AR053046A1 - Cristal de derivado de aminonopirrolidina y metodo de produccion del mismo - Google Patents

Cristal de derivado de aminonopirrolidina y metodo de produccion del mismo

Info

Publication number
AR053046A1
AR053046A1 ARP060101363A ARP060101363A AR053046A1 AR 053046 A1 AR053046 A1 AR 053046A1 AR P060101363 A ARP060101363 A AR P060101363A AR P060101363 A ARP060101363 A AR P060101363A AR 053046 A1 AR053046 A1 AR 053046A1
Authority
AR
Argentina
Prior art keywords
crystal
aminonopirrolidine
derivative
same
production method
Prior art date
Application number
ARP060101363A
Other languages
English (en)
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36607292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR053046(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of AR053046A1 publication Critical patent/AR053046A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Reivindicacion 2: Un cristal (R)-3-[2-(2-amino-5-trifluormetoxibenzamido)acetamida]-1-(6-metilindol-3-ilmetil)pirrolidina (cristal A) que exhibe un patron de difraccion de polvo de rayos X que tiene picos característicos expresados en el ángulo de reflexion 20(grado) en aproximadamente 5,7; 8,4; 15,2; 16,9; 19,7; 20,9; 21,3; 21,7 y 24,1. Reivindicacion 4: Un cristal de (R)-3-[2-(2-amino-5-trifluormetoxibenzamido) acetamido]-1-(6-metilindol-3-ilmetil)pirrolidina (cristal B) que . exhibe un patron de difraccion de polvo de rayos X que tiene picos característicos expresados en el ángulo de reflexion 20 (grado) en aproximadamente 9,6; 11,3; 15,5; 16,3; 19,3; 20,0; 20,5; 20,9; 22,7; 23,3; 24,2; 27,2; 27,8 y 31,6. Su forma amorfa, una composicion farmacéutica que contiene el cristal o la forma amorfa como un ingrediente activo, así como también métodos para su preparacion.
ARP060101363A 2005-04-07 2006-04-06 Cristal de derivado de aminonopirrolidina y metodo de produccion del mismo AR053046A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005110854 2005-04-07

Publications (1)

Publication Number Publication Date
AR053046A1 true AR053046A1 (es) 2007-04-18

Family

ID=36607292

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060101363A AR053046A1 (es) 2005-04-07 2006-04-06 Cristal de derivado de aminonopirrolidina y metodo de produccion del mismo

Country Status (13)

Country Link
US (1) US20090076120A1 (es)
EP (1) EP1871767A1 (es)
JP (1) JP2008534436A (es)
KR (1) KR20070116863A (es)
CN (1) CN101155802A (es)
AR (1) AR053046A1 (es)
AU (1) AU2006234545A1 (es)
BR (1) BRPI0609739A2 (es)
CA (1) CA2608078A1 (es)
PE (1) PE20061375A1 (es)
RU (1) RU2007141206A (es)
TW (1) TW200708512A (es)
WO (1) WO2006109836A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102898380A (zh) * 2007-06-21 2013-01-30 艾克提麦斯医药品有限公司 一种crth2 拮抗剂的胺盐
CN102119139A (zh) 2008-08-07 2011-07-06 杏林制药株式会社 二环[2.2.2]辛胺衍生物的制造方法
JPWO2010032723A1 (ja) * 2008-09-16 2012-02-09 杏林製薬株式会社 アミノアセチルピロリジンカルボニトリル誘導体の精製方法およびその塩
TW201016675A (en) * 2008-09-16 2010-05-01 Mitsubishi Tanabe Pharma Corp Crystalline benzoimidazole compound and salt thereof
TWI646091B (zh) 2012-12-28 2019-01-01 日商衛斯克慧特股份有限公司 鹽類及晶形
GB201420285D0 (en) * 2014-11-14 2014-12-31 Bergenbio As Process

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2373942A1 (en) * 1999-05-18 2000-11-23 Teijin Limited Remedies or prophylactis for diseases in association with chemokines
WO2005035493A1 (ja) * 2003-10-08 2005-04-21 Teijin Pharma Limited アミノピロリジン誘導体の製造方法および中間体化合物
JP2005112787A (ja) * 2003-10-08 2005-04-28 Teijin Pharma Ltd アミノピロリジン誘導体の製造法
EP1760075A4 (en) * 2004-06-14 2009-10-28 Teijin Pharma Ltd PROCESS FOR PRODUCING AN ACETAMIDOPYRROLIDINE DERIVATIVE AND AN INTERMEDIATE COMPOUND THEREOF

Also Published As

Publication number Publication date
WO2006109836A1 (en) 2006-10-19
TW200708512A (en) 2007-03-01
US20090076120A1 (en) 2009-03-19
EP1871767A1 (en) 2008-01-02
CA2608078A1 (en) 2006-10-19
JP2008534436A (ja) 2008-08-28
CN101155802A (zh) 2008-04-02
KR20070116863A (ko) 2007-12-11
RU2007141206A (ru) 2009-05-20
BRPI0609739A2 (pt) 2011-10-18
PE20061375A1 (es) 2007-01-23
AU2006234545A1 (en) 2006-10-19

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Legal Events

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