 alkoxy, C2-8-oxy alkenyl, C2-8-oxy alkynyl, C3-8 cycloalkoxy, wherein these radicals may be partially or totally halogenated; R5, R6 are, independently of each other, hydrogen; or C 1-6 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 3-8 cycloalkyl or C 3-8 cycloalkenyl, wherein these radicals may be partially or totally halogenated; and its tolerance salts in agriculture.

ARP060103001A 2005-07-13 2006-07-12 COMPOUNDS OF 7- AMINO-6- TRIAZOLIL-1,2,4-TRIAZOLO (1,5-A) PYRIMIDINE AND ITS USE FOR THE COMBAT OF DANINE FUNGES AR054554A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005033160 2005-07-13

Publications (1)

Publication Number Publication Date
AR054554A1 true AR054554A1 (en) 2007-06-27

Family

ID=36945617

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103001A AR054554A1 (en) 2005-07-13 2006-07-12 COMPOUNDS OF 7- AMINO-6- TRIAZOLIL-1,2,4-TRIAZOLO (1,5-A) PYRIMIDINE AND ITS USE FOR THE COMBAT OF DANINE FUNGES

Country Status (5)

Country Link
AR (1) AR054554A1 (en)
PE (1) PE20070424A1 (en)
TW (1) TW200740821A (en)
UY (1) UY29669A1 (en)
WO (1) WO2007023018A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007101870A1 (en) * 2006-03-08 2007-09-13 Basf Se Substituted triazolopyrimidines, methods for the production thereof and use thereof for controlling parasitic fungi and agents containing the latter
WO2009102761A1 (en) 2008-02-12 2009-08-20 Bristol-Myers Squibb Company 1,2,3-triazoles as 11-beta hydroxysteroid dehydrogenase type i inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1115926B (en) * 1977-03-30 1986-02-10 Minnesota Mining & Mfg MAGENTA 5-PYRAZOLONIC COPULANTS FOR PHOTOGRAPHIC USE PHOTOGRAPHIC ELEMENTS THAT CONTAIN THEM AND PROCEDURE FOR THEIR PRODUCTION
JPH04164084A (en) * 1990-10-26 1992-06-09 Hokko Chem Ind Co Ltd Triazole derivative and agricultural and horticultural germicide
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
DE10328481A1 (en) * 2003-06-25 2005-01-13 Bayer Ag triazolopyrimidines
MXPA05013579A (en) * 2003-06-27 2006-03-09 Warner Lambert Co Preparation of n2-alkylated 1,2,3-triazoles.

Also Published As

Publication number Publication date
TW200740821A (en) 2007-11-01
PE20070424A1 (en) 2007-04-27
UY29669A1 (en) 2007-02-28
WO2007023018A1 (en) 2007-03-01

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